4.8 Article

Intrinsic BET inhibitor resistance in SPOP-mutated prostate cancer is mediated by BET protein stabilization and AKT-mTORC1 activation

Related references

Note: Only part of the references are listed.
Article Oncology

TRIM24 Is an Oncogenic Transcriptional Activator in Prostate Cancer

Anna C. Groner et al.

CANCER CELL (2016)

Article Biochemical Research Methods

Organoid culture systems for prostate epithelial and cancer tissue

Jarno Drost et al.

NATURE PROTOCOLS (2016)

Article Biochemistry & Molecular Biology

The Molecular Taxonomy of Primary Prostate Cancer

Adam Abeshouse et al.

Article Biochemistry & Molecular Biology

Hijacking the E3 Ubiquitin Ligase Cereblon to Efficiently Target BRD4

Jing Lu et al.

CHEMISTRY & BIOLOGY (2015)

Article Multidisciplinary Sciences

Transcriptional plasticity promotes primary and acquired resistance to BET inhibition

Philipp Rathert et al.

NATURE (2015)

Article Multidisciplinary Sciences

BET inhibitor resistance emerges from leukaemia stem cells

Chun Yew Fong et al.

NATURE (2015)

Article Biochemical Research Methods

CrossMap: a versatile tool for coordinate conversion between genome assemblies

Hao Zhao et al.

BIOINFORMATICS (2014)

Article Multidisciplinary Sciences

Therapeutic targeting of BET bromodomain proteins in castration-resistant prostate cancer

Irfan A. Asangani et al.

NATURE (2014)

Article Multidisciplinary Sciences

Ubiquitylome analysis identifies dysregulation of effector substrates in SPOP-mutant prostate cancer

Jean-Philippe P. Theurillat et al.

SCIENCE (2014)

Article Biochemistry & Molecular Biology

Selective Inhibition of Tumor Oncogenes by Disruption of Super-Enhancers

Jakob Loven et al.

Article Biochemistry & Molecular Biology

BRCA1 is a negative modulator of the PRC2 complex

Lan Wang et al.

EMBO JOURNAL (2013)

Article Medicine, Research & Experimental

Multicolor microRNA FISH effectively differentiates tumor types

Neil Renwick et al.

JOURNAL OF CLINICAL INVESTIGATION (2013)

Article Multidisciplinary Sciences

Prostate cancer-associated mutations in speckle-type POZ protein (SPOP) regulate steroid receptor coactivator 3 protein turnover

Chuandong Geng et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2013)

Article Biochemical Research Methods

RSeQC: quality control of RNA-seq experiments

Liguo Wang et al.

BIOINFORMATICS (2012)

Article Genetics & Heredity

Exome sequencing identifies recurrent SPOP, FOXA1 and MED12 mutations in prostate cancer

Christopher E. Barbieri et al.

NATURE GENETICS (2012)

Article Biochemistry & Molecular Biology

BET Bromodomain Inhibition as a Therapeutic Strategy to Target c-Myc

Jake E. Delmore et al.

Article Biochemistry & Molecular Biology

Rac1 Regulates the Activity of mTORC1 and mTORC2 and Controls Cellular Size

Abdelhafid Saci et al.

MOLECULAR CELL (2011)

Article Multidisciplinary Sciences

RNAi screen identifies Brd4 as a therapeutic target in acute myeloid leukaemia

Johannes Zuber et al.

NATURE (2011)

Article Multidisciplinary Sciences

Targeting MYC dependence in cancer by inhibiting BET bromodomains

Jennifer A. Mertz et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2011)

Article Multidisciplinary Sciences

Suppression of inflammation by a synthetic histone mimic

Edwige Nicodeme et al.

NATURE (2010)

Article Multidisciplinary Sciences

Selective inhibition of BET bromodomains

Panagis Filippakopoulos et al.

NATURE (2010)

Article Biotechnology & Applied Microbiology

A scaling normalization method for differential expression analysis of RNA-seq data

Mark D. Robinson et al.

GENOME BIOLOGY (2010)

Article Biochemical Research Methods

TopHat: discovering splice junctions with RNA-Seq

Cole Trapnell et al.

BIOINFORMATICS (2009)

Article Biochemistry & Molecular Biology

Raft nanodomains contribute to Akt/PKB plasma membrane recruitment and activation

Remi Lasserre et al.

NATURE CHEMICAL BIOLOGY (2008)

Article Biochemical Research Methods

Mapping and quantifying mammalian transcriptomes by RNA-Seq

Ali Mortazavi et al.

NATURE METHODS (2008)

Article Biotechnology & Applied Microbiology

Model-based Analysis of ChIP-Seq (MACS)

Yong Zhang et al.

GENOME BIOLOGY (2008)

Article Biochemistry & Molecular Biology

Core transcriptional regulatory circuitry in human embryonic stem cells

LA Boyer et al.