Journal
ORGANIC & BIOMOLECULAR CHEMISTRY
Volume 15, Issue 24, Pages 5112-5116Publisher
ROYAL SOC CHEMISTRY
DOI: 10.1039/c7ob01135k
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Funding
- National Natural Science Foundation of China [21572149]
- Major Basic Research Project of the Natural Science Foundation of the Jiangsu Higher Education Institutions [15KJA150006]
- Young National Natural Science Foundation of China [21403148]
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With the assistance of the same bidentate directing group, the first example of sequential, controllable C-H functionalization of beta-arylethylamines at different positions for the construction of polysubstituted arenes is reported. Pd-Catalyzed highly regio-selective ortho-C-H functionalization reactions of meta-aryl substituted arylethylamines are performed, including alkynylation, iodination, acetoxylation and amination, which led to a concise approach to the synthesis of polysubstituted beta-arylethylamine derivatives.
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