Related references
Note: Only part of the references are listed.The G-Protein-Coupled Estrogen Receptor (GPER) Regulates Trimethylation of Histone H3 at Lysine 4 and Represses Migration and Proliferation of Ovarian Cancer Cells In Vitro
Nan Han et al.
CELLS (2021)
Phase 1 trial of a novel, first-in-class G protein-coupled estrogen receptor (GPER) agonist, LNS8801, in patients with advanced or recurrent treatment-refractory solid malignancies.
Carolyn Muller et al.
JOURNAL OF CLINICAL ONCOLOGY (2021)
G Protein-Coupled Estrogen Receptor Agonist G-1 Inhibits Mantle Cell Lymphoma Growth in Preclinical Models
Lixia Zhou et al.
FRONTIERS IN ONCOLOGY (2021)
Plasma membrane expression of G protein-coupled estrogen receptor (GPER)/G protein-coupled receptor 30 (GPR30) is associated with worse outcome in metachronous contralateral breast cancer
Julia Tutzauer et al.
PLOS ONE (2020)
Pharmacologic Activation of the G Protein-Coupled Estrogen Receptor Inhibits Pancreatic Ductal Adenocarcinoma
Christopher A. Natale et al.
CELLULAR AND MOLECULAR GASTROENTEROLOGY AND HEPATOLOGY (2020)
Reciprocality Between Estrogen Biology and Calcium Signaling in the Cardiovascular System
Quang-Kim Tran
FRONTIERS IN ENDOCRINOLOGY (2020)
Mitochondria as emerging targets for therapies against Tcell acute lymphoblastic leukemia
Miguel Olivas-Aguirre et al.
JOURNAL OF LEUKOCYTE BIOLOGY (2019)
The Peptide ERα17p Is a GPER Inverse Agonist that Exerts Antiproliferative Effects in Breast Cancer Cells
Rosamaria Lappano et al.
CELLS (2019)
G-Protein-Coupled Estrogen Receptor (GPER)-Specific Agonist G1 Induces ER Stress Leading to Cell Death in MCF-7 Cells
Diep-Khanh Ho Vo et al.
BIOMOLECULES (2019)
Expression and Effects of Ligand-activated Estrogen Receptors in Chronic Lymphocytic Leukemia
Mohammad Sharif Hasni et al.
ANTICANCER RESEARCH (2019)
G Protein-Coupled Estrogen Receptor: A Potential Therapeutic Target in Cancer
Shen Xu et al.
FRONTIERS IN ENDOCRINOLOGY (2019)
G-Protein Coupled Estrogen Receptor in Breast Cancer
Li-Han Hsu et al.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (2019)
Tamoxifen induces toxicity, causes autophagy, and partially reverses dexamethasone resistance in Jurkat T cells
Liliana Torres-Lopez et al.
JOURNAL OF LEUKOCYTE BIOLOGY (2019)
Understanding of ROS-Inducing Strategy in Anticancer Therapy
Su Ji Kim et al.
OXIDATIVE MEDICINE AND CELLULAR LONGEVITY (2019)
Estrogen Signaling in ERα-Negative Breast Cancer: ERβ and GPER
Rainer Girgert et al.
FRONTIERS IN ENDOCRINOLOGY (2019)
Activation of the G Protein-Coupled Estrogen Receptor Elicits Store Calcium Release and Phosphorylation of the Mu-Opioid Receptors in the Human Neuroblastoma SH-SY5Y Cells
Xiaowei Ding et al.
FRONTIERS IN NEUROSCIENCE (2019)
Role of G Protein-Coupled Estrogen Receptor in Cancer Progression
Joohee Jung
TOXICOLOGICAL RESEARCH (2019)
G protein-coupled estrogen receptor-1 agonist induces chemotherapeutic effect via ER stress signaling in gastric cancer
Seon-Jin Lee et al.
BMB REPORTS (2019)
T cell acute lymphoblastic leukemia (T-ALL): New insights into the cellular origins and infiltration mechanisms common and unique among hematologic malignancies
Eduardo Vadillo et al.
BLOOD REVIEWS (2018)
(-)-Epicatechin stimulates mitochondrial biogenesis and cell growth in C2C12 myotubes via the G-protein coupled estrogen receptor
Aldo Moreno-Ulloa et al.
EUROPEAN JOURNAL OF PHARMACOLOGY (2018)
Rab22A recruits BLOC-1 and BLOC-2 to promote the biogenesis of recycling endosomes
Saurabh Shakya et al.
EMBO REPORTS (2018)
The emerging role of estrogen in B cell malignancies
Eleni-Eirini Ladikou et al.
LEUKEMIA & LYMPHOMA (2017)
Epigenetic down regulation of G protein-coupled estrogen receptor (GPER) functions as a tumor suppressor in colorectal cancer
Qiao Liu et al.
MOLECULAR CANCER (2017)
G-1 Inhibits Breast Cancer Cell Growth via Targeting Colchicine-Binding Site of Tubulin to Interfere with Microtubule Assembly
Xiangmin Lv et al.
MOLECULAR CANCER THERAPEUTICS (2017)
GPER is involved in the regulation of the estrogen-metabolizing CYP1B1 enzyme in breast cancer
Francesca Cirillo et al.
ONCOTARGET (2017)
Inter-dependent apical microtubule and actin dynamics orchestrate centrosome retention and neuronal delamination
Ioannis Kasioulis et al.
ELIFE (2017)
The activation of the G protein-coupled estrogen receptor (GPER) inhibits the proliferation of mouse melanoma K1735-M2 cells
Mariana P. C. Ribeiro et al.
CHEMICO-BIOLOGICAL INTERACTIONS (2017)
Role of GPR30 in estrogen-induced prostate epithelial apoptosis and benign prostatic hyperplasia
Deng-Liang Yang et al.
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS (2017)
T-cell acute lymphoblastic leukemia
Elizabeth A. Raetz et al.
HEMATOLOGY-AMERICAN SOCIETY OF HEMATOLOGY EDUCATION PROGRAM (2016)
Regulation of hematopoietic progenitors by estrogens as a basis for new antileukemic strategies
Abel Sanchez-Aguilera et al.
MOLECULAR & CELLULAR ONCOLOGY (2016)
Activation of G-protein coupled estrogen receptor inhibits the proliferation of cervical cancer cells via sustained activation of ERK1/2
Qiong Zhang et al.
CELL BIOCHEMISTRY AND FUNCTION (2015)
Estrogen receptors regulate innate immune cells and signaling pathways
Susan Kovats
CELLULAR IMMUNOLOGY (2015)
G protein-coupled estrogen receptor 1 agonist G-1 induces cell cycle arrest in the mitotic phase, leading to apoptosis in endometriosis
Taisuke Mori et al.
FERTILITY AND STERILITY (2015)
The G protein-coupled estrogen receptor 1 (GPER-1) contributes to the proliferation and survival of mantle cell lymphoma cells
Martina Rudelius et al.
HAEMATOLOGICA (2015)
Receptors, G proteins, and integration of calcium signalling
Thomas Gudermann et al.
JOURNAL OF MOLECULAR MEDICINE-JMM (2015)
G protein-coupled estrogen receptor-mediated effects on cytosolic calcium and nanomechanics in brain microvascular endothelial cells
Joseph B. Altmann et al.
JOURNAL OF NEUROCHEMISTRY (2015)
Oxidative/antioxidative enzyme-mediated antiproliferative and proapoptotic effects of the GPER1 agonist G-1 on lung cancer cells
Akif Hakan Kurt et al.
ONCOLOGY LETTERS (2015)
GPER agonist G-1 decreases adrenocortical carcinoma (ACC) cell growth in vitro and in vivo
Adele Chimento et al.
ONCOTARGET (2015)
The G protein-coupled estrogen receptor 1 (GPER-1) contributes to the proliferation and survival of mantle cell lymphoma cells
Martina Rudelius et al.
HAEMATOLOGICA (2015)
The GPER Agonist G-1 Induces Mitotic Arrest and Apoptosis in Human Vascular Smooth Muscle Cells Independent of GPER
Yu Gui et al.
JOURNAL OF CELLULAR PHYSIOLOGY (2015)
Lack of G protein-coupled estrogen receptor (GPER) in the plasma membrane is associated with excellent long-term prognosis in breast cancer
Martin Sjostrom et al.
BREAST CANCER RESEARCH AND TREATMENT (2014)
GPER-mediated proliferation and estradiol production in breast cancer-associated fibroblasts
Haojun Luo et al.
ENDOCRINE-RELATED CANCER (2014)
Recent developments in tubulin polymerization inhibitors: An overview
Ramandeep Kaur et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
GPER functions as a tumor suppressor in triple-negative breast cancer cells
Christine Weissenborn et al.
JOURNAL OF CANCER RESEARCH AND CLINICAL ONCOLOGY (2014)
Targeting Microtubules by Natural Agents for Cancer Therapy
Eiman Mukhtar et al.
MOLECULAR CANCER THERAPEUTICS (2014)
The activation of G protein-coupled receptor 30 (GPR30) inhibits proliferation of estrogen receptor-negative breast cancer cells in vitro and in vivo
W. Wei et al.
CELL DEATH & DISEASE (2014)
G15, a GPR30 antagonist, induces apoptosis and autophagy in human oral squamous carcinoma cells
Li-Yuan Bai et al.
CHEMICO-BIOLOGICAL INTERACTIONS (2013)
Bradycardic effects mediated by activation of G protein-coupled estrogen receptor in rat nucleus ambiguus
G. Cristina Brailoiu et al.
EXPERIMENTAL PHYSIOLOGY (2013)
Histone deacetylase inhibitors down-regulate G-protein-coupled estrogen receptor and the GPER-antagonist G-15 inhibits proliferation in endometriotic cells
Patrick Imesch et al.
FERTILITY AND STERILITY (2013)
Estrogen receptor α and β in the normal immune system and in lymphoid malignancies
Konstantin Yakimchuk et al.
MOLECULAR AND CELLULAR ENDOCRINOLOGY (2013)
The G-protein-coupled estrogen receptor agonist G-1 suppresses proliferation of ovarian cancer cells by blocking tubulin polymerization
C. Wang et al.
CELL DEATH & DISEASE (2013)
Enhanced expression of G-protein coupled estrogen receptor (GPER/GPR30) in lung cancer
Venkatakrishna Rao Jala et al.
BMC CANCER (2012)
17β-Estradiol Rapidly Activates Calcium Release from Intracellular Stores via the GPR30 Pathway and MAPK Phosphorylation in Osteocyte-Like MLO-Y4 Cells
Jian Ren et al.
CALCIFIED TISSUE INTERNATIONAL (2012)
The G protein-coupled oestrogen receptor 1 agonist G-1 disrupts endothelial cell microtubule structure in a receptor-independent manner
Anders Holm et al.
MOLECULAR AND CELLULAR BIOCHEMISTRY (2012)
Estrogen and Signaling in the Cells of Immune System
Deena Khan et al.
ADVANCES IN NEUROIMMUNE BIOLOGY (2012)
Identification of a GPER/GPR30 antagonist with improved estrogen receptor counterselectivity
Megan K. Dennis et al.
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY (2011)
The G-protein-coupled estrogen receptor GPER in health and disease
Eric R. Prossnitz et al.
NATURE REVIEWS ENDOCRINOLOGY (2011)
Drugs That Target Dynamic Microtubules: A New Molecular Perspective
Richard A. Stanton et al.
MEDICINAL RESEARCH REVIEWS (2011)
Influence of Charge on Cell Permeability and Tumor Imaging of GPR30-Targeted 111In-Labeled Nonsteroidal Imaging Agents
Tapan K. Nayak et al.
ACS CHEMICAL BIOLOGY (2010)
The G Protein-Coupled Receptor GPR30 Inhibits Proliferation of Estrogen Receptor-Positive Breast Cancer Cells
Eric A. Ariazi et al.
CANCER RESEARCH (2010)
Attenuation of CXCR4 Responses by CCL18 in Acute Lymphocytic Leukemia B Cells
J. Catusse et al.
JOURNAL OF CELLULAR PHYSIOLOGY (2010)
In vivo effects of a GPR30 antagonist
Megan K. Dennis et al.
NATURE CHEMICAL BIOLOGY (2009)
G protein-coupled receptor 30 (GPR30) mediates gene expression changes and growth response to 17β-estradiol and selective GPR30 ligand G-1 in ovarian cancer cells
Lidia Albanito et al.
CANCER RESEARCH (2007)
Monitoring lymphocyte proliferation in vitro and in vivo with the intracellular fluorescent dye carboxyfluorescein diacetate succinimidyl ester
Ben J. C. Quah et al.
NATURE PROTOCOLS (2007)
Distribution of GPR30, a seven membrane-spanning estrogen receptor, in primary breast cancer and its association with clinicopathologic determinants of tumor progression
Edward J. Filardo et al.
CLINICAL CANCER RESEARCH (2006)
Virtual and biomolecular screening converge on a selective agonist for GPR30
CG Bologa et al.
NATURE CHEMICAL BIOLOGY (2006)
A transmembrane intracellular estrogen receptor mediates rapid cell signaling
CM Revankar et al.
SCIENCE (2005)
17-β-estradiol alters Jurkat lymphocyte cell cycling and induces apoptosis through suppression of Bcl-2 and cyclin A
JK Jenkins et al.
INTERNATIONAL IMMUNOPHARMACOLOGY (2001)