Related references
Note: Only part of the references are listed.Recent updates on 1,2,3-triazole-containing hybrids with in vivo therapeutic potential against cancers: A mini-review
Shijia Zhao et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2023)
Click chemistry inspired syntheses of new amide linked 1,2,3-triazoles from naphthols: biological evaluation and in silico computational study
Satish V. V. Akolkar et al.
RESEARCH ON CHEMICAL INTERMEDIATES (2023)
Substituted naphthoxy-phthalonitrile derivatives: Synthesis, substituent effects, DFT, TD-DFT Calculations, antimicrobial properties and DNA interaction studies
Musa Erdogan et al.
COMPUTATIONAL BIOLOGY AND CHEMISTRY (2023)
Recent Advancements in Triazole-based Click Chemistry in Cancer Drug Discovery and Development
Arun Kumar et al.
SYNOPEN (2023)
Preparation of antioxidant-biodegradable poly(acrylic acid-co-2-hydroxyethyl methacrylate) hydrogel using rutin as a crosslinker: Drug release and anticancer activity
Ferah Comert Onder et al.
REACTIVE & FUNCTIONAL POLYMERS (2023)
Combinatorial Synthesis of Sulfonate Derivatives of α/β-Naphthol as Anti-Oomycete Agents
Zhiping Che et al.
COMBINATORIAL CHEMISTRY & HIGH THROUGHPUT SCREENING (2022)
Synthesis, antimicrobial evaluation and docking studies of fluorinated imine linked 1,2,3-triazoles
Aman Kumar et al.
RESEARCH ON CHEMICAL INTERMEDIATES (2022)
A 1,2,3-Triazole Derivative of Quinazoline Exhibits Antitumor Activity by Tethering RNF168 to SQSTM1/P62
Fu-Cheng Wang et al.
JOURNAL OF MEDICINAL CHEMISTRY (2022)
Click approach for synthesis of 3,4-dihydro-2(1H) quinolinone, coumarin moored 1,2,3-triazoles as inhibitor of mycobacteria tuberculosis H37RV, their antioxidant, cytotoxicity and in-silico studies
Nagashree U. Hebbar et al.
JOURNAL OF MOLECULAR STRUCTURE (2022)
Novel 1,3-Thiazole Analogues with Potent Activity against Breast Cancer: A Design, Synthesis, In Vitro, and In Silico Study
Manar G. Salem et al.
MOLECULES (2022)
Gene expression profile analysis to discover molecular signatures for early diagnosis and therapies of triple-negative breast cancer
Md Shahin Alam et al.
FRONTIERS IN MOLECULAR BIOSCIENCES (2022)
Fluorinated triazoles as privileged potential candidates in drug development-focusing on their biological and pharmaceutical properties
Ihsan Ullah et al.
FRONTIERS IN CHEMISTRY (2022)
Flavone-1,2,3-triazole derivatives as potential α-glucosidase inhibitors: Synthesis, enzyme inhibition, kinetic analysis and molecular docking study
Manoj Dhameja et al.
BIOORGANIC CHEMISTRY (2022)
The 1,2,3-triazole 'all-in-one' ring system in drug discovery: a good bioisostere, a good pharmacophore, a good linker, and a versatile synthetic tool
Deniz Lengerli et al.
EXPERT OPINION ON DRUG DISCOVERY (2022)
A New Naphthopyran Derivative Combines c-Myb Inhibition, Microtubule-Targeting Effects, and Antiangiogenic Properties
Leonhard H. F. Koehler et al.
ACS MEDICINAL CHEMISTRY LETTERS (2022)
Coumarin-4-yl‐1,2,3‐triazol‐4-yl-methyl-thiazolidine-2,4-diones: Synthesis, glucose uptake activity and cytotoxic evaluation
Tukaram V. Metre et al.
BIOORGANIC CHEMISTRY (2022)
A novel series of substituted 1,2,3-triazoles as cancer stem cell inhibitors: Synthesis and biological evaluation
Komal N. Padhariya et al.
DRUG DEVELOPMENT RESEARCH (2021)
Synthesis and structural characterization of novelO-substituted phenolic and chalcone derivatives with antioxidant activity
Bathelemy Ngameni et al.
JOURNAL OF CHEMICAL RESEARCH (2021)
1,2,3-Triazole derivatives: synthesis, docking, cytotoxicity analysis and in vivo antimalarial activity
Fernanda Valerio Lopes et al.
CHEMICO-BIOLOGICAL INTERACTIONS (2021)
Fluorine-containing pharmaceuticals approved by the FDA in 2020: Synthesis and biological activity
Yingjie Yu et al.
CHINESE CHEMICAL LETTERS (2021)
Sulfonamide derivatives as potential anti-cancer agents and their SARs elucidation
Yichao Wan et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2021)
Synthesis and docking calculations of tetrafluoronaphthalene derivatives and their inhibition profiles against some metabolic enzymes
Musa Erdogan et al.
ARCHIV DER PHARMAZIE (2021)
A novel fluorinated monomer: Synthesis, characterization and ATRP of 5,6,7,8-tetrafluoronaphthalen-1-yl acrylate
Musa Erdogan et al.
JOURNAL OF FLUORINE CHEMISTRY (2021)
Synthesis and biological evaluation of some 1-naphthol derivatives as antioxidants, acetylcholinesterase, and carbonic anhydrase inhibitors
Musa Erdogan et al.
ARCHIV DER PHARMAZIE (2021)
Synthesis, in vitro evaluation, and molecular docking studies of novel hydrazineylideneindolinone linked to 1,2,3-triazole derivatives as potential α-glucosidase inhibitors
Diba Shareghi-Boroujeni et al.
BIOORGANIC CHEMISTRY (2021)
Thiazole Ring-A Biologically Active Scaffold
Anthi Petrou et al.
MOLECULES (2021)
An in vivo evaluation of anti-inflammatory, analgesic and anti-pyretic activities of newly synthesized 1, 2, 4 Triazole derivatives
Tabinda Azim et al.
BMC COMPLEMENTARY MEDICINE AND THERAPIES (2021)
Click Chemistry-Based Synthesis of New 1-formyl-naphthalen-2-yloxymethyl-1,2,3-triazoles, Anticancer Screening and 2D-NMR Studies
Gautam Kumar Dhuda et al.
ANALYTICAL CHEMISTRY LETTERS (2021)
Synthesis and biological evaluation of indazole derivatives as anti-cancer agents
Wei Wei et al.
RSC ADVANCES (2021)
Target-Driven Design of a Coumarinyl Chalcone Scaffold Based Novel EF2 Kinase Inhibitor Suppresses Breast Cancer Growth In Vivo
Ferah Comert Onder et al.
ACS PHARMACOLOGY & TRANSLATIONAL SCIENCE (2021)
Identifying novel sphingosine kinase 1 inhibitors as therapeutics against breast cancer
Faez Iqbal Khan et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2020)
Synthesis and Biological Evaluation of New Naphthoquinones Derivatives
El-Mahdi Ourhzif et al.
CURRENT ORGANIC SYNTHESIS (2020)
One-pot synthesis and biological evaluation of novel 4-[3-fluoro-4-(morpholin-4-yl)]phenyl-1H-1,2,3-triazole derivatives as potent antibacterial and anticancer agents
Sirassu Narsimha et al.
JOURNAL OF HETEROCYCLIC CHEMISTRY (2020)
Discovery of Lonafarnib-Like Compounds: Pharmacophore Modeling and Molecular Dynamics Studies
Shailima Rampogu et al.
ACS OMEGA (2020)
Synthesis, characterization, molecular docking, and biological activities of coumarin-1,2,3-triazole-acetamide hybrid derivatives
Nima Sepehri et al.
ARCHIV DER PHARMAZIE (2020)
Structure-activity relationship studies and bioactivity evaluation of 1,2,3-triazole containing analogues as a selective sphingosine kinase-2 inhibitors
Vijai Kumar Reddy Tangadanchu et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2020)
Identification of Sphingosine Kinase-1 Inhibitors from Bioactive Natural Products Targeting Cancer Therapy
Deeba Shamim Jairajpuri et al.
ACS OMEGA (2020)
Recent advances in the synthesis of fluorinated compounds via an aryne intermediate
Matiur Rahman et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2020)
Fluorine-Containing Drugs Approved by the FDA in 2018
Haibo Mei et al.
CHEMISTRY-A EUROPEAN JOURNAL (2019)
PRODRUGS FOR NITROREDUCTASE BASED CANCER THERAPY-2: Novel amide/Ntr combinations targeting PC3 cancer cells
Tugba Gungor et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2019)
Synthesis of novel (R)-4-fluorophenyl-1H-1,2,3-triazoles: A new class of α-glucosidase inhibitors
Satya Kumar Avula et al.
BIOORGANIC CHEMISTRY (2019)
Synthesis and biological evaluation of pyrazole linked benzothiazole-β-naphthol derivatives as topoisomerase I inhibitors with DNA binding ability
Burri Nagaraju et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2019)
Vitamin C Inhibits Triple-Negative Breast Cancer Metastasis by Affecting the Expression of YAP1 and Synaptopodin 2
Liping Gan et al.
NUTRIENTS (2019)
Evaluation of binding and inhibition mechanism of dietary phytochemicals with sphingosine kinase 1: Towards targeted anticancer therapy
Preeti Gupta et al.
SCIENTIFIC REPORTS (2019)
Synthesis of some novel pyridine compounds containing bis-1,2,4-triazole/thiosemicarbazide moiety and investigation of their antioxidant properties, carbonic anhydrase, and acetylcholinesterase enzymes inhibition profiles
Nilufer Bulut et al.
JOURNAL OF BIOCHEMICAL AND MOLECULAR TOXICOLOGY (2018)
Thymoquinone inhibits cell proliferation, migration, and invasion by regulating the elongation factor 2 kinase (eEF-2K) signaling axis in triple-negative breast cancer
Nashwa Kabil et al.
BREAST CANCER RESEARCH AND TREATMENT (2018)
Identification of a Small Molecule That Selectively Inhibits ERG-Positive Cancer Cell Growth
Ahmed A. Mohamed et al.
CANCER RESEARCH (2018)
Synthesis, crystal structure and antimicrobial potential of some fluorinated chalcone-1,2,3-triazole conjugates
Pinki Yadav et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2018)
Annulation-Induced Cascade Transformation of 5-Iodo-1,2,3-triazoles to 2-(1-Aminoalkyl)benzoxazoles
Yury N. Kotovshchikov et al.
ORGANIC LETTERS (2018)
Triple-negative breast cancer: is there a treatment on the horizon?
Hui Yao et al.
ONCOTARGET (2017)
Synthesis, characterization and anti cancer activity of some fluorinated 3,6-diaryl-[1,2,4] triazolo[3,4-b] [1,3,4] thiadiazoles
Deepak Chowrasia et al.
ARABIAN JOURNAL OF CHEMISTRY (2017)
Microbial degradation of fluorinated drugs: biochemical pathways, impacts on the environment and potential applications
Cormac D. Murphy
APPLIED MICROBIOLOGY AND BIOTECHNOLOGY (2016)
Next Generation of Fluorine-Containing Pharmaceuticals, Compounds Currently in Phase II-III Clinical Trials of Major Pharmaceutical Companies: New Structural Trends and Therapeutic Areas
Yu Zhou et al.
CHEMICAL REVIEWS (2016)
Polyfluorinated Ethanes as Versatile Fluorinated C2-Building Blocks for Organic Synthesis
Valentine G. Nenajdenko et al.
CHEMICAL REVIEWS (2015)
Potent efficacy of metronomic topotecan and pazopanib combination therapy in preclinical models of primary or late stage metastatic triple-negative breast cancer
Teresa Di Desidero et al.
ONCOTARGET (2015)
A convergent synthesis of alkyne-azide cycloaddition derivatives of 4-α,β-2-propyne podophyllotoxin depicting potent cytotoxic activity
Mahesh K. Zilla et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Sirtuin inhibitors as anticancer agents
Jing Hu et al.
FUTURE MEDICINAL CHEMISTRY (2014)
Protein and ligand preparation: parameters, protocols, and influence on virtual screening enrichments
G. Madhavi Sastry et al.
JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN (2013)
Current and emerging targeted therapies for metastatic breast cancer
Edith A. Perez et al.
CANCER (2012)
Pharmacological significance of triazole scaffold
Rajeev Kharb et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2011)
Click chemistry to probe Hsp90: Synthesis and evaluation of a series of triazole-containing novobiocin analogues
Laura B. Peterson et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2010)
Membranes in Balance: Mechanisms of Sphingolipid Homeostasis
David K. Breslow et al.
MOLECULAR CELL (2010)
Epik:: a software program for pK a prediction and protonation state generation for drug-like molecules
John C. Shelley et al.
JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN (2007)
Synthesis of 1,2,3,12a,12b-hexahydrocyclopropa-[1,2-d]benzo[f]pyrrolo[1,2-b]isoquinolin-5,7-dione related to Duocarmycins and Anthramycin
A Venkatram et al.
JOURNAL OF HETEROCYCLIC CHEMISTRY (2005)
Glide: A new approach for rapid, accurate docking and scoring. 1. Method and assessment of docking accuracy
RA Friesner et al.
JOURNAL OF MEDICINAL CHEMISTRY (2004)