Journal
ORGANIC & BIOMOLECULAR CHEMISTRY
Volume 17, Issue 18, Pages 4446-4451Publisher
ROYAL SOC CHEMISTRY
DOI: 10.1039/c9ob00622b
Keywords
-
Categories
Funding
- Zhejiang Province Science and Technology Plan Project [LGF18B060004]
- National Natural Science Foundation of China [21406201]
Ask authors/readers for more resources
A facile decarboxylative acylation of N-free indoles with a-ketonates via liquid-assisted grinding was reported. The reaction requires only a catalytic amount of Cu( OAc)2 center dot H2O in combination with O2 as the terminal oxidant to give various 3-acylindoles with high efficiency. Additionally, this new methodology was applicable to a gram-scale synthesis.
Authors
I am an author on this paper
Click your name to claim this paper and add it to your profile.
Reviews
Recommended
No Data Available