Journal
CHEMISTRY-A EUROPEAN JOURNAL
Volume 21, Issue 41, Pages 14342-14346Publisher
WILEY-V C H VERLAG GMBH
DOI: 10.1002/chem.201502891
Keywords
amidation; cyclization; homogeneous catalysis; oxazolines; quinazolines
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Funding
- GlaxoSmithKline
- EPSRC
- Engineering and Physical Sciences Research Council [1614974] Funding Source: researchfish
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A Rh-catalyzed ortho-amidation cyclocondensation sequence gave a range of 4-aminoquinazolines in high yield. The method features a remarkably mild C(sp(2))- H activation step and can be exploited to rapidly access compounds with established biological activity.
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