Journal
ORGANIC LETTERS
Volume 19, Issue 23, Pages 6272-6275Publisher
AMER CHEMICAL SOC
DOI: 10.1021/acs.orglett.7b02784
Keywords
-
Categories
Funding
- European Research Council [ERC-337776]
- MINECO [CTQ2016-78779-R]
- National Science Foundation [1151092, 1543699]
- Division Of Chemistry
- Direct For Mathematical & Physical Scien [1151092] Funding Source: National Science Foundation
Ask authors/readers for more resources
In this report, the enantioselective, copper-catalyzed borylation of beta-amidoacrylates is disclosed. A broad variety of biologically important alpha-aminoboronates has been prepared with consistently high levels of enantiocontrol using an inexpensive copper catalyst and a commercially available chiral ligand. The method can be applied to the synthesis of novel boron-containing dipeptides and hemiboronates.
Authors
I am an author on this paper
Click your name to claim this paper and add it to your profile.
Reviews
Recommended
No Data Available