4.6 Article

Biological and Cheminformatics Studies of Newly Designed Triazole Based Derivatives as Potent Inhibitors against Mushroom Tyrosinase

Related references

Note: Only part of the references are listed.
Article Biochemistry & Molecular Biology

Novel 1,2,4-triazole analogues as mushroom tyrosinase inhibitors: synthesis, kinetic mechanism, cytotoxicity and computational studies

Balasaheb D. Vanjare et al.

Summary: A novel series of mushroom tyrosinase inhibitors with 1,2,4-triazole as the fundamental skeleton was created in this study. Compound 9k showed significantly higher activity compared to the standard drug. Cytotoxicity experiments, molecular docking, and dynamic simulation studies were conducted to evaluate the efficacy and mechanism of action of the most effective compounds.

MOLECULAR DIVERSITY (2021)

Review Biochemistry & Molecular Biology

A comprehensive review on tyrosinase inhibitors

Samaneh Zolghadri et al.

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2019)

Article Biochemistry & Molecular Biology

Investigation of tyrosinase inhibition by some 1,2,4 triazole derivative compounds: in vitro and in silico mechanisms

Elif Ayazoglu Demir et al.

TURKISH JOURNAL OF BIOCHEMISTRY-TURK BIYOKIMYA DERGISI (2019)

Article Mathematical & Computational Biology

Exploration of Novel Human Tyrosinase Inhibitors by Molecular Modeling, Docking and Simulation Studies

Mubashir Hassan et al.

INTERDISCIPLINARY SCIENCES-COMPUTATIONAL LIFE SCIENCES (2018)

Article Mathematical & Computational Biology

Molecular Docking and Dynamic Simulation of AZD3293 and Solanezumab Effects Against BACE1 to Treat Alzheimer's Disease

Mubashir Hassan et al.

FRONTIERS IN COMPUTATIONAL NEUROSCIENCE (2018)

Article Chemistry, Medicinal

Development of highly potent melanogenesis inhibitor by in vitro, in vivo and computational studies

Qamar Abbas et al.

DRUG DESIGN DEVELOPMENT AND THERAPY (2017)

Article Biochemistry & Molecular Biology

Synthesis, Bioevaluation and Molecular Dynamic Simulation Studies of Dexibuprofen-Antioxidant Mutual Prodrugs

Zaman Ashraf et al.

INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (2016)

Editorial Material Dermatology

Melanin Transfer: The Keratinocytes Are More than Gluttons

Cedric Delevoye

JOURNAL OF INVESTIGATIVE DERMATOLOGY (2014)

Article Dermatology

Mechanisms regulating melanogenesis*

Inês Ferreira dos Santos Videira et al.

ANAIS BRASILEIROS DE DERMATOLOGIA (2013)

Review Oncology

Cellular and molecular mechanisms controlling the migration of melanocytes and melanoma cells

Jacky Bonaventure et al.

PIGMENT CELL & MELANOMA RESEARCH (2013)

Article Biochemistry & Molecular Biology

Knowledge-Based, Central Nervous System (CNS) Lead Selection and Lead Optimization for CNS Drug Discovery

Arup K. Ghose et al.

ACS CHEMICAL NEUROSCIENCE (2012)

Article Biochemical Research Methods

Bacterial tyrosinases: old enzymes with new relevance to biotechnology

Michael Fairhead et al.

NEW BIOTECHNOLOGY (2012)

Article Chemistry, Medicinal

Molecular properties prediction, synthesis and antimicrobial activity of some newer oxadiazole derivatives

Mohammed Afroz Bakht et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2010)

Article Physics, Applied

Antitumor Effect of Plasma Treatment on U87 Glioma Xenografts: Preliminary Results

Marc Vandamme et al.

PLASMA PROCESSES AND POLYMERS (2010)

Article Biochemistry & Molecular Biology

MolProbity: all-atom contacts and structure validation for proteins and nucleic acids

Ian W. Davis et al.

NUCLEIC ACIDS RESEARCH (2007)

Review Multidisciplinary Sciences

Melanocyte biology and skin pigmentation

Jennifer Y. Lin et al.

NATURE (2007)

Article Chemistry, Multidisciplinary

UCSF chimera - A visualization system for exploratory research and analysis

EF Pettersen et al.

JOURNAL OF COMPUTATIONAL CHEMISTRY (2004)

Article Biochemistry & Molecular Biology

VADAR: a web server for quantitative evaluation of protein structure quality

L Willard et al.

NUCLEIC ACIDS RESEARCH (2003)

Article Biochemistry & Molecular Biology

Structure validation by Cα geometry:: φ,ψ and Cβ deviation

SC Lovell et al.

PROTEINS-STRUCTURE FUNCTION AND GENETICS (2003)

Review Cell Biology

Keratinocyte-melanocyte interactions during melanosome transfer

M Seiberg

PIGMENT CELL RESEARCH (2001)