Journal
ORGANIC & BIOMOLECULAR CHEMISTRY
Volume 14, Issue 36, Pages 8615-8622Publisher
ROYAL SOC CHEMISTRY
DOI: 10.1039/c6ob01348a
Keywords
-
Categories
Funding
- National Natural Science Foundation of China [21372044]
- Fuzhou University [022494]
Ask authors/readers for more resources
An operationally simple method for the copper-mediated trifluoromethylthiolation of iodopyridinones employing (bpy) CuSCF3 (1; bpy = 2,2'-bipyridine) as a trifluoromethylthiolating reagent is presented. Various types of iodopyridinones are applicable and the trifluoromethylthiolated pyridinones are obtained in moderate to excellent yields. This method tolerates a variety of protecting groups on the nitrogen atom of pyridinones. In addition, scalability of the reaction is demonstrated.
Authors
I am an author on this paper
Click your name to claim this paper and add it to your profile.
Reviews
Recommended
No Data Available