Journal
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
Volume 2017, Issue 16, Pages 2272-2279Publisher
WILEY-V C H VERLAG GMBH
DOI: 10.1002/ejoc.201700095
Keywords
Nitrogen heterocycles; C-H activation; Diazo compounds; Annulation; Iridium
Categories
Funding
- Department of Science and Technology - Innovation in Science Pursuit for Inspired Research (DST-INSPIRE) Faculty program [GAP-0738]
Ask authors/readers for more resources
A one-pot synthesis of indole derivatives from readily available acetanilides and diazo compounds was developed. This Ir-III-catalyzed C-H alkylation and annulation reaction proceeds under mild conditions and generates molecular nitrogen and water as byproducts. Various types of synthetically versatile N-substituted indoles, including N-acetyl, N-pivolyl, and N-benzoyl indoles, were prepared.
Authors
I am an author on this paper
Click your name to claim this paper and add it to your profile.
Reviews
Recommended
No Data Available