Journal
ORGANIC LETTERS
Volume 18, Issue 6, Pages 1286-1289Publisher
AMER CHEMICAL SOC
DOI: 10.1021/acs.orglett.6b00198
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Funding
- National Basic Research Program of China [2012CB821600]
- Fundamental Research Funds for the Central Universities [20720160030]
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3-Arylsulfonylquinoline derivatives play important roles as pharmaceutical drugs. A new method for the synthesis of 3-arylsulfonylquinoline derivatives has been achieved through tert-butyl hydroperoxide mediated cycloaddition between N-propargyl aromatic amine derivatives and arylsulfonylhydrazides without the addition of any metals. This transformation offers a straightforward route to the formation of a C-S bond and quinoline ring in one step-via a sulfonylation-cyclization-aromatization process.
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