Journal
RSC ADVANCES
Volume 9, Issue 25, Pages 13959-13967Publisher
ROYAL SOC CHEMISTRY
DOI: 10.1039/c9ra02569c
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Funding
- National Natural Science Foundation of China [21702184, 21772175]
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An efficient palladium-catalyzed intramolecular deacetylative dearomatization reaction of 3-acetoxyindoles has been developed. A range of tetracyclic indolin-3-ones bearing C2-quaternary stereocenters are achieved in good yields, showing a wide substrate scope for this reaction. A preliminary enantioselective reaction is established to furnish the product in 63% ee by using (R,R,R)-phosphoramide-PE as a chiral ligand.
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