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BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2013)
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Kamaldeep Paul et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2013)
Synthesis, structure-activity relationship and biological evaluation of 2,4,5-trisubstituted pyrimidine CDK inhibitors as potential anti-tumour agents
Hao Shao et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2013)
Identification and characterization of novel indole based small molecules as anticancer agents through SIRT1 inhibition
Naveen Panathur et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2013)
Design and synthesis of novel 1,2,3-triazole-dithiocarbamate hybrids as potential anticancer agents
Ying-Chao Duan et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2013)
Design, modeling, synthesis and biological activity evaluation of camptothecin-linked platinum anticancer agents
Raffaella Cincinelli et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2013)
Advances in the development of hybrid anticancer drugs
Sebastien Fortin et al.
EXPERT OPINION ON DRUG DISCOVERY (2013)
Development of N-Hydroxycinnamamide-Based Histone Deacetylase Inhibitors with an Indole-Containing Cap Group
Yingjie Zhang et al.
ACS MEDICINAL CHEMISTRY LETTERS (2013)
Design and synthesis of benzo[c,d]indolone-pyrrolobenzodiazepine conjugates as potential anticancer agents
Ahmed Kamal et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2012)
New derivatives of 11-methyl-6-[2-(dimethylamino)ethyl]-6H-indolo[2,3-b]quinoline as cytotoxic DNA topoisomerase II inhibitors
Wojciech Luniewski et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2012)
Design, synthesis and cytotoxic activities of novel hybrid compounds between 2-phenylbenzofuran and imidazole
Xiao-Dong Yang et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2012)
Hybrids of privileged structures benzothiazoles and pyrrolo[2,1-c] [1,4] benzodiazepin-5-one, and diversity-oriented synthesis of benzothiazoles
D. Subhas Bose et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2012)
Regulation of EMT by TGFβ in cancer
Carl-Henrik Heldin et al.
FEBS LETTERS (2012)
Antitumor Platinum(II) Complexes Containing Platinum-Based Moieties of Present Platinum Drugs and Furoxan Groups as Nitric Oxide Donors: Synthesis, DNA Interaction, and Cytotoxicity
Jian Zhao et al.
INORGANIC CHEMISTRY (2012)
Synthesis and cytotoxicity studies of bifunctional hybrids of nitrogen mustards with potential enzymes inhibitors based on melamine framework
Beata Kolesinska et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2012)
Synthesis, Aqueous Reactivity, and Biological Evaluation of Carboxylic Acid Ester-Functionalized Platinum-Acridine Hybrid Anticancer Agents
Leigh A. Graham et al.
JOURNAL OF MEDICINAL CHEMISTRY (2012)
One-pot synthesis and antiproliferative evaluation of pyrazolo[3,4-d]pyrimidine derivatives
Yu-Ying Huang et al.
TETRAHEDRON (2012)
Synthesis and cytotoxic activities of novel hybrid compounds of imidazole scaffold-based 2-substituted benzofurans
Wen-Jian Song et al.
RSC ADVANCES (2012)
Resveratrol Sensitizes Acute Myelogenous Leukemia Cells to Histone Deacetylase Inhibitors through Reactive Oxygen Species-Mediated Activation of the Extrinsic Apoptotic Pathway
Alae Yaseen et al.
MOLECULAR PHARMACOLOGY (2012)
Hybrid Molecules Incorporating Natural Products: Applications in Cancer Therapy, Neurodegenerative Disorders and Beyond
M. Decker
CURRENT MEDICINAL CHEMISTRY (2011)
Antineoplastic activity of the thiazolo[5,4-b]quinoline derivative D3CLP in K-562 cells is mediated through effector caspases activation
Ignacio Gonzalez-Sanchez et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2011)
Synthesis of novel alkyltriazole tagged pyrido[2,3-d]pyrimidine derivatives and their anticancer activity
C. Kurumurthy et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2011)
Synthesis and antitumor activity of new sulfonamide derivatives of thiadiazolo [3,2-a]pyrimidines
Nadia S. El-Sayed et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2011)
Ferrocene-indole hybrids for cancer and malaria therapy
Josefina Quirante et al.
JOURNAL OF ORGANOMETALLIC CHEMISTRY (2011)
Biological importance of imidazole nucleus in the new millennium
Balasubramanian Narasimhan et al.
MEDICINAL CHEMISTRY RESEARCH (2011)
EGFR Tyrosine Kinase Inhibitors Activate Autophagy as a Cytoprotective Response in Human Lung Cancer Cells
Weidong Han et al.
PLOS ONE (2011)
Promise and challenges in drug discovery and development of hybrid anticancer drugs
Lalji K. Gediya et al.
EXPERT OPINION ON DRUG DISCOVERY (2009)
Current status of cediranib: the rapid development of a novel anti-angiogenic therapy
Colin R. Lindsay et al.
FUTURE ONCOLOGY (2009)
Oral small-molecule tyrosine kinase inhibitor midostaurin (PKC412) inhibits growth and induces megakaryocytic differentiation in human leukemia cells
Yu-Chuen Huang et al.
TOXICOLOGY IN VITRO (2009)
Antitumor effect of the histone deacetylase inhibitor LAQ824 in combination with 13-cis-retinoic acid in human malignant melanoma
Yukihiko Kato et al.
MOLECULAR CANCER THERAPEUTICS (2007)
Transient exposure of mammary tumors to PD184352 and UCN-01 causes tumor cell death in vivo and prolonged suppression of tumor regrowth
W Hawkins et al.
CANCER BIOLOGY & THERAPY (2005)