Journal
ORGANIC LETTERS
Volume 19, Issue 20, Pages 5649-5652Publisher
AMER CHEMICAL SOC
DOI: 10.1021/acs.orglett.7b02788
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Funding
- National Natural Science Foundation of China [21672089, 21472080]
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Based upon a radical polar effect, an intermolecular azidoheteroarylation of simple alkenes via a metal-free radical multi component cascade process was achieved. It allows a mild, rapid, and step economic access to a broad range of azidoalkylated heteroaromatics. Given the diversity in transformations of organic azides and medicinally privileged scaffolds of heteroarenes, this strategy enables efficient synthesis and late stage derivatization of drugs and candidates.
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