Related references
Note: Only part of the references are listed.CYX-5, a G-protein biassed MOP receptor agonist, DOP receptor antagonist and KOP receptor agonist, evokes constipation but not respiratory depression relative to morphine in rats
Mohammad Zafar Imam et al.
PHARMACOLOGICAL REPORTS (2023)
Intracerebroventricular administration of CYX-6, a potent μ-opioid receptor agonist, a δ- and κ-opioid receptor antagonist and a biased ligand at μ, δ & κ-opioid receptors, evokes antinociception with minimal constipation and respiratory depression in rats in contrast to morphine
Mohammad Zafar Imam et al.
EUROPEAN JOURNAL OF PHARMACOLOGY (2020)
Retrospective assessment of rat liver microsomal stability at NCATS: data and QSAR models
Vishal B. Siramshetty et al.
SCIENTIFIC REPORTS (2020)
[Dmt1]DALDA analogues modified with tyrosine analogues at position 1
Yunxin Cai et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2016)
In Vitro Metabolic Stability and in Vivo Biodistribution of 3-Methyl-4-furoxancarbaldehyde Using PET Imaging in Rats
Adam B. Pippin et al.
ACS MEDICINAL CHEMISTRY LETTERS (2016)
The dipeptidyl peptidase IV (CD26, EC 3 4 14 5) inhibitor vildagliptin is a potent antihyperalgesic in rats by promoting endomorphin-2 generation in the spinal cord
Kornel Kiraly et al.
EUROPEAN JOURNAL OF PHARMACOLOGY (2011)
Design, Synthesis and Pharmacological Characterization of Endomorphin Analogues with Non-Cyclic Amino Acid Residues in Position 2
Renata Perlikowska et al.
BASIC & CLINICAL PHARMACOLOGY & TOXICOLOGY (2010)
Biological activity of endomorphin and [Dmt1] endomorphin analogs with six-membered proline surrogates in position 2
Renata Perlikowska et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2009)
Synthesis and biological activity of endomorphin-2 analogs incorporating piperidine-2-, 3- or 4-carboxylic acids instead of proline in position 2
Renata Staniszewska et al.
CHEMICAL BIOLOGY & DRUG DESIGN (2008)
Enzymatic degradation of endomorphins
Anna Janecka et al.
PEPTIDES (2008)
Degradation of endomorphin-2 at the supraspinal level in mice is initiated by dipeptidyl peptidase IV:: an in vitro and in vivo study
C Sakurada et al.
BIOCHEMICAL PHARMACOLOGY (2003)
Share Paper
