Journal
ASIAN JOURNAL OF ORGANIC CHEMISTRY
Volume 5, Issue 5, Pages 625-628Publisher
WILEY-V C H VERLAG GMBH
DOI: 10.1002/ajoc.201600096
Keywords
arylsulfonyl chlorides; copper catalysis; indoles; pyrrolo[2,3-b]pyridine; sulfenylation
Categories
Funding
- NSF of Jiangsu Province [BK20150129]
- Jiangsu Province for the Cultivation of Innovation and Pioneering Doctor [1016010241151030]
- 111 Project [111-2-06]
- Jiangsu province Collaborative Innovation Center for Advanced Industrial Fermentation industry development program
- Project for Jiangsu Scientific and Technological Innovation Team
Ask authors/readers for more resources
A copper-catalyzed regioselective sulfenylation of indoles and a pyrrolo[ 2,3-b]pyridine with arylsulfonyl chlorides has been developed by using low loadings of a copper catalyst and the cheap reductant PPh3. This method is effective for both N-protected and unprotected indoles, providing a series of structurally diverse indole thioethers in good to excellent yields with extremely high regioselectivity.
Authors
I am an author on this paper
Click your name to claim this paper and add it to your profile.
Reviews
Recommended
No Data Available
Share Paper
