4.6 Article

GZD824 overcomes FGFR1-V561F/M mutant resistance in vitro and in vivo

Related references

Note: Only part of the references are listed.
Review Pharmacology & Pharmacy

Overview of the clinical use of erdafitinib as a treatment option for the metastatic urothelial carcinoma: where do we stand

Alberto D'Angelo et al.

EXPERT REVIEW OF CLINICAL PHARMACOLOGY (2020)

Review Oncology

Fibroblast growth factor receptors as treatment targets in clinical oncology

Masaru Katoh

NATURE REVIEWS CLINICAL ONCOLOGY (2019)

Article Chemistry, Multidisciplinary

LY2874455 potently inhibits FGFR gatekeeper mutants and overcomes mutation-based resistance

Daichao Wu et al.

CHEMICAL COMMUNICATIONS (2018)

Article Chemistry, Medicinal

2-Aminopyrimidine Derivatives as New Selective Fibroblast Growth Factor Receptor 4 (FGFR4) Inhibitors

Cheng Mo et al.

ACS MEDICINAL CHEMISTRY LETTERS (2017)

Article Chemistry, Medicinal

Insight into resistance mechanisms of AZD4547 and E3810 to FGFR1 gatekeeper mutation via theoretical study

Donglou Liang et al.

DRUG DESIGN DEVELOPMENT AND THERAPY (2017)

Review Oncology

Advances and challenges in targeting FGFR signalling in cancer

Irina S. Babina et al.

NATURE REVIEWS CANCER (2017)

Article Clinical Neurology

Germline and somatic FGFR1 abnormalities in dysembryoplastic neuroepithelial tumors

Barbara Rivera et al.

ACTA NEUROPATHOLOGICA (2016)

Review Medicine, Research & Experimental

FGFR inhibitors: Effects on cancer cells, tumor microenvironment and whole-body homeostasis (Review)

Masaru Katoh

INTERNATIONAL JOURNAL OF MOLECULAR MEDICINE (2016)

Article Multidisciplinary Sciences

Development of covalent inhibitors that can overcome resistance to first-generation FGFR kinase inhibitors

Li Tan et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2014)

Letter Hematology

The 8p11 myeloproliferative syndrome owing to rare FGFR1OP2-FGFR1 fusion

Masahiro Onozawa et al.

EUROPEAN JOURNAL OF HAEMATOLOGY (2011)