Related references
Note: Only part of the references are listed.α-Cyclodextrin Encapsulation of Bicyclo[1.1.1]pentane Derivatives: a Storable Feedstock for Preparation of [1.1.1]Propellane
Tadafumi Matsunaga et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2021)
Large-Scale Synthesis and Modifications of Bicyclo[1.1.1]pentane-1,3-dicarboxylic Acid (BCP)
Vasyl Ripenko et al.
JOURNAL OF ORGANIC CHEMISTRY (2021)
1,2-Difunctionalized bicyclo[1.1.1]pentanes: Long-sought-after mimetics for ortho/ meta-substituted arenes
Jin-Xin Zhao et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2021)
Radical-mediated sulfonyl alkynylation, allylation, and cyanation of propellane
Zhen Wu et al.
CHEMICAL COMMUNICATIONS (2021)
Strain-release 2-azaallyl anion addition/borylation of [1.1.1]propellane: synthesis and functionalization of benzylamine bicyclo[1.1.1]pentyl boronates
Russell A. Shelp et al.
CHEMICAL SCIENCE (2021)
Development of Scalable Routes to 1-Bicyclo[1.1.1]pentylpyrazoles
Cayetana Zarate et al.
ORGANIC PROCESS RESEARCH & DEVELOPMENT (2021)
Silaboration of [1.1.1]Propellane: A Storable Feedstock for Bicyclo[1.1.1]pentane Derivatives
Masaki Kondo et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2020)
1,3-Difunctionalizations of [1.1.1]Propellane via 1,2-Metallate Rearrangements of Boronate Complexes
Songjie Yu et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2020)
Divergent Strain-Release Amino-Functionalization of [1.1.1]Propellane with Electrophilic Nitrogen-Radicals
Ji Hye Kim et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2020)
Copper-mediated synthesis of drug-like bicyclopentanes
Xiaheng Zhang et al.
NATURE (2020)
Continuous Flow-Enabled Synthesis of Bench-Stable Bicyclo[1.1.1]pentane Trifluoroborate Salts and Their Utilization in Metallaphotoredox Cross-Couplings
Michael D. VanHeyst et al.
ORGANIC LETTERS (2020)
Strain release - an old tool for new transformations
Joanna Turkowska et al.
CHEMICAL COMMUNICATIONS (2020)
A General Copper-Catalyzed Synthesis of Ynamides from 1,2-Dichloroenannides
Steven J. Mansfield et al.
ORGANIC LETTERS (2019)
Reactions of 2-Aryl-1,3-Dithianes and [1.1.1]Propellane
Nisalak Trongsiriwat et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2019)
Aminoalkylation of [1.1.1]Propellane Enables Direct Access to High-Value 3-Alkylbicyclo[1.1.1]pentan-1-amines
Jonathan M. E. Hughes et al.
ORGANIC LETTERS (2019)
Nonconjugated Hydrocarbons as Rigid-Linear Motifs: Isosteres for Material Sciences and Bioorganic and Medicinal Chemistry
Gemma M. Locke et al.
CHEMISTRY-A EUROPEAN JOURNAL (2019)
Recent Advances in the Synthetic Chemistry of Bicyclo[1.1.1]pentane
Junichiro Kanazawa et al.
SYNLETT (2019)
Saturated bioisosteres of benzene: where to go next?
Pavel K. Mykhailiuk
ORGANIC & BIOMOLECULAR CHEMISTRY (2019)
Synthesis and applications of highly functionalized 1-halo-3-substituted bicyclo[1.1.1]pentanes
Dimitri F. J. Caputo et al.
CHEMICAL SCIENCE (2018)
Synthesis of BCP Benzylamines From 2-Azaallyl Anions and [1.1.1]Propellane
Russell A. Shelp et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2018)
Investigation of a Bicyclo[1.1.1]pentane as a Phenyl Replacement within an LpPLA(2) Inhibitor
Nicholas D. Measom et al.
ACS MEDICINAL CHEMISTRY LETTERS (2017)
Bicyclo[1.1.1]pentane-Derived Building Blocks for Click Chemistry
Serhii O. Kokhan et al.
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2017)
Radical Multicomponent Carboamination of [1.1.1]Propellane
Junichiro Kanazawa et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2017)
Photoinduced decarboxylative borylation of carboxylic acids
Alexander Fawcett et al.
SCIENCE (2017)
Toward Resolving the Resveratrol Conundrum: Synthesis and in Vivo Pharmacokinetic Evaluation of BCP-Resveratrol
Yi Ling Goh et al.
ACS MEDICINAL CHEMISTRY LETTERS (2017)
Propellanes-From a Chemical Curiosity to Explosive Materials and Natural Products
Alicia M. Dilmac et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2017)
Improving Nonspecific Binding and Solubility: Bicycloalkyl Groups and Cubanes as para-Phenyl Bioisosteres
Yves P. Auberson et al.
CHEMMEDCHEM (2017)
Synthesis and Biopharmaceutical Evaluation of Imatinib Analogues Featuring Unusual Structural Motifs
Kyriacos C. Nicolaou et al.
CHEMMEDCHEM (2016)
Design, Synthesis, and Application of an Optimized Monofluorinated Aliphatic Label for Peptide Studies by Solid-State 19F NMR Spectroscopy
Serhii O. Kokhan et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2016)
Design and Performance Validation of a Conductively Heated Sealed-Vessel Reactor for Organic Synthesis
David Obermayer et al.
JOURNAL OF ORGANIC CHEMISTRY (2016)
Expedient synthesis of 3-phenylbicyclo[1.1.1]pentan-1-amine via metal-free homolytic aromatic alkylation of benzene
Navanita T. Thirumoorthi et al.
CHEMICAL COMMUNICATIONS (2015)
A New Route to Bicyclo[1.1.1]pentan-1-amine from 1-Azido-3-iodobicyclo[1.1.1]pentane
Yi Ling Goh et al.
ORGANIC LETTERS (2014)
Crystalline Arrays of Pairs of Molecular Rotors: Correlated Motion, Rotational Barriers, and Space-Inversion Symmetry Breaking Due to Conformational Mutations
Cyprien Lemouchi et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2013)
Escape from Flatland 2: complexity and promiscuity
Frank Lovering
MEDCHEMCOMM (2013)
A walk around the A(3)-coupling
Vsevolod A. Peshkov et al.
CHEMICAL SOCIETY REVIEWS (2012)
1,3-Diethynylbicyclo[1.1.1]pentane, a Useful Molecular Building Block
Jiri Kaleta et al.
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2012)
Application of the Bicyclo[1.1.1]pentane Motif as a Nonclassical Phenyl Ring Bioisostere in the Design of a Potent and Orally Active γ-Secretase Inhibitor
Antonia F. Stepan et al.
JOURNAL OF MEDICINAL CHEMISTRY (2012)
Synopsis of Some Recent Tactical Application of Bioisosteres in Drug Design
Nicholas A. Meanwell
JOURNAL OF MEDICINAL CHEMISTRY (2011)
Escape from Flatland: Increasing Saturation as an Approach to Improving Clinical Success
Frank Lovering et al.
JOURNAL OF MEDICINAL CHEMISTRY (2009)
Synthesis of a chiral amino acid with bicyclo[1.1.1]pentane moiety and its incorporation into linear and cyclic antimicrobial peptides
Stephan Pritz et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2007)
Synthesis and biological evaluation of (2S)-and (2R)-2-(3′-phosphonobicyclo[1.1.1]pentyl)glycines as novel group III selective metabotropic glutamate receptor ligands
Rosanna Filosa et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2006)
Synthesis and preliminary biological evaluation of 2′-substituted 2-(3′-carboxybicyclo[1.1.1]-pentyl)glycine derivatives as group I selective metabotropic glutamate receptor ligands
Roberto Pellicciari et al.
CHEMMEDCHEM (2006)
Conformationally rigid trifluoromethyl-substituted alpha-amino acid designed for peptide structure analysis by solid-state F-19 NMR spectroscopy
Pavel K. Mikhailiuk et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2006)
3-aminobicyclo[1.1.1]pentane-1-carboxylic acid derivatives:: Synthesis and incorporation into peptides
M Pätzel et al.
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2004)
Synthesis and structure of trigonal and tetragonal connectors for a tinkertoy construction set
PFH Schwab et al.
JOURNAL OF ORGANIC CHEMISTRY (2002)
Share Paper
