Related references
Note: Only part of the references are listed.Copper-Catalyzed Three-Component Cascade Annulation for Divergent Syntheses of Imidazoles and Dihydroimidazoles
Gaochen Xu et al.
ORGANIC LETTERS (2022)
Discovery of 1-Amino-1H-imidazole-5-carboxamide Derivatives as Highly Selective, Covalent Bruton's Tyrosine Kinase (BTK) Inhibitors
Chunhua Ma et al.
JOURNAL OF MEDICINAL CHEMISTRY (2021)
Discovery of Ethyl Ketone-Based Highly Selective HDACs 1, 2, 3 Inhibitors for HIV Latency Reactivation with Minimum Cellular Potency Serum Shift and Reduced hERG Activity
Wensheng Yu et al.
JOURNAL OF MEDICINAL CHEMISTRY (2021)
Rhodium-Catalyzed Denitrogenative Diazole-Triazole Coupling toward Aza-Bridged Structures and Imidazole-Based Chelating Ligands
Julia O. Strelnikova et al.
ORGANIC LETTERS (2021)
Y Discovery of Novel Acetamide-Based Heme Oxygenase-1 Inhibitors with Potent In Vitro Antiproliferative Activity
Antonino N. Fallica et al.
JOURNAL OF MEDICINAL CHEMISTRY (2021)
Iodine-Mediated Cyclization of Enamines to Imidazole-4-Carboxylic Derivatives with Sequential Removal of Nitrogen Atoms from TMSN3
Peng Gao et al.
JOURNAL OF ORGANIC CHEMISTRY (2021)
Multicomponent Cascade Reaction of 3-Formylchromones: Highly Selective Synthesis of Functionalized 9-Azabicyclo[3.3.1]nonane Derivatives
Ying-Gang Duan et al.
ORGANIC LETTERS (2021)
2-Imidazole as a Substitute for the Electrophilic Group Gives Highly Potent Prolyl Oligopeptidase Inhibitors
Henri T. Patsi et al.
ACS MEDICINAL CHEMISTRY LETTERS (2021)
Multi-component cascade reaction of 3-formylchromones: highly selective synthesis of 4,5-dihydro-[4,5′-bipyrimidin]-6(1H)-one derivatives
Li Chen et al.
CHEMICAL COMMUNICATIONS (2021)
Multicomponent cascade reactions of HKAs: synthesis of highly functionalized 5H-chromeno[4,3-d]pyrimidines
Yun-Xiang Fan et al.
ORGANIC CHEMISTRY FRONTIERS (2021)
Recent advances in multi-component reactions and their mechanistic insights: a triennium review
Stephy Elza John et al.
ORGANIC CHEMISTRY FRONTIERS (2021)
Employing TosMIC as a C1N1 Two-Atom Synthon in Imidazole Synthesis by Neighboring Group Assistance Strategy
Xiao Geng et al.
ORGANIC LETTERS (2020)
Palladium-Catalyzed Four-Component Carbonylative Cyclization Reaction of Trifluoroacetimidoyl Chlorides, Propargyl Amines, and Diaryliodonium Salts: Access to Trifluoromethyl-Containing Trisubstituted Imidazoles
Zhengkai Chen et al.
ORGANIC LETTERS (2020)
Cu(II)/lodine(III) Oxide Dimerization of Heterocyclic Ketene Aminals: Tandem TEMPO Oxidation for the Highly Selective Synthesis of Functionalized 2H-Pyrrolo[1,2-a]imidazol-7(3H)-ones
Kun Li et al.
ORGANIC LETTERS (2020)
An environmentally benign cascade reaction of chromone-3-carboxaldehydes with ethyl 2-(pyridine-2-yl)acetate derivatives for highly site-selective synthesis of quinolizines and quinolizinium salts in water
Li Chen et al.
GREEN CHEMISTRY (2020)
Silver-catalyzed cascade reactions of 3-cyanochromone with 1,1-enediamines: synthesis of highly functionalized 2-(pyridin-3-yl)-chromeno[2,3-d]pyrimidines
Qiang Xiao et al.
ORGANIC CHEMISTRY FRONTIERS (2020)
Cascade reaction of isatins with nitro-substituted enamines: highly selective synthesis of functionalized (Z)-3-(1-(arylamino)-2-oxoarylidene)indolin-2-ones
Cong-Hai Zhang et al.
CHEMICAL COMMUNICATIONS (2020)
Metal-Free C-B Bond Cleavage: An Acid Catalyzed Three-Component Reaction Construction of Imidazole-Containing Triarylmethanes
Changcheng Wang et al.
ORGANIC LETTERS (2019)
Recent advances in heterogeneous catalysts for the synthesis of imidazole derivatives
Nagaraju Kerru et al.
SYNTHETIC COMMUNICATIONS (2019)
Development of DNA-Compatible Van Leusen Three-Component Imidazole Synthesis
Stefanie N. Geigle et al.
ORGANIC LETTERS (2019)
Base-Promoted Nitrile-Alkyne.Dbmino-Type Cyclilatioti: A Gelieral Method to Trisubstituted ImidazoleS
Qiang Wang et al.
ORGANIC LETTERS (2019)
Organocatalytic diastereoselective [3+2] cyclization of MBH carbonates with dinucleophiles: synthesis of bicyclic imidazoline derivatives that inhibit MDM2-p53 interaction
Hong-Ping Zhu et al.
CHEMICAL COMMUNICATIONS (2019)
Discovery and Preclinical Development of IIIM-290, an Orally Active Potent Cyclin-Dependent Kinase Inhibitor
Sandip B. Bharate et al.
JOURNAL OF MEDICINAL CHEMISTRY (2018)
Three-Component Site-Selective Synthesis of Highly Substituted 5H-Chromeno-[4,3-b]pyridines
Cong-Hai Zhang et al.
JOURNAL OF ORGANIC CHEMISTRY (2018)
A Novel Naphthyridine Derivative, 3u, Induces Necroptosis at Low Concentrations and Apoptosis at High Concentrations in Human Melanoma A375 Cells
Qinghong Kong et al.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (2018)
An efficient and eco-friendly synthesis of 2-pyridones and functionalized azaxanthone frameworks via indium triflate catalyzed domino reaction
N. Poomathi et al.
GREEN CHEMISTRY (2017)
Chromone as a Privileged Scaffold in Drug Discovery: Recent Advances
Joana Reis et al.
JOURNAL OF MEDICINAL CHEMISTRY (2017)
A Direct Cycloaminative Approach to Imidazole Derivatives via Dual C-H Functionalization
Sagar Arepally et al.
ORGANIC LETTERS (2017)
Synthesis of Benzoaryl-5-yl(2-hydroxyphenyl)methanones via Photoinduced Rearrangement of (E)-3-Arylvinyl-4H-chromen-4-ones
Jinming Fang et al.
ORGANIC LETTERS (2017)
Metal-Free Cascade Approach toward Polysubstituted Indolizines from Chromone-Based Michael Acceptors
Thomas Lepitre et al.
ORGANIC LETTERS (2017)
Three-component reactions of isocyanoacetates, amines and 3-formylchromones initiated by an unexpected aza-Michael addition
Jia-Yu Liao et al.
CHEMICAL COMMUNICATIONS (2017)
Regioselective construction of diverse and multifunctionalized 2-hydroxybenzophenones for sun protection by indium(III)-catalyzed benzannulation
Hongyun Cai et al.
CHEMICAL COMMUNICATIONS (2016)
Specific Synergist for Neonicotinoid Insecticides: IPPA08, a cis-Neonicotinoid Compound with a Unique Oxabridged Substructure
Haibo Bao et al.
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY (2016)
Enantioselective synthesis of (-)-chloramphenicol via silver-catalysed asymmetric isocyanoacetate aldol reaction
Allegra Franchino et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2016)
Eco-friendly synthesis of diverse and valuable 2-pyridones by catalyst- and solvent-free thermal multicomponent domino reaction
Tej Narayan Poudel et al.
GREEN CHEMISTRY (2015)
Discovery of (R)-8-(1-(3,5-Difluorophenylamino)ethyl)-N,N-dimethy12-morpholino-4-oxo-4H-chromene-6-carboxamide (AZD8186): A Potent and Selective Inhibitor of PI3Kβ and P13Kδ for the Treatment of PTEN-Deficient Cancers
Bernard Barlaam et al.
JOURNAL OF MEDICINAL CHEMISTRY (2015)
A cation-directed two-component cascade approach to enantioenriched pyrroloindolines
Jamie R. Wolstenhulme et al.
CHEMICAL COMMUNICATIONS (2014)
A Photochemical One-Pot Three-Component Synthesis of Tetrasubstituted Imidazoles
Stefan Pusch et al.
ORGANIC LETTERS (2014)
NIR-fluorescent coumarin-fused BODIPY dyes with large Stokes shifts
Andrei Y. Bochkov et al.
CHEMICAL COMMUNICATIONS (2013)
Synthesis and Cancer Stem Cell-Based Activity of Substituted 5-Morpholino-7H-thieno[3,2-b]pyran-7-ones Designed as Next Generation PI3K Inhibitors
Guillermo A. Morales et al.
JOURNAL OF MEDICINAL CHEMISTRY (2013)
Copper-Catalyzed Oxidative Diamination of Terminal Alkynes by Amidines: Synthesis of 1,2,4-Trisubstituted Imidazoles
Jihui Li et al.
ORGANIC LETTERS (2013)
Four-Component Cascade Heteroannulation of Heterocyclic Ketene Aminals: Synthesis of Functionalized Tetrahydroimidazo[1,2-a]pyridine Derivatives
Ming Li et al.
JOURNAL OF ORGANIC CHEMISTRY (2012)
Three-Component Domino Reactions for Selective Formation of Indeno[1,2-b]indole Derivatives
Bo Jiang et al.
ORGANIC LETTERS (2012)
Catalyst-Free Preparation of 1,2,4,5-Tetrasubstituted Imidazoles from a Novel Unexpected Domino Reaction of 2-Azido Acrylates and Nitrones
Bao Hu et al.
ORGANIC LETTERS (2011)
One-Pot Electrochemical Synthesis of Fused Indole Derivatives Containing Active Hydroxyl Groups in Aqueous Medium
Cheng-Chu Zeng et al.
JOURNAL OF ORGANIC CHEMISTRY (2009)
Characterization of structurally distinct, isoform-selective phosphoinositide 3′-kinase inhibitors in combination with radiation in the treatment of glioblastoma
Jack S. Chen et al.
MOLECULAR CANCER THERAPEUTICS (2008)
Enantioselective nonsteroidal aromatase inhibitors identified through a Multidisciplinary medicinal chemistry approach
A Cavalli et al.
JOURNAL OF MEDICINAL CHEMISTRY (2005)
Synthesis of trisubstituted imidazoles by palladium-catalyzed cyclization of O-pentafluorobenzoylamidoximes:: Application to amino acid mimetics with a C-terminal imidazole
S Zaman et al.
ORGANIC LETTERS (2005)
Efficient synthesis of imidazoles from aldehydes and 1,2-diketones using microwave irradiation
SE Wolkenberg et al.
ORGANIC LETTERS (2004)
Tetrasubstituted imidazole inhibitors of cytokine release: Probing substituents in the N-1 position
SA Laufer et al.
JOURNAL OF MEDICINAL CHEMISTRY (2004)
Synthesis and antiviral evaluation of polyhalogenated imidazole nucleosides:: Dimensional analogues of 2,5,6-trichloro-1-(β-D-ribofuranosyl)benzimidazole
TC Chien et al.
JOURNAL OF MEDICINAL CHEMISTRY (2004)
Development of potent non-carbohydrate imidazole-based small molecule selectin inhibitors with antiinflammatory activity
DH Slee et al.
JOURNAL OF MEDICINAL CHEMISTRY (2001)
New inhibitors of p38 kinase
JC Boehm et al.
EXPERT OPINION ON THERAPEUTIC PATENTS (2000)
Share Paper
