Related references
Note: Only part of the references are listed.Design, synthesis, biological screening and molecular docking studies of novel multifunctional 1,4-di (aryl/heteroaryl) substituted piperazine derivatives as potential antitubercular and antimicrobial agents
Bruktawit Mekonnen T. Sanka et al.
BIOORGANIC CHEMISTRY (2022)
Design, synthesis and SAR of antitubercular benzylpiperazine ureas
Sohal Satish et al.
MOLECULAR DIVERSITY (2022)
An appraisal of anti-mycobacterial activity with structure-activity relationship of piperazine and its analogues: A review
Pankaj S. Girase et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2021)
Design, synthesis and biological evaluation of novel 1,2,3-triazole analogues of Imidazo-[1,2-a]-pyridine-3-carboxamide against Mycobacterium tuberculosis
Adinarayana Nandikolla et al.
TOXICOLOGY IN VITRO (2021)
Design and synthesis of novel Imidazo[2,1-b]thiazole derivatives as potent antiviral and antimycobacterial agents
Elif Gursoy et al.
BIOORGANIC CHEMISTRY (2020)
Intracellular and in vivo evaluation of imidazo [2,1-b]thiazole-5-carboxamide antituberculosis compounds
Garrett C. Moraski et al.
PLOS ONE (2020)
Discovery of 1,2,3-triazole based quinoxaline-1,4-di- N -oxide derivatives as potential anti -tubercular agents
Singireddi Srinivasarao et al.
BIOORGANIC CHEMISTRY (2020)
Features of the biochemistry of Mycobacterium smegmatis, as a possible model for Mycobacterium tuberculosis
Joseph Antony Sundarsingh T et al.
Journal of Infection and Public Health (2020)
Inhibitors of pantothenate synthetase ofMycobacterium tuberculosis- a medicinal chemist perspective
Amaroju Suresh et al.
RSC ADVANCES (2020)
2,6-Disubstituted imidazo[2,1-b][1,3,4]thiadiazole derivatives as potent staphylococcal biofilm inhibitors
Stella Cascioferro et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2019)
Opportunities for Overcoming Mycobacterium tuberculosis Drug Resistance: Emerging Mycobacterial Targets and Host-Directed Therapy
Eveline Torfs et al.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (2019)
The synthesis and in vitro biological evaluation of novel fluorinated tetrahydrobenzo[j]phenanthridine-7,12-diones against Mycobacterium tuberculosis
Davie Cappoen et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2019)
RCSB Protein Data Bank: biological macromolecular structures enabling research and education in fundamental biology, biomedicine, biotechnology and energy
Stephen K. Burley et al.
NUCLEIC ACIDS RESEARCH (2019)
Treatment of Mycobacterium abscessus Complex
Luke Strnad et al.
SEMINARS IN RESPIRATORY AND CRITICAL CARE MEDICINE (2018)
Design, synthesis and antitubercular potency of 4-hydroxyquinolin-2(1H)-ones
Maira Bidart de Macedo et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2017)
Identification and development of pyrazolo[4,3-c]pyridine carboxamides as Mycobacterium tuberculosis pantothenate synthetase inhibitors
Suresh Amaroju et al.
NEW JOURNAL OF CHEMISTRY (2017)
SwissADME: a free web tool to evaluate pharmacokinetics, drug-likeness and medicinal chemistry friendliness of small molecules
Antoine Daina et al.
SCIENTIFIC REPORTS (2017)
FAF-Drugs4: free ADME-tox filtering computations for chemical biology and early stages drug discovery
David Lagorce et al.
BIOINFORMATICS (2017)
Optimization of Inhibitors of Mycobacterium tuberculosis Pantothenate Synthetase Based on Group Efficiency Analysis
Alvin W. Hung et al.
CHEMMEDCHEM (2016)
Design, synthesis and biological evaluation of imidazo[2,1-b]thiazole and benzo[d]imidazo[2,1-b]thiazole derivatives as Mycobacterium tuberculosis pantothenate synthetase inhibitors
Ganesh Samala et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2016)
Design, synthesis and biological evaluation of novel quinoline-based carboxylic hydrazides as anti-tubercular agents
Subhash Chander et al.
CHEMICAL BIOLOGY & DRUG DESIGN (2016)
Biological activities of imidazo[2,1-b][1,3,4]-thiadiazole derivatives: A review
Bhoomendra A. Bhongade et al.
JOURNAL OF SAUDI CHEMICAL SOCIETY (2016)
Arrival of Imidazo[2,1-b]thiazole-5-carboxamides: Potent Antituberculosis Agents That Target QcrB
Garrett C. Moraski et al.
ACS INFECTIOUS DISEASES (2016)
1,2,3-Triazole derivatives as antitubercular agents: synthesis, biological evaluation and molecular docking study
Mubarak H. Shaikh et al.
MEDCHEMCOMM (2015)
Design, synthesis and evaluation of 1,2,3-triazole-adamantylacetamide hybrids as potent inhibitors of Mycobacterium tuberculosis
Dinesh Addla et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2014)
Rational design and synthesis of novel dibenzo[b,d]furan-1,2,3-triazole conjugates as potent inhibitors of Mycobacterium tuberculosis
Thirumal Yempala et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Synthesis of novel 1,2,3-triazole derivatives of isoniazid and their in vitro and in vivo antimycobacterial activity evaluation
Deepak Kumar et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Synthesis and evaluation of α-ketotriazoles and α,β-diketotriazOles as inhibitors of Mycobacterium tuberculosis
Christophe Menendez et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2013)
3-Substituted 2-Phenylimidazo[2,1-b]benzothiazoles: Synthesis, Anticancer Activity, and Inhibition of Tubulin Polymerization
Ahmed Kamal et al.
CHEMMEDCHEM (2012)
Chemical synthesis and biological evaluation of triazole derivatives as inhibitors of InhA and antituberculosis agents
Christophe Menendez et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2012)
Synthesis and biological evaluation of imidazolo[2,1-b]benzothiazole derivatives, as potential p53 inhibitors
Michael S. Christodoulou et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2011)
Efficient synthesis and in vitro antitubercular activity of 1,2,3-triazoles as inhibitors of Mycobacterium tuberculosis
Poovan Shanmugavelan et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2011)
Imidazo[2,1-b]thiazole carbohydrate derivatives: Synthesis and antiviral activity against Junin virus, agent of Argentine hemorrhagic fever
Jose Sebastian Barradas et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2011)
Design, synthesis and in vitro antimicrobial evaluation of novel Imidazo[1,2-a]pyridine and imidazo[2,1-b][1,3]benzothiazole motifs
Taleb H. Al-Tel et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2011)
Imidazo[2,1-b]thiazole guanylhydrazones as RSK2 inhibitors [1]
Aldo Andreani et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2011)
Synthesis and Antibacterial Activity of a Novel Series of 2,3-Diaryl-substituted-imidazo(2,1-b)-benzothiazole Derivatives
Mahesh Palkar et al.
ARCHIV DER PHARMAZIE (2010)
Discovery and optimization of N-acyl and N-aroylpyrazolines as B-Raf kinase inhibitors
Christopher Blackburn et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2010)
Synthesis, Anthelmintic and Anti-inflammatory Activities of Some Novel Imidazothiazole Sulfides and Sulfones
Nitinkumar S. Shetty et al.
BULLETIN OF THE KOREAN CHEMICAL SOCIETY (2010)
Targeting mycobacterium protein tyrosine phosphatase B for antituberculosis agents
Bo Zhou et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2010)
Application of Fragment Growing and Fragment Linking to the Discovery of Inhibitors of Mycobacterium tuberculosis Pantothenate Synthetase
Alvin W. Hung et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2009)
Arylcarboxyamino-substituted diaryl ureas as potent and selective FLT3 inhibitors
Hitesh K. Patel et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2009)
Potential Antitumor Agents.: 42.: New antitumor imidazo[2,1-b]thiazole guanylhydrazones and analogues'
Aldo Andreani et al.
JOURNAL OF MEDICINAL CHEMISTRY (2008)
Synthesis of phosphorus and sulfur heterocycles via ring-closing olefin metathesis
MD McReynolds et al.
CHEMICAL REVIEWS (2004)
Synthesis and antitubercular activity of imidazo[2,1-b] thiazoles
A Andreani et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2001)
Synthesis of cyclic sulfonamides through intramolecular Diels-Alder reactions
IR Greig et al.
ORGANIC LETTERS (2001)
Synthesis of cyclic sulfonamides via intramolecular copper-catalyzed reaction of unsaturated iminoiodinanes
P Dauban et al.
ORGANIC LETTERS (2000)
Investigation of the Alamar Blue (resazurin) fluorescent dye for the assessment of mammalian cell cytotoxicity
J O'Brien et al.
EUROPEAN JOURNAL OF BIOCHEMISTRY (2000)