Related references
Note: Only part of the references are listed.A partial trace amine-associated receptor 1 agonist exhibits properties consistent with a methamphetamine substitution treatment
Yue Pei et al.
ADDICTION BIOLOGY (2017)
New insights into the structure of the trace amine-associated receptor 2: Homology modelling studies exploring the binding mode of 3-iodothyron amine
Elena Cichero et al.
CHEMICAL BIOLOGY & DRUG DESIGN (2017)
Role of TAAR1 within the Subregions of the Mesocorticolimbic Dopaminergic System in Cocaine-Seeking Behavior
Jian-Feng Liu et al.
JOURNAL OF NEUROSCIENCE (2017)
Trace Amine-Associated Receptor | Regulates Wakefulness and EEG Spectral Composition
Michael D. Schwartz et al.
NEUROPSYCHOPHARMACOLOGY (2017)
The Trace Amine-Associated Receptor 1 Agonist RO5256390 Blocks Compulsive, Binge-like Eating in Rats
Antonio Ferragud et al.
NEUROPSYCHOPHARMACOLOGY (2017)
Novel biguanide-based derivatives scouted as TAAR1 agonists: Synthesis, biological evaluation, ADME prediction and molecular docking studies
Michele Tonelli et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2017)
Thyronamines and Analogues - The Route from Rediscovery to Translational Research on Thyronergic Amines
Grazia Chiellini et al.
MOLECULAR AND CELLULAR ENDOCRINOLOGY (2017)
Trace Amine-Associated Receptor 1 Agonists as Narcolepsy Therapeutics
Sarah W. Black et al.
BIOLOGICAL PSYCHIATRY (2017)
Moroxydine hydrochloride inhibits grass carp reovirus replication and suppresses apoptosis in Ctenopharyngodon idella kidney cells
Xiao-Bo Yu et al.
ANTIVIRAL RESEARCH (2016)
The emerging roles of human trace amines and human trace amine- associated receptors (hTAARs) in central nervous system
Muhammad Zahid Khan et al.
BIOMEDICINE & PHARMACOTHERAPY (2016)
3-iodothyronamine (T1AM), a novel antagonist of muscarinic receptors
Annunziatina Laurino et al.
EUROPEAN JOURNAL OF PHARMACOLOGY (2016)
Effects of Trace Amine-associated Receptor 1 Agonists on the Expression, Reconsolidation, and Extinction of Cocaine Reward Memory
Jian-Feng Liu et al.
INTERNATIONAL JOURNAL OF NEUROPSYCHOPHARMACOLOGY (2016)
Hit-to-Lead Optimization of Mouse Trace Amine Associated Receptor 1 (mTAAR1) Agonists with a Diphenylmethane-Scaffold: Design, Synthesis, and Biological Study
Grazia Chiellini et al.
JOURNAL OF MEDICINAL CHEMISTRY (2016)
Increased context-dependent conditioning to amphetamine in mice lacking TAAR1
Ilya Sukhanov et al.
PHARMACOLOGICAL RESEARCH (2016)
Combinatorial effects of odorants on mouse behavior
Luis R. Saraiva et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2016)
Thyronamines and Derivatives: Physiological Relevance, Pharmacological Actions, and Future Research Directions
Carolin Stephanie Hoefig et al.
THYROID (2016)
A homology modelling-driven study leading to the discovery of the first mouse trace amine-associated receptor 5 (TAAR5) antagonists
Elena Cichero et al.
MEDCHEMCOMM (2016)
Discovery and Characterization of 2-Aminooxazolines as Highly Potent, Selective, and Orally Active TAAR1 Agonists
Guido Galley et al.
ACS MEDICINAL CHEMISTRY LETTERS (2016)
Trace Amines and the Trace Amine-Associated Receptor 1: Pharmacology, Neurochemistry, and Clinical Implications
Yue Pei et al.
FRONTIERS IN NEUROSCIENCE (2016)
Incretin-like effects of small molecule trace amine-associated receptor 1 agonists
Susanne Raab et al.
MOLECULAR METABOLISM (2016)
In Vitro Characterization of Psychoactive Substances at Rat, Mouse, and Human Trace Amine-Associated Receptor 1
Linda D. Simmler et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2016)
Thyronamine induces TRPM8 channel activation in human conjunctival epithelial cells
Noushafarin Khajavi et al.
CELLULAR SIGNALLING (2015)
Behavioral, biological, and chemical perspectives on atypical agents targeting the dopamine transporter
Maarten E. A. Reith et al.
DRUG AND ALCOHOL DEPENDENCE (2015)
Design, Synthesis, and Evaluation of Thyronamine Analogues as Novel Potent Mouse Trace Amine Associated Receptor 1 (mTAAR1) Agonists
Grazia Chiellini et al.
JOURNAL OF MEDICINAL CHEMISTRY (2015)
3-iodothyronamine differentially modulates α-2A-adrenergic receptor-mediated signaling
Juliane Dinter et al.
JOURNAL OF MOLECULAR ENDOCRINOLOGY (2015)
Modulation by Trace Amine-Associated Receptor 1 of Experimental Parkinsonism, L-DOPA Responsivity, and Glutamatergic Neurotransmission
Alexandra Alvarsson et al.
JOURNAL OF NEUROSCIENCE (2015)
Postsynaptic D2 dopamine receptor supersensitivity in the striatum of mice lacking TAAR1
Stefano Espinoza et al.
NEUROPHARMACOLOGY (2015)
TAAR1 Modulates Cortical Glutamate NMDA Receptor Function
Stefano Espinoza et al.
NEUROPSYCHOPHARMACOLOGY (2015)
Trace Amine-Associated Receptor 1 Regulation of Methamphetamine Intake and Related Traits
John H. Harkness et al.
NEUROPSYCHOPHARMACOLOGY (2015)
Selective activation of the trace amine-associated receptor 1 decreases cocaine's reinforcing efficacy and prevents cocaine-induced changes in brain reward thresholds
Yue Pei et al.
PROGRESS IN NEURO-PSYCHOPHARMACOLOGY & BIOLOGICAL PSYCHIATRY (2015)
Discovery of trace amine-associated receptor 1 ligands by molecular docking screening against a homology model
V. M. Lam et al.
MEDCHEMCOMM (2015)
Non-classical amine recognition evolved in a large clade of olfactory receptors
Qian Li et al.
ELIFE (2015)
Inverse Agonistic Action of 3-Iodothyronamine at the Human Trace Amine-Associated Receptor 5
Juliane Dinter et al.
PLOS ONE (2015)
The Multitarget Ligand 3-Iodothyronamine Modulates β-Adrenergic Receptor 2 Signaling
Juliane Dinter et al.
EUROPEAN THYROID JOURNAL (2015)
Evolutionary Conservation of 3-Iodothyronamine as an Agonist at the Trace Amine-Associated Receptor 1
Maxi Coester et al.
EUROPEAN THYROID JOURNAL (2015)
Further Insights Into the Pharmacology of the Human Trace Amine-Associated Receptors: Discovery of Novel Ligands for TAAR1 by a Virtual Screening Approach
Elena Cichero et al.
CHEMICAL BIOLOGY & DRUG DESIGN (2014)
Exploring the Determinants of Trace Amine-Associated Receptor 1's Functional Selectivity for the Stereoisomers of Amphetamine and Methamphetamine
Edmund A. Reese et al.
JOURNAL OF MEDICINAL CHEMISTRY (2014)
Olfactory Receptor Patterning in a Higher Primate
Lisa F. Horowitz et al.
JOURNAL OF NEUROSCIENCE (2014)
Taar1-mediated modulation of presynaptic dopaminergic neurotransmission: Role of D2 dopamine autoreceptors
D. Leo et al.
NEUROPHARMACOLOGY (2014)
Activation of the Trace Amine-Associated Receptor 1 Prevents Relapse to Cocaine Seeking
Yui Pei et al.
NEUROPSYCHOPHARMACOLOGY (2014)
Anatomical and functional evidence for trace amines as unique modulators of locomotor function in the mammalian spinal cord
Elizabetha A. Gozal et al.
FRONTIERS IN NEURAL CIRCUITS (2014)
Insights into the Structure and Pharmacology of the Human Trace Amine-Associated Receptor 1 (hTAAR1): Homology Modelling and Docking Studies
Elena Cichero et al.
CHEMICAL BIOLOGY & DRUG DESIGN (2013)
Functional evaluation of the receptors mediating vasoconstriction of rat aorta by trace amines and amphetamines
Kenneth J. Broadley et al.
EUROPEAN JOURNAL OF PHARMACOLOGY (2013)
Potential applications for biguanides in oncology
Michael Pollak
JOURNAL OF CLINICAL INVESTIGATION (2013)
Biogenic amines activate blood leukocytes via trace amine-associated receptors TAAR1 and TAAR2
Agne Babusyte et al.
JOURNAL OF LEUKOCYTE BIOLOGY (2013)
Ultrasensitive Detection of Amines by a Trace Amine-Associated Receptor
Jingji Zhang et al.
JOURNAL OF NEUROSCIENCE (2013)
A new perspective for schizophrenia: TAAR1 agonists reveal antipsychotic- and antidepressant-like activity, improve cognition and control body weight
F. G. Revel et al.
MOLECULAR PSYCHIATRY (2013)
Human Trace Amine-Associated Receptor TAAR5 Can Be Activated by Trimethylamine
Ivonne Wallrabenstein et al.
PLOS ONE (2013)
Trace Amine-Associated Receptor 1 Partial Agonism Reveals Novel Paradigm for Neuropsychiatric Therapeutics
Florent G. Revel et al.
BIOLOGICAL PSYCHIATRY (2012)
Optimisation of imidazole compounds as selective TAAR1 agonists: Discovery of RO5073012
Guido Galley et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2012)
Vasoconstrictor and vasodilator responses to tryptamine of rat-isolated perfused mesentery: comparison with tyramine and β-phenylethylamine
M. A. Anwar et al.
BRITISH JOURNAL OF PHARMACOLOGY (2012)
Role of Catechol-O-Methyltransferase (COMT)-Dependent Processes in Parkinson's Disease and L-DOPA Treatment
Stefano Espinoza et al.
CNS & NEUROLOGICAL DISORDERS-DRUG TARGETS (2012)
Synthesis, Biological Evaluation, and Docking Studies of Tetrahydrofuran- Cyclopentanone- and Cyclopentanol-Based Ligands Acting at Adrenergic α1- and Serotonine 5-HT1A Receptors
Adolfo Prandi et al.
JOURNAL OF MEDICINAL CHEMISTRY (2012)
Avenues for the Development of Therapeutics That Target Trace Amine Associated Receptor 1 (TAAR1)
Gregory M. Miller
JOURNAL OF MEDICINAL CHEMISTRY (2012)
Brain-Specific Overexpression of Trace Amine-Associated Receptor I Alters Monoaminergic Neurotransmission and Decreases Sensitivity to Amphetamine
Florent G. Revel et al.
NEUROPSYCHOPHARMACOLOGY (2012)
Augmentation of methamphetamine-induced behaviors in transgenic mice lacking the trace amine-associated receptor 1
Cindy Achat-Mendes et al.
PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR (2012)
Neurons expressing trace amine-associated receptors project to discrete glomeruli and constitute an olfactory subsystem
Mark A. Johnson et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2012)
An Olfactory Subsystem that Mediates High-Sensitivity Detection of Volatile Amines
Rodrigo Pacifico et al.
CELL REPORTS (2012)
Selective antagonists of mouse trace amine-associated receptor 1 (mTAAR1): Discovery of EPPTB (RO5212773)
Henri Stalder et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2011)
The emerging role of trace amine-associated receptor 1 in the functional regulation of monoamine transporters and dopaminergic activity
Gregory M. Miller
JOURNAL OF NEUROCHEMISTRY (2011)
Genetic Deletion of Trace Amine 1 Receptors Reveals Their Role in Auto-Inhibiting the Actions of Ecstasy (MDMA)
Benjamin Di Cara et al.
JOURNAL OF NEUROSCIENCE (2011)
Structure and function of an irreversible agonist-β2 adrenoceptor complex
Daniel M. Rosenbaum et al.
NATURE (2011)
TAAR1 activation modulates monoaminergic neurotransmission, preventing hyperdopaminergic and hypoglutamatergic activity
Florent G. Revel et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2011)
Human and mouse trace amine-associated receptor 1 have distinct pharmacology towards endogenous monoamines and imidazoline receptor ligands
Liaoyuan A. Hu et al.
BIOCHEMICAL JOURNAL (2009)
Anatomical and histological profiling of orphan G-protein-coupled receptor expression in gastrointestinal tract of C57BL/6J mice
Junko Ito et al.
CELL AND TISSUE RESEARCH (2009)
A Receptor Mechanism for Methamphetamine Action in Dopamine Transporter Regulation in Brain
Zhihua Xie et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2009)
The selective antagonist EPPTB reveals TAAR1-mediated regulatory mechanisms in dopaminergic neurons of the mesolimbic system
Amyaouch Bradaia et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2009)
Synthesis, structure elucidation and identification of antitumoural properties of novel fused 1,2,4-triazine aryl derivatives
Krzysztof Sztanke et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2008)
Modulation of monoamine transporters by common biogenic amines via trace amine-associated receptor 1 and monoamine autoreceptors in human embryonic kidney 293 cells and brain synaptosomes
Zhihua Xie et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2008)
Trace amine associated receptor 1 and movement control
Tatyana D. Sotnikova et al.
PARKINSONISM & RELATED DISORDERS (2008)
Trace amine-associated receptor 1 modulates dopaminergic activity
Lothar Lindemann et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2008)
The trace amine 1 receptor knockout mouse: an animal model with relevance to schizophrenia
T. D. Wolinsky et al.
GENES BRAIN AND BEHAVIOR (2007)
Exploring the structure-activity relationship of the ethylamine portion of 3-iodothyronamine for rat and mouse trace amine-associated receptor 1
Edwin S. Tan et al.
JOURNAL OF MEDICINAL CHEMISTRY (2007)
Rhesus monkey trace amine-associated receptor 1 signaling: Enhancement by monoamine transporters and attenuation by the D2 autoreceptor in vitro
Zhihua Xie et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2007)
Pharmacologic characterization of the cloned human trace amine-associated receptor1 (TAAR1) and evidence for species differences with the rat TAAR1
David B. Wainscott et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2007)
A second class of chemosensory receptors in the olfactory epithelium
Stephen D. Liberles et al.
NATURE (2006)
Effects of intravenous glucagon-like peptide-1 on gastric emptying and intragastric distribution in healthy subjects: Relationships with postprandial glycemic and insulinemic responses
TJ Little et al.
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM (2006)
Trace amine-associated receptor agonists: Synthesis and evaluation of thyronamines and related analogues
ME Hart et al.
JOURNAL OF MEDICINAL CHEMISTRY (2006)
Contributions of the amygdala to emotion processing: From animal models to human behavior
EA Phelps et al.
NEURON (2005)
A renaissance in trace amines inspired by a novel GPCR family
L Lindemann et al.
TRENDS IN PHARMACOLOGICAL SCIENCES (2005)
Trace amine-associated receptors form structurally and functionally distinct subfamilies of novel G protein-coupled receptors
L Lindemann et al.
GENOMICS (2005)
Mammalian central nervous system trace amines. Pharmacologic amphetamines, physiologic neuromodulators
MD Berry
JOURNAL OF NEUROCHEMISTRY (2004)
Arylguanidine and arylbiguanide binding at 5-HT3 serotonin receptors:: A QSAR study
RA Glennon et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2003)
Trace amines: Identification of a family of mammalian G protein-coupled receptors
B Borowsky et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2001)