Related references
Note: Only part of the references are listed.Preclinical candidate for the treatment of visceral leishmaniasis that acts through proteasome inhibition
Susan Wyllie et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2019)
Improvement of Asparagine Ethylenediamines as Anti-malarial Plasmodium-Selective Proteasome Inhibitors
Wenhu Zhan et al.
JOURNAL OF MEDICINAL CHEMISTRY (2019)
The proteasome as a target for protozoan parasites
Stanley C. Xie et al.
EXPERT OPINION ON THERAPEUTIC TARGETS (2019)
Identification of Small Molecules Disrupting the Ubiquitin Proteasome System in Malaria
Lydia Mata-Cantero et al.
ACS INFECTIOUS DISEASES (2019)
Ubiquitin Proteasome System as a Potential Drug Target for Malaria
Pedro H. Scarpelli Pereira et al.
CURRENT TOPICS IN MEDICINAL CHEMISTRY (2018)
Antimalarial proteasome inhibitor reveals collateral sensitivity from intersubunit interactions and fitness cost of resistance
Laura A. Kirkman et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2018)
Defining the Determinants of Specificity of Plasmodium Proteasome Inhibitors
Euna Yoo et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2018)
Artemisinin kills malaria parasites by damaging proteins and inhibiting the proteasome
Jessica L. Bridgford et al.
NATURE COMMUNICATIONS (2018)
Target Validation and Identification of Novel Boronate Inhibitors of the Plasmodium falciparum Proteasome
Stanley C. Xie et al.
JOURNAL OF MEDICINAL CHEMISTRY (2018)
Use of Calculated Physicochemical Properties to Enhance Quantitative Response When Using Charged Aerosol Detection
Max W. Robinson et al.
ANALYTICAL CHEMISTRY (2017)
Development of a Novel High-Density [3H] Hypoxanthine Scintillation Proximity Assay To Assess Plasmodium falciparum Growth
Cristina de Cozar et al.
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY (2016)
New insights into host-parasite ubiquitin proteome dynamics in P. falciparum infected red blood cells using a TUBEs-MS approach
Lydia Mata-Cantero et al.
JOURNAL OF PROTEOMICS (2016)
Structure- and function-based design of Plasmodium-selective proteasome inhibitors
Hao Li et al.
NATURE (2016)
The inhibition mechanism of human 20S proteasomes enables next-generation inhibitor design
Jil Schrader et al.
SCIENCE (2016)
Development of two novel high-throughput assays to quantify ubiquitylated proteins in cell lysates: application to screening of new anti-malarials
Lydia Mata-Cantero et al.
MALARIA JOURNAL (2015)
Identifying rapidly parasiticidal anti-malarial drugs using a simple and reliable in vitro parasite viability fast assay
Maria Linares et al.
MALARIA JOURNAL (2015)
Targeting the Cell Stress Response of Plasmodium falciparum to Overcome Artemisinin Resistance
Con Dogovski et al.
PLOS BIOLOGY (2015)
Assessing Subunit Dependency of the Plasmodium Proteasome Using Small Molecule Inhibitors and Active Site Probes
Hao Li et al.
ACS CHEMICAL BIOLOGY (2014)
A Male and Female Gametocyte Functional Viability Assay To Identify Biologically Relevant Malaria Transmission-Blocking Drugs
A. Ruecker et al.
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY (2014)
Optimal assay design for determining the in vitro sensitivity of ring stage Plasmodium falciparum to artemisinins
Stanley C. Xie et al.
INTERNATIONAL JOURNAL FOR PARASITOLOGY (2014)
Fueling Open-Source Drug Discovery: 177 Small-Molecule Leads against Tuberculosis
Lluis Ballell et al.
CHEMMEDCHEM (2013)
Validation of the Proteasome as a Therapeutic Target in Plasmodium Using an Epoxyketone Inhibitor with Parasite-Specific Toxicity
Hao Li et al.
CHEMISTRY & BIOLOGY (2012)
Getting physical in drug discovery II: the impact of chromatographic hydrophobicity measurements and aromaticity
Robert J. Young et al.
DRUG DISCOVERY TODAY (2011)
Thousands of chemical starting points for antimalarial lead identification
Francisco-Javier Gamo et al.
NATURE (2010)
Assembly, structure, and function of the 26S proteasome
Lynn Bedford et al.
TRENDS IN CELL BIOLOGY (2010)
Selective Inhibitor of Proteasome's Caspase-like Sites Sensitizes Cells to Specific Inhibition of Chymotrypsin-like Sites
Matthew Britton et al.
CHEMISTRY & BIOLOGY (2009)
Artemisinin and a series of novel endoperoxide Antimalarials exert early effects on digestive vacuole morphology
Maria del Pilar Crespo et al.
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY (2008)
An overview of drug combination analysis with isobolograms
Ronald J. Tallarida
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2006)
Crystal structure of the boronic acid-based proteasome inhibitor bortezomib in complex with the yeast 20S proteasome
M Groll et al.
STRUCTURE (2006)