Related references
Note: Only part of the references are listed.Final Efficacy Results of Neratinib in HER2-positive Hormone Receptor-positive Early-stage Breast Cancer From the Phase III ExteNET Trial
Arlene Chan et al.
CLINICAL BREAST CANCER (2021)
Novel oxindole/benzofuran hybrids as potential dual CDK2/GSK-3β inhibitors targeting breast cancer: design, synthesis, biological evaluation, and in silico studies
Wagdy M. Eldehna et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2021)
Genome-wide synthetic lethal screen unveils novel CAIX-NFS1/xCT axis as a targetable vulnerability in hypoxic solid tumors
Shawn C. Chafe et al.
SCIENCE ADVANCES (2021)
Design, synthesis, anticancer, antibacterial, and antifungal evaluation of 4-aminoquinoline-1,3,5-triazine derivatives
Hans Raj Bhat et al.
JOURNAL OF HETEROCYCLIC CHEMISTRY (2020)
Progress in the development of human carbonic anhydrase inhibitors and their pharmacological applications: Where are we today?
Chandra B. Mishra et al.
MEDICINAL RESEARCH REVIEWS (2020)
Carbonic Anhydrases: Versatile and Useful Biocatalysts in Chemistry and Biochemistry
Andrea Angeli et al.
CATALYSTS (2020)
Antitumor properties of certain spirooxindoles towards hepatocellular carcinoma endowed with antioxidant activity
Sara T. Al-Rashood et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2020)
Design, eco-friendly synthesis, molecular modeling and anticancer evaluation of thiazol-5(4H)-ones as potential tubulin polymerization inhibitors targeting the colchicine binding site
Abeer M. El-Naggar et al.
RSC ADVANCES (2020)
The role of carbonic anhydrase IX in cancer development: links to hypoxia, acidosis, and beyond
Silvia Pastorekova et al.
CANCER AND METASTASIS REVIEWS (2019)
Design, synthesis and anticancer evaluation of thieno[2,3-d]pyrimidine derivatives as dual EGFR/HER2 inhibitors and apoptosis inducers
Souad A. Elmetwally et al.
BIOORGANIC CHEMISTRY (2019)
Synthesis, biological evaluation and in silico studies with 4-benzylidene-2phenyl-5(4H)-imidazolone-based benzenesulfonamides as novel selective carbonic anhydrase IX inhibitors endowed with anticancer activity
Wagdy M. Eldehna et al.
BIOORGANIC CHEMISTRY (2019)
Role of Carbonic Anhydrases and Inhibitors in Acid-Base Physiology: Insights from Mathematical Modeling
Rossana Occhipinti et al.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (2019)
A New Kid on the Block? Carbonic Anhydrases as Possible New Targets in Alzheimer's Disease
Gustavo Provensi et al.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (2019)
The use of cobalt chloride as a chemical hypoxia model
Jorge Munoz-Sanchez et al.
JOURNAL OF APPLIED TOXICOLOGY (2019)
Synthesis and biological evaluation of novel 8-substituted quinoline-2-carboxamides as carbonic anhydrase inhibitors
Pavitra S. Thacker et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2019)
CoCl2 simulated hypoxia induce cell proliferation and alter the expression pattern of hypoxia associated genes involved in angiogenesis and apoptosis
Nishant Kumar Rana et al.
BIOLOGICAL RESEARCH (2019)
Synthesis and biological evaluation of novel 3-(quinolin-4-ylamino)benzenesulfonamidesAQ3 as carbonic anhydrase isoforms I and II inhibitors
Mohammad M. Al-Sanea et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2019)
Carbonic anhydrase IX enhances tumor cell proliferation and tumor progression in osteosarcoma
Kazuma Okuno et al.
ONCOTARGETS AND THERAPY (2018)
An overview of quinoline as a privileged scaffold in cancer drug discovery
Robert Musiol
EXPERT OPINION ON DRUG DISCOVERY (2017)
Carbonic anhydrase XII functions in health and disease
Abdul Waheed et al.
GENE (2017)
The human carbonic anhydrase isoenzymes I and II (hCA I and II) inhibition effects of trimethoxyindane derivatives
Parham Taslimi et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2016)
Evaluation of CAIX and CAXII Expression in Breast Cancer at Varied O2 Levels: CAIX is the Superior Surrogate Imaging Biomarker of Tumor Hypoxia
Narges K. Tafreshi et al.
MOLECULAR IMAGING AND BIOLOGY (2016)
Intrinsic thermodynamics of 4-substituted-2,3,5,6-tetrafluorobenzenesulfonamide binding to carbonic anhydrases by isothermal titration calorimetry
Asta Zubriene et al.
BIOPHYSICAL CHEMISTRY (2015)
Pelitinib (EKB-569) targets the up-regulation of ABCB1 and ABCG2 induced by hyperthermia to eradicate lung cancer
Kenneth K. W. To et al.
BRITISH JOURNAL OF PHARMACOLOGY (2015)
Efficient Expression and Crystallization System of Cancer-Associated Carbonic Anhydrase Isoform IX
Janis Leitans et al.
JOURNAL OF MEDICINAL CHEMISTRY (2015)
Anticonvulsant/antiepileptic carbonic anhydrase inhibitors: a patent review
Mayank Aggarwal et al.
EXPERT OPINION ON THERAPEUTIC PATENTS (2013)
Structural annotation of human carbonic anhydrases
Mayank Aggarwal et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2013)
Phase II study of single-agent bosutinib, a Src/Abl tyrosine kinase inhibitor, in patients with locally advanced or metastatic breast cancer pretreated with chemotherapy
M. Campone et al.
ANNALS OF ONCOLOGY (2012)
A new approach to antiglaucoma drugs: carbonic anhydrase inhibitors with or without NO donating moieties. Mechanism of action and preliminary pharmacology
Francesca Fabrizi et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2012)
Meldrum's Acids and 5-Alkylidene Meldrum's Acids in Catalytic Carbon-Carbon Bond-Forming Processes
Aaron M. Dumas et al.
ACCOUNTS OF CHEMICAL RESEARCH (2010)
Hypoxia-Inducible Carbonic Anhydrase IX and XII Promote Tumor Cell Growth by Counteracting Acidosis through the Regulation of the Intracellular pH
Johanna Chiche et al.
CANCER RESEARCH (2009)
One-pot and sequential organic chemistry on an enzyme surface to tether a fluorescent probe at the proximity of the active site with restoring enzyme activity
Y Takaoka et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2006)
Synthesis of ring-substituted 4-aminoquinolines and evaluation of their antimalarial activities
PB Madrid et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2005)