Journal
ORGANIC LETTERS
Volume 19, Issue 6, Pages 1314-1317Publisher
AMER CHEMICAL SOC
DOI: 10.1021/acs.orglett.7b00358
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- Duke University
- National Institute of General Medical Sciences of the National Institutes of Health [GM118786]
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Selective C-H amidation of 1H-indoles at the C3 position is reported as a direct entry to biologically important 3-aminoindoles. This transformation is achieved using novel N-[(benzenesulfonyl)oxy]amides as electrophilic nitrogen agents in the presence of ZnCl2. Interestingly, analogous reactions in the absence of ZnCl2 resulted in the formation of indole aminal products.
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