Journal
ORGANIC LETTERS
Volume 19, Issue 19, Pages 5134-5137Publisher
AMER CHEMICAL SOC
DOI: 10.1021/acs.orglett.7b02425
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Funding
- Shenzhen Peacock Plan [KQTD2015071714043444]
- NSFC [21272011, 21572007]
- SZSTDF [JCYJ20140419131807793, JCYJ20130329175740481, JCYJ20160527100424909, ZDSYS201504301539161]
- GDNSF [2014A030312004, 2014B030301003]
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A one-pot regio- and stereospecific strategy for the construction of 3a-(3-indolyl)-hexahydropyrrolo[2,3-b]indoles based on the condensation of an indole and an in situ generated cyclopropylazetoindoline has been developed. This unified strategy works with a variety of substituted indoles to produce 3a-(3-indolyl)-hexahydropyrrolo[2,3-b]indole products in high yields. The utility of this transformation was highlighted in the formal total syntheses of gliocladins B and C.
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