Related references
Note: Only part of the references are listed.Validating Eaton's Hypothesis: Cubane as a Benzene Bioisostere
Benjamin A. Chalmers et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2016)
Redox-Active Esters in Fe-Catalyzed C-C Coupling
Fumihiko Toriyama et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2016)
Expedient synthesis of 3-phenylbicyclo[1.1.1]pentan-1-amine via metal-free homolytic aromatic alkylation of benzene
Navanita T. Thirumoorthi et al.
CHEMICAL COMMUNICATIONS (2015)
Radical fluorination powered expedient synthesis of 3-fluorobicyclo[1.1.1]pentan-1-amine
Yi Ling Goh et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2015)
Design, Synthesis, and Characterization of SO2-Containing Azabicyclo[3.n.1]alkanes: Promising Building Blocks for Drug Discovery
Tetiana Druzhenko et al.
ORGANIC LETTERS (2015)
Late-Stage Functionalization of Biologically Active Heterocycles Through Photoredox Catalysis
Daniel A. DiRocco et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2014)
A New Route to Bicyclo[1.1.1]pentan-1-amine from 1-Azido-3-iodobicyclo[1.1.1]pentane
Yi Ling Goh et al.
ORGANIC LETTERS (2014)
Cubanes in Medicinal Chemistry: Synthesis of Functionalized Building Blocks
Joanna Wlochal et al.
ORGANIC LETTERS (2014)
Application of the Bicyclo[1.1.1]pentane Motif as a Nonclassical Phenyl Ring Bioisostere in the Design of a Potent and Orally Active γ-Secretase Inhibitor
Antonia F. Stepan et al.
JOURNAL OF MEDICINAL CHEMISTRY (2012)
Fluorine Transfer to Alkyl Radicals
Montserrat Rueda-Becerril et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2012)
Silver-Catalyzed Decarboxylative Fluorination of Aliphatic Carboxylic Acids in Aqueous Solution
Feng Yin et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2012)
Synopsis of Some Recent Tactical Application of Bioisosteres in Drug Design
Nicholas A. Meanwell
JOURNAL OF MEDICINAL CHEMISTRY (2011)
Scalable Synthesis of 1-Bicyclo[1.1.1]pentylamine via a Hydrohydrazination Reaction
Kevin D. Bunker et al.
ORGANIC LETTERS (2011)
Minisci reactions: Versatile CH-functionalizations for medicinal chemists
Matthew A. J. Duncton
MEDCHEMCOMM (2011)
Oxetanes as Versatile Elements in Drug Discovery and Synthesis
Johannes A. Burkhard et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2010)
Discovery and Evaluation of BMS-708163, a Potent, Selective and Orally Bioavailable γ-Secretase Inhibitor
Kevin W. Gillman et al.
ACS MEDICINAL CHEMISTRY LETTERS (2010)
The impact of aromatic ring count on compound developability - are too many aromatic rings a liability in drug design?
Timothy J. Ritchie et al.
DRUG DISCOVERY TODAY (2009)
Escape from Flatland: Increasing Saturation as an Approach to Improving Clinical Success
Frank Lovering et al.
JOURNAL OF MEDICINAL CHEMISTRY (2009)
Synthesis using aromatic homolytic substitution - recent advances
W. Russell Bowman et al.
CHEMICAL SOCIETY REVIEWS (2007)
Synthesis and biological evaluation of 2-(3′-(1H-tetrazol-5-yl) bicyclo[1.1.1]pent-1-yl)glycine (S-TBPG), a novel mGlu1 receptor antagonist
G Costantino et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2001)
Share Paper
