Related references
Note: Only part of the references are listed.Synthesis and In Vitro Cytotoxicity Evaluation of Phenanthrene Linked 2,4-Thiazolidinediones as Potential Anticancer Agents
Upasana Yadav et al.
ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY (2021)
Phenothiazines Modified with the Pyridine Ring as Promising Anticancer Agents
Beata Morak-Mlodawska et al.
LIFE-BASEL (2021)
Oridonin and its derivatives for cancer treatment and overcoming therapeutic resistance
Xi Liu et al.
GENES & DISEASES (2021)
Structural Activity Relationship and Importance of Benzothiazole Derivatives in Medicinal Chemistry: A Comprehensive Review
Mahesh Bhat et al.
MINI-REVIEWS IN ORGANIC CHEMISTRY (2020)
Reliability of Click Chemistry on Drug Discovery: A Personal Account
Nagula Shankaraiah et al.
CHEMICAL RECORD (2020)
An Insight into the Synthesis and SAR of 2,4-Thiazolidinediones (2,4-TZD) as Multifunctional Scaffold: A Review
Navjot Singh Sethi et al.
MINI-REVIEWS IN MEDICINAL CHEMISTRY (2020)
Synthesis, Biological and Computational Evaluation of Novel 2,3-dihydro-2-aryl-4-(4-isobutylphenyl)-1,5-benzothiazepine Derivatives as Anticancer and Anti-EGFR Tyro-sine Kinase Agents
Afzal B. Shaik et al.
ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY (2020)
Synthesis and bioevaluation of new vascular-targeting and anti-angiogenic thieno[2,3-d]pyrimidin-4(3H)-ones
Madeleine Gold et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2020)
Design, synthesis, biological evaluation and molecular docking study of novel thieno[3,2-d]pyrimidine derivatives as potent FAK inhibitors
Ruifeng Wang et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2020)
Ferrocenes as new anticancer drug candidates: Determination of the mechanism of action
Hana Skoupilova et al.
EUROPEAN JOURNAL OF PHARMACOLOGY (2020)
The Design and Synthesis of Novel Phenothiazine Derivatives as Potential Cytotoxic Agents
Yepeng Luan et al.
LETTERS IN DRUG DESIGN & DISCOVERY (2020)
Benzothiazole derivatives as anticancer agents
Ali Irfan et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2020)
Novel cyanoacetamide integrated phenothiazines: Synthesis, characterization, computational studies and in vitro antioxidant and anticancer evaluations
Kannan Gokula Krishnan et al.
JOURNAL OF MOLECULAR STRUCTURE (2020)
The Smiles rearrangement in the syntheses of azaphenothiazines. Part I
Krystian Pluta et al.
JOURNAL OF MOLECULAR STRUCTURE (2020)
Synthesis, spectral characterization and antitumor activity of phenothiazine derivatives
Kasi Venkatesan et al.
JOURNAL OF HETEROCYCLIC CHEMISTRY (2020)
Design and Synthesis of 5-Morpholino-Thiophene-Indole/ Oxindole Hybrids as Cytotoxic Agents
Upasana Yadav et al.
CHEMISTRYSELECT (2020)
Sex-Specific Differences of Steroid Receptors Following Exposure to Environmentally Relevant Concentrations of Phenothiazine in Fundulus heteroclitus
John B. Chiari et al.
ARCHIVES OF ENVIRONMENTAL CONTAMINATION AND TOXICOLOGY (2020)
Evaluation of the Lipophilicity of New Anticancer 1,2,3-Triazole-Dipyridothiazine Hybrids Using RP TLC and Different Computational Methods
Beata Morak-Mlodawska et al.
PROCESSES (2020)
Screening and Molecular Docking of Novel Benzothiazole Derivatives as Potential Antimicrobial Agents
Mohamed A. Morsy et al.
ANTIBIOTICS-BASEL (2020)
Recent advances in the synthetic chemistry of 1,5-benzothiazepines: A minireview
Varsha Devi et al.
JOURNAL OF HETEROCYCLIC CHEMISTRY (2020)
A Review on Anticancer Activities of Thiophene and Its Analogs
Raghav Mishra et al.
MINI-REVIEWS IN MEDICINAL CHEMISTRY (2020)
Dual Action of Dipyridothiazine and Quinobenzothiazine Derivatives-Anticancer and Cholinesterase-Inhibiting Activity
Jakub Jonczyk et al.
MOLECULES (2020)
The Smiles rearrangement in the syntheses of azaphenothiazines. Part II. The review of the various types of phenyl azinyl and diazinyl sulfides undergoing this rearrangement
Krystian Pluta et al.
JOURNAL OF MOLECULAR STRUCTURE (2020)
Phenothiazine and amide-ornamented novel nitrogen heterocyclic hybrids: synthesis, biological and molecular docking studies
Ramar Sivaramakarthikeyan et al.
NEW JOURNAL OF CHEMISTRY (2020)
Construction of sulfur-containing moieties in the total synthesis of natural products
Nengzhong Wang et al.
NATURAL PRODUCT REPORTS (2020)
Colchicine-Binding Site Inhibitors from Chemistry to Clinic: A Review
Eavan C. McLoughlin et al.
PHARMACEUTICALS (2020)
Synthesis and anticancer activity of novel 3,6-disubstituted 1,2,4-triazolo-[3,4-b]-1,3, 4-thiadiazole derivatives
Georgios Charitos et al.
ARABIAN JOURNAL OF CHEMISTRY (2019)
Diverse Targeted Approaches to Battle Multidrug Resistance in Cancer
Nagula Shankaraiah et al.
CURRENT MEDICINAL CHEMISTRY (2019)
Oridonin-induced mitochondria-dependent apoptosis in esophageal cancer cells by inhibiting PI3K/AKT/mTOR and Ras/Raf pathways
Jin-Huan Jiang et al.
JOURNAL OF CELLULAR BIOCHEMISTRY (2019)
Novel thienopyrimidine derivatives as dual EGFR and VEGFR-2 inhibitors: design, synthesis, anticancer activity and effect on cell cycle profile
Aml E. -S. Mghwary et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2019)
Design, synthesis and anticancer activities of halogenated Phenstatin analogs as microtubule destabilizing agent
Shengquan Hu et al.
MEDICINAL CHEMISTRY RESEARCH (2019)
Thieno[2,3-d] pyrimidine as a promising scaffold in medicinal chemistry: Recent advances
Eslam M. H. Ali et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2019)
Synthesis of substituted biphenyl methylene indolinones as apoptosis inducers and tubulin polymerization inhibitors
Kavitha Donthiboina et al.
BIOORGANIC CHEMISTRY (2019)
Pyrazoles containing thiophene, thienopyrimidine and thienotriazolopyrimidine as COX-2 selective inhibitors: Design, synthesis, in vivo anti-inflammatory activity, docking and in silico chemo-informatic studies
Mai S. El-Shoukrofy et al.
BIOORGANIC CHEMISTRY (2019)
A conceptual review of rhodanine: current applications of antiviral drugs, anticancer and antimicrobial activities
Seyyed Mojtaba Mousavi et al.
ARTIFICIAL CELLS NANOMEDICINE AND BIOTECHNOLOGY (2019)
Novel Thienopyrimidine Derivative, RP-010, Induces β-Catenin Fragmentation and Is Efficacious against Prostate Cancer Cells
Haneen Amawi et al.
CANCERS (2019)
Evaluation of thioamides, thiolactams and thioureas as hydrogen sulfide (H2S) donors for lowering blood pressure
Ewelina Zaorska et al.
BIOORGANIC CHEMISTRY (2019)
Evaluation of angularly condensed diquinothiazines as potential anticancer agents
Malgorzata Jelen et al.
BIOORGANIC CHEMISTRY (2019)
Employing alpha-Diazocarbonyl Compound Chemistry in the Assembly of Medicinally Important Aryl(alkyl)thiolactam Scaffold
Darina Barkhatova et al.
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2019)
Lipophilicity estimation of anti-proliferative and anti-inflammatory 6-substituted 9-fluoroquino[3,2-b]benzo[1,4]thiazines
Malgorzata Jelen et al.
JOURNAL OF LIQUID CHROMATOGRAPHY & RELATED TECHNOLOGIES (2019)
Design, click synthesis, anticancer screening and docking studies of novel benzothiazole-1,2,3-triazoles appended with some bioactive benzofused heterocycles
Mohamed Reda Aouad et al.
JOURNAL OF MOLECULAR STRUCTURE (2019)
A review on anticancer potentials of benzothiazole derivatives
Nandini Pathak et al.
MINI-REVIEWS IN MEDICINAL CHEMISTRY (2019)
Recent advances of thiazole hybrids in biological applications
Mehmet Gumus et al.
FUTURE MEDICINAL CHEMISTRY (2019)
Role of sulphur-heterocycles in medicinal chemistry: An update
Shelly Pathania et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2019)
Pyrazolo-benzothiazole hybrids: Synthesis, anticancer properties and evaluation of antiangiogenic activity using in vitro VEGFR-2 kinase and in vivo transgenic zebrafish model
Velma Ganga Reddy et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2019)
Design, Synthesis, and Structural Characterization of Novel Diazaphenothiazines with 1,2,3-Triazole Substituents as Promising Antiproliferative Agents
Beata Morak-Mlodawska et al.
MOLECULES (2019)
Therapeutic advancement of benzothiazole derivatives in the last decennial period
Sana Tariq et al.
ARCHIV DER PHARMAZIE (2019)
Synthesis of Novel Analogs of Thieno[2,3-d] Pyrimidin-4(3H)-ones as Selective Inhibitors of Cancer Cell Growth
Sheng Zhang et al.
BIOMOLECULES (2019)
Synthesis, Anticancer Activity, and Apoptosis Induction of Novel 3,6-Diazaphenothiazines
Beata Morak-Mlodawska et al.
MOLECULES (2019)
Design and synthesis of DNA-intercalative naphthalimide-benzothiazole/cinnamide derivatives: cytotoxicity evaluation and topoisomerase-IIα inhibition
N. Sankara Rao et al.
MEDCHEMCOMM (2019)
The Prospective Value of Dopamine Receptors on Bio-Behavior of Tumor
Xu Wang et al.
JOURNAL OF CANCER (2019)
10H-1,9-diazaphenothiazine and its 10-derivatives: synthesis, characterisation and biological evaluation as potential anticancer agents
Beata Morak-Mlodawska et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2019)
Sulfamic acid promoted one-pot synthesis of phenanthrene fused-dihydrodibenzo-quinolinones: Anticancer activity, tubulin polymerization inhibition and apoptosis inducing studies
Niggula Praveen Kumar et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2018)
Synthesis of 1,2,4-triazole-linked urea/thiourea conjugates as cytotoxic and apoptosis inducing agents
Ramya Tokala et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2018)
Synthesis, biological evaluation and molecular modeling of novel thienopyrimidinone and triazolothienopyrimidinone derivatives as dual anti-inflammatory antimicrobial agents
Adnan A. Bekhit et al.
BIOORGANIC CHEMISTRY (2018)
Design and synthesis of thienopyrimidine urea derivatives with potential cytotoxic and pro-apoptotic activity against breast cancer cell line MCF-7
Eman F. Abdelhaleem et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2018)
Synthesis of podophyllotoxin linked β-carboline congeners as potential anticancer agents and DNA topoisomerase II inhibitors
Manda Sathish et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2018)
Synthesis, anticancer activity and mechanism of action of new thiazole derivatives
Temistocles Italo de Santana et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2018)
Microwave-assisted synthesis of γ-thiolactams from ethyl isocyanoacetate
Massimiliano Lamberto
HETEROCYCLIC COMMUNICATIONS (2018)
Lipophilicity of New Anticancer 1,6-and 3,6-diazaphenothiazines by of Use RP TLC and Different Computational Methods
Beata Morak-Mlodawska et al.
JOURNAL OF CHROMATOGRAPHIC SCIENCE (2018)
Synthesis, Antimicrobial, and Anticancer Activities of a New Series of Thieno[2,3-d] Pyrimidine Derivatives
Abdelreheem Abdelfatah Saddik et al.
JOURNAL OF HETEROCYCLIC CHEMISTRY (2018)
Synthesis of 1,4-Thiazepines
Yilmaz Kelgokmen et al.
JOURNAL OF ORGANIC CHEMISTRY (2018)
Synthesis and Preliminarily Cytotoxicity to A549, HCT116 and MCF-7 Cell Lines of Thieno[2,3-d]pyrimidine Derivatives containing Isoxazole Moiety
Jianping Yong et al.
LETTERS IN DRUG DESIGN & DISCOVERY (2018)
Antiproliferative Phenothiazine Hybrids as Novel Apoptosis Inducers against MCF-7 Breast Cancer
Jun-Xia Zhang et al.
MOLECULES (2018)
Role of Dopamine Receptors in the Anticancer Activity of ONC201
Christina Leah B. Kline et al.
NEOPLASIA (2018)
Synthesis and in vitro antitumor evaluation of some new thiophenes and thieno[2,3-d]pyrimidine derivatives
Mahasen M. Fouad et al.
BIOORGANIC CHEMISTRY (2018)
Thienopyrimidine-Chalcone Hybrid Molecules Inhibit Fas-Activated Serine/Threonine Kinase: An Approach To Ameliorate Antiproliferation in Human Breast Cancer Cells
Nashrah Sharif Khan et al.
MOLECULAR PHARMACEUTICS (2018)
Synthesis and in vitro cytotoxicity evaluation of β-carboline-linked 2,4-thiazolidinedione hybrids: potential DNA intercalation and apoptosis-inducing studies
Ramya Tokala et al.
NEW JOURNAL OF CHEMISTRY (2018)
Therapeutic importance of synthetic thiophene
Rashmi Shah et al.
CHEMISTRY CENTRAL JOURNAL (2018)
Canagliflozin Slows Progression of Renal Function Decline Independently of Glycemic Effects
Hiddo J. L. Heerspink et al.
JOURNAL OF THE AMERICAN SOCIETY OF NEPHROLOGY (2017)
Azaphenothiazines - promising phenothiazine derivatives. An insight into nomenclature, synthesis, structure elucidation and biological properties
Krystian Pluta et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2017)
Conventional and microwave-assisted synthesis of new 1H-benzimidazole-thiazolidinedione derivatives: A potential anticancer scaffold
Pankaj Sharma et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2017)
Therapeutic journey of 2,4-thiazolidinediones as a versatile scaffold: An insight into structure activity relationship
Mohd. Javed Naim et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2017)
Thienopyrimidine derivatives exert their anticancer efficacy via apoptosis induction, oxidative stress and mitotic catastrophe
Haneen Amawi et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2017)
Synthesis of substituted phenanthrene-9-benzimidazole conjugates: Cytotoxicity evaluation, and apoptosis inducing studies
Niggula Praveen Kumar et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2017)
Synthesis and anti-proliferative activity evaluation of novel benzo[d] [1,3] dioxoles-fused 1,4-thiazepines
Liqiang Wu et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2017)
Novel 2,4-thiazolidinediones: Synthesis, in vitro cytotoxic activity, and mechanistic investigation
Kamel Metwally et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2017)
An overview of benzo[b]thiophene-based medicinal chemistry
Rangappa S. Keri et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2017)
Design, synthesis and biological evaluations of N-Hydroxy thienopyrimidine-2,4-diones as inhibitors of HIV reverse transcriptase-associated RNase H
Jayakanth Kankanala et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2017)
Novel Thiazolo[5,4-b] phenothiazine Derivatives: Synthesis, Structural Characterization, and In Vitro Evaluation of Antiproliferative Activity against Human Leukaemia
Balazs Brem et al.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (2017)
N-acylhydrazones containing thiophene nucleus: a new anticancer class
Laura N. F. Cardoso et al.
MEDICINAL CHEMISTRY RESEARCH (2017)
Molecular diversity of phenothiazines: design and synthesis of phenothiazine-dithiocarbamate hybrids as potential cell cycle blockers
Dong-Jun Fu et al.
MOLECULAR DIVERSITY (2017)
New benzothiazole/benzoxazole-pyrazole hybrids with potential as COX inhibitors: design, synthesis and anticancer activity evaluation
Amany Belal et al.
RESEARCH ON CHEMICAL INTERMEDIATES (2017)
10H-3,6-Diazaphenothiazine induces G(2)/M phase cell cycle arrest and caspase-dependent apoptosis and inhibits cell invasion of A2780 ovarian carcinoma cells through the regulation of NF-kappa B and (BIRC6-XIAP) complexes
Jianxin Zhang et al.
DRUG DESIGN DEVELOPMENT AND THERAPY (2017)
Targeting DNA Minor Groove by Hybrid Molecules as Anticancer Agents
Shalini Nekkanti et al.
CURRENT MEDICINAL CHEMISTRY (2017)
Medicinal Attributes of Thienopyrimidine Based Scaffold Targeting Tyrosine Kinases and Their Potential Anticancer Activities
Amna Ghith et al.
ARCHIV DER PHARMAZIE (2017)
Design, synthesis and anticancer activity of N-(1-(4-(dibenzo[bf][1,4] thiazepin-11-yl)piperazin-1-yl)-1-oxo-3-phenylpropan-2-yl derivatives
Mura Reddy Gudisela et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2017)
Fas-activated serine/threonine kinase: Structure and function
Saurabha Srivastava et al.
GENE REPORTS (2017)
Synthesis of different heterocycles-linked chalcone conjugates as cytotoxic agents and tubulin polymerization inhibitors
Nagula Shankaraiah et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2017)
Design, synthesis, in silico and in vitro evaluation of thiophene derivatives: A potent tyrosine phosphatase 1B inhibitor and anticancer activity
Kali Charan Gulipalli et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2017)
FGFR a promising druggable target in cancer: Molecular biology and new drugs
Rut Porta et al.
CRITICAL REVIEWS IN ONCOLOGY HEMATOLOGY (2017)
Novel 2-phenyl-4,5,6,7-tetrahydro[b]benzothiophene analogues as selective COX-2 inhibitors: Design, synthesis, anti-inflammatory evaluation, and molecular docking studies
Chetan K. Khatri et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2017)
Identification of Novel Class of TriazoloThiadiazoles as Potent Inhibitors of Human Heparanase and their Anticancer Activity
C. P. Baburajeev et al.
BMC CANCER (2017)
Synthesis and anticancer and lipophilic properties of 10-dialkylaminobutynyl derivatives of 1,8-and 2,7-diazaphenothiazines
Beata Morak-Mlodawska et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2016)
1,3,4-Thiadiazole Based Anticancer Agents
Alireza Aliabadi
ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY (2016)
Synthesis and anticancer activity of novel 4-morpholino-7,8-dihydro-5H-thiopyrano[4,3-d]pyrimidine derivatives bearing chromone moiety
Chengyu Sun et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2016)
Novel aminoalkylated azaphenothiazines as potential inhibitors of T98G, H460 and SNU80 cancer cell lines in vitro
Khushbu Kushwaha et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2016)
Synthesis of new tricyclic thiolactams as potent antitumor agent for pancreatic cancer
Takuya Okada et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2016)
Ferrocenyl-nucleobase complexes: Synthesis, chemistry and applications
Konrad Kowalski
COORDINATION CHEMISTRY REVIEWS (2016)
Sulfur Containing Scaffolds in Drugs: Synthesis and Application in Medicinal Chemistry
Minghao Feng et al.
CURRENT TOPICS IN MEDICINAL CHEMISTRY (2016)
Synthesis, anticancer activity and photostability of novel 3-ethyl-2-mercapto-thieno[2,3-d]pyrimidin-4(3H)-ones
Anelia Ts Mavrova et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2016)
Synthesis and evaluation of bis-thiazole derivatives as new anticancer agents
Gulhan Turan-Zitouni et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2016)
Synthesis, binding assays, cytotoxic activity and docking studies of benzimidazole and benzothiophene derivatives with selective affinity for the CB2 cannabinoid receptor
Javier Romero-Parra et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2016)
Synthesis and biological evaluation of new benzimidazole-thiazolidinedione hybrids as potential cytotoxic and apoptosis inducing agents
Pankaj Sharma et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2016)
Synthesis and biological evaluation of D-ring fused 1,2,3-thiadiazole dehydroepiandrosterone derivatives as antitumor agents
Hai-Wei Cui et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2016)
Synthesis and biological evaluation of novel propargylquinobenzothiazines and their derivatives as potential antiproliferative, anti-inflammatory, and anticancer agents
Malgorzata Jelen et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2016)
3,6-Diazaphenothiazines as potential lead molecules - synthesis, characterization and anticancer activity
Beata Morak-Mlodawska et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2016)
Synthesis, spectroscopic structure identification, X-ray study and anticancer activities of new angularly fused quinobenzothiazines
K. Pluta et al.
JOURNAL OF MOLECULAR STRUCTURE (2016)
Synthesis, spectroscopic characterization, and anticancer activity of new 10-substituted 1,6-diazaphenothiazines
Beata Morak-Mlodawska et al.
MEDICINAL CHEMISTRY RESEARCH (2016)
Synthesis and In Vitro Antiproliferative Activity of Novel Phenyl Ring-Substituted 5-Alkyl-12(H)-quino[3,4-b][1,4]benzothiazineDerivatives
Andrzej Zieba et al.
MOLECULES (2016)
Discovery of Novel Tricyclic Thiazepine Derivatives as Anti-Drug Resistant Cancer Agents by Combining Diversity-Oriented Synthesis and Converging Screening Approach
Jinbao Xiang et al.
ACS COMBINATORIAL SCIENCE (2016)
One-pot synthesis and in-vitro anticancer evaluation of 5-(2′-indolyl)thiazoles
Buchi Reddy Vaddula et al.
SCIENTIFIC REPORTS (2016)
Synthesis and antiproliferative activity of diethyl 5-acetyl-4-methyl- 6-(2-fluorophenylimino)-6H-thiopyran-2,3-dicarboxylate (3TM)
Baghipour Tayebeh et al.
AFRICAN JOURNAL OF BIOTECHNOLOGY (2016)
Pharmacological exploitation of the phenothiazine antipsychotics to develop novel antitumor agents-A drug repurposing strategy
Chia-Hsien Wu et al.
SCIENTIFIC REPORTS (2016)
Recent Advances in the Chemistry and Biology of Benzothiazoles
Rupinder K. Gill et al.
ARCHIV DER PHARMAZIE (2015)
Design, synthesis and biological evaluation of N-phenylthieno[2,3-d]pyrimidin-4-amines as inhibitors of FGFR1
A. A. Gryshchenko et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2015)
Chrysin-benzothiazole conjugates as antioxidant and anticancer agents
Bhupendra M. Mistry et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2015)
One-pot synthesis of podophyllotoxin-thiourea congeners by employing NH2SO3H/NaI: Anticancer activity, DNA topoisomerase-II inhibition, and apoptosis inducing agents
Nagula Shankaraiah et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2015)
Synthesis and evaluation of benzosuberone embedded with 1,3,4-oxadiazole, 1,3,4-thiadiazole and 1,2,4-triazole moieties as new potential anti proliferative agents
Bandi Yadagiri et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2015)
Synthesis, in vitro anticancer and antimycobacterial evaluation of new 5-(2,5-dimethoxyphenyl)-1,3,4-thiadiazole-2-amino derivatives
Naveen Polkam et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2015)
Synthesis and Anticancer Activity of Some New Thiopyrano[2,3-d]thiazoles Incorporating Pyrazole Moiety
Nadia Hanafy Metwally et al.
CHEMICAL & PHARMACEUTICAL BULLETIN (2015)
Isavuconazonium: First Global Approval
Paul L. McCormack
DRUGS (2015)
Synthesis, anticancer activity and effects on cell cycle profile and apoptosis of novel thieno[2,3-d]pyrimidine and thieno[3,2-e] triazolo[4,3-c]pyrimidine derivatives
Manal M. Kandeel et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2015)
Synthesis, anticancer activity and molecular docking studies on a series of heterocyclic trans-cyanocombretastatin analogues as antitubulin agents
Narsimha Reddy Penthala et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2015)
Synthesis, antiproliferative activity, and in silico insights of new 3-benzoylamino-benzo[b]thiophene derivatives
Annamaria Martorana et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2015)
Ring fusion strategy for synthesis and lead optimization of sulfur-substituted anthra[1,2-c][1,2,5]thiadiazole-6,11-dione derivatives as promising scaffold of antitumor agents
Yu-Ru Lee et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2015)
Synthesis of thiophene-thiosemicarbazone derivatives and evaluation of their in vitro and in vivo antitumor activities
Jamerson Ferreira de Oliveira et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2015)
6-Substituted 9-fluoroquino[3,2-b]benzo[1,4]thiazines display strong antiproliferative and antitumor properties
Malgorzata Jelen et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2015)
1,3,4-Thiadiazoles: A potent multi targeted pharmacological scaffold
Saqlain Haider et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2015)
Therapeutic potential of benzothiazoles: a patent review (2010-2014)
Ahmed Kamal et al.
EXPERT OPINION ON THERAPEUTIC PATENTS (2015)
Quinonaphthothiazines, syntheses, structures and anticancer activities
M. Jelen et al.
JOURNAL OF MOLECULAR STRUCTURE (2015)
Synthesis and anticancer activity studies of ferrocenyl-thymine-3,6-dihydro-2H-thiopyranes - A new class of metallocene-nucleobase derivatives
Joanna Skiba et al.
JOURNAL OF ORGANOMETALLIC CHEMISTRY (2015)
Dabrafenib and trametinib versus dabrafenib and placebo for Val600 BRAF-mutant melanoma: a multicentre, double-blind, phase 3 randomised controlled trial
Georgina V. Long et al.
LANCET (2015)
Synthesis and Preliminary Biological Evaluation of New Heterocyclic Carboxamide Models
Kamal Sweidan et al.
LETTERS IN DRUG DESIGN & DISCOVERY (2015)
Synthesis and anticancer evaluation of 2-phenyl thiaolidinone substituted 2-phenyl benzothiazole-6-carboxylic acid derivatives
Padmavathi P. Prabhu et al.
JOURNAL OF SAUDI CHEMICAL SOCIETY (2015)
Estimation of the Lipophilicity of New Anticancer and Immunosuppressive 1,8-Diazaphenothiazine Derivatives
Beata Morak-Mlodawska et al.
JOURNAL OF CHROMATOGRAPHIC SCIENCE (2015)
Synthesis of quinoline/naphthalene-containing azaphenothiazines and their potent in vitro antioxidant properties
Malgorzata Jelen et al.
MEDICINAL CHEMISTRY RESEARCH (2015)
An efficient L-proline catalyzed synthesis of pyrazolo[3,4-e][1,4]thiazepine derivatives and their in vitro cytotoxicity studies
A. Srikanth et al.
MEDICINAL CHEMISTRY RESEARCH (2015)
Synthesis and selected immunological properties of 10-substituted 1,8-diazaphenothiazines
Beata Morak-Mlodawska et al.
MEDICINAL CHEMISTRY RESEARCH (2015)
Cancer multidrug resistance: mechanisms involved and strategies for circumvention using a drug delivery system
Golam Kibria et al.
ARCHIVES OF PHARMACAL RESEARCH (2014)
Synthesis and biological evaluation of podophyllotoxin congeners as tubulin polymerization inhibitors
Ahmed Kamal et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2014)
Design, synthesis, anticancer activity and docking studies of novel 4-morpholino-7,8-dihydro-5H-thiopyrano[4,3-d] pyrimidine derivatives as mTOR inhibitors
Wufu Zhu et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2014)
Synthesis and anticancer potential of benzothiazole linked phenylpyridopyrimidinones and their diones as mitochondrial apoptotic inducers
Ahmed Kamal et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2014)
Synthesis and anticancer evaluation of 3-aryl-6-phenylimidazo [2,1-b]thiazoles
Satish Koppireddi et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2014)
Design, synthesis and anticancer evaluation of tetrahydro-β-carboline-hydantoin hybrids
Nagula Shankaraiah et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2014)
Design, synthesis and biological evaluation of novel diphenylthiazole-based cyclooxygenase inhibitors as potential anticancer agents
Ahmed H. Abdelazeem et al.
BIOORGANIC CHEMISTRY (2014)
Synthesis and anticancer activity of (E)-2-benzothiazole hydrazones
Eric B. Lindgren et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Thiophene-3-carboxamide analogue of annonaceous acetogenins as antitumor drug lead
Naoto Kojima et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Anilides and quinolones with nitrogen-bearing substituents from benzothiophene and thienothiophene series: Synthesis, photochemical synthesis, cytostatic evaluation, 3D-derived QSAR analysis and DNA-binding properties
Maja Aleksic et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Studies on the synthetic and structural aspects of benzosuberones bearing 2, 4-thiazolidenone moiety as potential anti-cancer agents
Lingaiah Nagarapu et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Thiazolidine-2,4-diones as multi-targeted scaffold in medicinal chemistry: Potential anticancer agents
Vivek Asati et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Bifunctional ethyl 2-amino-4-methylthiazole-5-carboxylate derivatives: Synthesis and in vitro biological evaluation as antimicrobial and anticancer agents
Sherif A. F. Rostom et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Synthesis, in vitro anticancer evaluation and in silico studies of novel imidazo[2,1-b]thiazole derivatives bearing pyrazole moieties
Ahmed R. Ali et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Novel thiazole derivatives: a patent review (2008-2012. Part 2)
Alberto Leoni et al.
EXPERT OPINION ON THERAPEUTIC PATENTS (2014)
DETERMINATION OF THE LIPOPHILICITY PARAMETERS OF NEW ANTIPROLIFERATIVE 8-10-SUBSTITUTED QUINOBENZOTHIAZINES BY COMPUTATIONAL METHODS AND RP TLC
Malgorzata Jelen et al.
JOURNAL OF LIQUID CHROMATOGRAPHY & RELATED TECHNOLOGIES (2014)
Data-Mining for Sulfur and Fluorine: An Evaluation of Pharmaceuticals To Reveal Opportunities for Drug Design and Discovery
Elizabeth A. Ilardi et al.
JOURNAL OF MEDICINAL CHEMISTRY (2014)
Synthesis, in vitro anticancer activity and in silico study of new disubstituted thiazolidinedione derivatives
Moacyr Jesus Barreto de Melo Rego et al.
MEDICINAL CHEMISTRY RESEARCH (2014)
SKLB-163, a new benzothiazole-2-thiol derivative, exhibits potent anticancer activity by affecting RhoGDI/JNK-1 signaling pathway
X. Peng et al.
CELL DEATH & DISEASE (2014)
Brexpiprazole I: In Vitro and In Vivo Characterization of a Novel Serotonin-Dopamine Activity Modulator
Kenji Maeda et al.
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS (2014)
Synthesis and anti-angiogenic activity of benzothiazole, benzimidazole containing phthalimide derivatives
Shunmugam Nagarajan et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2013)
1,3,4-Thiadiazole and its Derivatives: A Review on Recent Progress in Biological Activities
Abhishek Kumar Jain et al.
CHEMICAL BIOLOGY & DRUG DESIGN (2013)
Thiadiazole-a Promising Structure in Medicinal Chemistry
Yijing Li et al.
CHEMMEDCHEM (2013)
Synthesis and cytotoxic evaluation of new colchicine derivatives bearing 1,3,4-thiadiazole moieties
Li-Hong Shen et al.
CHINESE CHEMICAL LETTERS (2013)
Synthesis, biological evaluation and molecular modeling studies of some novel thiazolidinediones with triazole ring
Yakaiah Chinthala et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2013)
Chiral 6,7-bis(hydroxymethyl)-1H,3H-pyrrolo[1,2-c]thiazoles with anti-breast cancer properties
Maria I. L. Soares et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2013)
New anticancer active and selective phenylene-bisbenzothiazoles: Synthesis, antiproliferative evaluation and DNA binding
Livio Racane et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2013)
Benzimidazole clubbed with triazolo-thiadiazoles and triazolo-thiadiazines: New anticancer agents
Asif Husain et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2013)
Synthesis and biological activity evaluation of 5-pyrazoline substituted 4-thiazolidinones
Dmytro Havrylyuk et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2013)
Synthesis, antimicrobial, antiquorum-sensing, antitumor and cytotoxic activities of new series of fused [1,3,4]thiadiazoles
Nadia S. El-Gohary et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2013)
Synthesis and selected immunological properties of substituted quino[3,2-b]benzo[1,4]thiazines
Malgorzata Jelen et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2013)
Synthesis of some new pyrazole-based 1,3-thiazoles and 1,3,4-thiadiazoles as anticancer agents
Kamal M. Dawood et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2013)
Medicinal significance of benzothiazole scaffold: an insight view
Prabodh Chander Sharma et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2013)
Discovery of Novel and Ligand-Efficient Inhibitors of Plasmodium falciparum and Plasmodium vivax N-Myristoyltransferase
Mark D. Rackham et al.
JOURNAL OF MEDICINAL CHEMISTRY (2013)
Novel Nitrogen-Enriched Oridonin Analogues with Thiazole-Fused A-Ring: Protecting Group-Free Synthesis, Enhanced Anticancer Profile, and Improved Aqueous Solubility
Chunyong Ding et al.
JOURNAL OF MEDICINAL CHEMISTRY (2013)
Synthesis and Biological Evaluation of 2-(Alkoxycarbonyl)-3-Anilinobenzo[b]thiophenes and Thieno[2,3-b]pyridines as New Potent Anticancer Agents
Romeo Romagnoli et al.
JOURNAL OF MEDICINAL CHEMISTRY (2013)
Pyrazolines: A Biological Review
Akranth Marella et al.
MINI-REVIEWS IN MEDICINAL CHEMISTRY (2013)
Synthesis and Biological Evaluation of Some Novel Thieno[2,3-d] pyrimidine Derivatives as Potential Anti-inflammatory and Analgesic Agents
Alaa El-Tombary et al.
Medicinal Chemistry (2013)
Synthesis and in vitro antiproliferative activity of novel 12(H)-quino[3,4-b][1,4]benzothiazine derivatives
Andrzej Zieba et al.
MEDICINAL CHEMISTRY RESEARCH (2013)
Synthesis and evaluation of a series of benzothiophene acrylonitrile analogs as anticancer agents
Narsimha Reddy Penthala et al.
MEDCHEMCOMM (2013)
A Drug Repositioning Approach Identifies Tricyclic Antidepressants as Inhibitors of Small Cell Lung Cancer and Other Neuroendocrine Tumors
Nadine S. Jahchan et al.
CANCER DISCOVERY (2013)
Synthesis and biological evaluation of 2-substituted-4-(3′,4′,5′-trimethoxyphenyl)-5-aryl thiazoles as anticancer agents
Romeo Romagnoli et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2012)
Synthesis and cytotoxic evaluation of thiourea and N-bis-benzothiazole derivatives: A novel class of cytotoxic agents
Ravindra M. Kumbhare et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2012)
Synthesis, characterization and biological evaluation of some novel 2,4-thiazolidinediones as potential cytotoxic, antimicrobial and antihyperglycemic agents
Vasudeva Rao Avupati et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2012)
Substituted thiazoles VII. Synthesis and antitumor activity of certain 2-(substituted amino)-4-phenyl-1,3-thiazole analogs
Ghada S. Hassan et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2012)
Efficacy and Safety of a 12-week Treatment with Twice-daily Aclidinium Bromide in COPD Patients (ACCORD COPD I)
Edward M. Kerwin et al.
COPD-JOURNAL OF CHRONIC OBSTRUCTIVE PULMONARY DISEASE (2012)
Antiproliferative Activity of Novel Derivative of Thiopyran on Breast and Colon Cancer Lines and DNA Binding
Mehdi Rajabi et al.
DNA AND CELL BIOLOGY (2012)
A series of 2-arylamino-5-(indolyl)-1,3,4-thiadiazoles as potent cytotoxic agents
Dalip Kumar et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2012)
Synthesis and biological evaluation of combretastatin-amidobenzothiazole conjugates as potential anticancer agents
Ahmed Kamal et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2012)
3,5-Disubstituted-thiazolidine-2,4-dione analogs as anticancer agents: Design, synthesis and biological characterization
Kai Liu et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2012)
2,6-Disubstituted imidazo[2,1-b][1,3,4]thiadiazoles: Search for anticancer agents
Malleshappa N. Noolvi et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2012)
Benzothiazoles: Search for anticancer agents
Malleshappa N. Noolvi et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2012)
Identification of new aminoacid amides containing the imidazo[2,1-b]benzothiazol-2-ylphenyl moiety as inhibitors of tumorigenesis by oncogenic Met signaling
Alessandro Furlan et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2012)
Novel Substituted Benzothiophene and Thienothiophene Carboxanilides and Quinolones: Synthesis, Photochemical Synthesis, DNA-Binding Properties, Antitumor Evaluation and 3D-Derived QSAR Analysis
Maja Aleksic et al.
JOURNAL OF MEDICINAL CHEMISTRY (2012)
10-(3′-Nitro-4′-pyridy1)-1,8-diazaphenothiazine as the double Smiles rearrangement product
Beata Morak-Mlodawska et al.
JOURNAL OF MOLECULAR STRUCTURE (2012)
Synthesis and Biological Evaluation of Novel Benzothiazole-2-thiol Derivatives as Potential Anticancer Agents
Xuan-Hong Shi et al.
MOLECULES (2012)
Synthesis and Anticancer Activity of Di(3-thienyl)methanol and Di(3-thienyl)methane
Nagendra Kumar Kaushik et al.
MOLECULES (2012)
MET: a promising anticancer therapeutic target
Solange Peters et al.
NATURE REVIEWS CLINICAL ONCOLOGY (2012)
New thiazolidinedione-5-acetic acid amide derivatives: synthesis, characterization and investigation of antimicrobial and cytotoxic properties
Shankar G. Alegaon et al.
MEDICINAL CHEMISTRY RESEARCH (2012)
Synthesis, antimicrobial, antioxidant, anti-inflammatory, and analgesic activities of some new 3-(2'-thienyl)pyrazole-based heterocycles
Bakr F. Abdel-Wahab et al.
MEDICINAL CHEMISTRY RESEARCH (2012)
Synthesis of new potential anticancer agents based on 4-thiazolidinone and oleanane scaffolds
Danylo Kaminskyy et al.
MEDICINAL CHEMISTRY RESEARCH (2012)
Antiproliferative Activity of Novel Thiopyran Analogs on MCF-7 Breast and HCT-15 Colon Cancer Cells: Synthesis, Cytotoxicity, Cell Cycle Analysis, and DNA-Binding
Fatemeh Tavakolinia et al.
NUCLEIC ACID THERAPEUTICS (2012)
An efficient one-pot synthesis of benzothiazolo-4 beta-anilino-podophyllotoxin congeners: DNA topoisomerase-II inhibition and anticancer activity
Ahmed Kamal et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2011)
One-pot synthesis and anticancer studies of 2-arylamino-5-aryl-1,3,4-thiadiazoles
Dalip Kumar et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2011)
Benzothiazole-based N-(phenylsulfonyl)amides as a novel family of PPARα antagonists
Alessandra Ammazzalorso et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2011)
Phase 2 trial of romidepsin in patients with peripheral T-cell lymphoma
Richard L. Piekarz et al.
BLOOD (2011)
Coumarin-Based Bioactive Compounds: Facile Synthesis and Biological Evaluation of Coumarin-Fused 1,4-Thiazepines
Mehdi Khoobi et al.
CHEMICAL BIOLOGY & DRUG DESIGN (2011)
Rivaroxaban Population Pharmacokinetic Analyses in Patients Treated for Acute Deep-Vein Thrombosis and Exposure Simulations in Patients with Atrial Fibrillation Treated for Stroke Prevention
Wolfgang Mueck et al.
CLINICAL PHARMACOKINETICS (2011)
Edoxaban A New Oral Direct Factor Xa Inhibitor
A. John Camm et al.
DRUGS (2011)
Design, synthesis and anti-tubercular evaluation of new 2-acylated and 2-alkylated amino-5-(4-(benzyloxy)phenyl)thiophene-3-carboxylic acid derivatives. Part 1
Xiaoyun Lu et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2011)
New imidazo[2,1-b]thiazole derivatives: Synthesis, in vitro anticancer evaluation, and in silico studies
Jin-Hun Park et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2011)
Recent progress in biological activities of synthesized phenothiazines
Krystian Pluta et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2011)
Synthesis and anticancer evaluation of novel 2-cyclopropylimidazo[2,1-b] [1,3,4]-thiadiazole derivatives
Malleshappa N. Noolvi et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2011)
Synthesis and biological evaluation of novel 2-aralkyl-5-substituted-6-(4′-fluorophenyl)-imidazo[2,1-b][1,3,4]thiadiazole derivatives as potent anticancer agents
Subhas S. Karki et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2011)
Anti-breast cancer activity of some novel 1,2-dihydropyridine, thiophene and thiazole derivatives
Mansour S. Al-Said et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2011)
Mirabegron: a safety review
Pradeep Tyagi et al.
EXPERT OPINION ON DRUG SAFETY (2011)
Benzothiophene Carboxamide Derivatives as Novel Antimalarials
Tanushree Banerjee et al.
IUBMB LIFE (2011)
DETERMINATION OF THE LIPOPHILICITY PARAMETERS LOG PCALCD, RM0 AND LOG PTLC OF NEW ANTICANCER ACYLAMINOALKYL- AND SULFONYLAMINOALKYLAZAPHENOTHIAZINES BY COMPUTATIONAL METHODS AND REVERSED-PHASE THIN-LAYER CHROMATOGRAPHY
Beata Morak-Mlodawska et al.
JOURNAL OF LIQUID CHROMATOGRAPHY & RELATED TECHNOLOGIES (2011)
Design, Synthesis, and SAR Studies of 4-Substituted Methoxylbenzoyl-aryl-thiazoles Analogues as Potent and Orally Bioavailable Anticancer Agents
Yan Lu et al.
JOURNAL OF MEDICINAL CHEMISTRY (2011)
Novel Synthesis of Hydrazide-Hydrazone Derivatives and Their Utilization in the Synthesis of Coumarin, Pyridine, Thiazole and Thiophene Derivatives with Antitumor Activity
Rafat M. Mohareb et al.
MOLECULES (2011)
Synthesis and anti-inflammatory activity of new arylidene-thiazolidine-2,4-diones as PPARγ ligands
Cleiton Diniz Barros et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2010)
RhoGDI signaling provides targets for cancer therapy
Michael A. Harding et al.
EUROPEAN JOURNAL OF CANCER (2010)
Synthesis of some p-toluenesulfonyl-hydrazinothiazoles and hydrazino-bis-thiazoles and their anticancer activity
Valentin Zaharia et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2010)
Synthesis and anticancer activity of 5-(3-indolyl)-1,3,4-thiadiazoles
Dalip Kumar et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2010)
Synthesis and anticancer activity evaluation of 4-thiazolidinones containing benzothiazole moiety
Dmytro Havrylyuk et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2010)
Synthesis and primary cytotoxicity evaluation of new 5-benzylidene-2, 4-thiazolidinedione derivatives
Vijay Patil et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2010)
Anticancer activity of newly synthesized azaphenothiazines from NCI's anticancer screening bank
Krystian Pluta et al.
PHARMACOLOGICAL REPORTS (2010)
Synthesis of bis-1,2,3-triazolo-bridged unsymmetrical pyrrolobenzodiazepine trimers via 'click' chemistry and their DNA-binding studies
Ahmed Kamal et al.
TETRAHEDRON (2010)
PTP1B: a double agent in metabolism and oncogenesis
Shu-Chin Yip et al.
TRENDS IN BIOCHEMICAL SCIENCES (2010)
6[3-(4-Fluorophenyl)-1H-pyrazol-4-yl]-3-[(2-naphthyloxy)methyl][1,2,4]triazolo[3,4-b][1,3,4]-thiadiazole as a potent antioxidant and an anticancer agent induces growth inhibition followed by apoptosis in HepG2 cells
Dhanya Sunil et al.
ARABIAN JOURNAL OF CHEMISTRY (2010)
2-Arylbenzothiazole as a Privileged Scaffold in Drug Discovery
A. A. Weekes et al.
CURRENT MEDICINAL CHEMISTRY (2009)
Synthesis and pharmacological evaluation of 2-substituted benzo[b]thiophenes as anti-inflammatory and analgesic agents
Issa M. I. Fakhr et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2009)
Synthesis and Properties of Diaza-, Triaza-, and Tetraazaphenothiazines
Krystian Pluta et al.
JOURNAL OF HETEROCYCLIC CHEMISTRY (2009)
Discovery of 4-Substituted Methoxybenzoyl-aryl-thiazole as Novel Anticancer Agents: Synthesis, Biological Evaluation, and Structure-Activity Relationships
Yan Lu et al.
JOURNAL OF MEDICINAL CHEMISTRY (2009)
Phase 1 Study of the Pittsburgh Compound B Derivative 18F-Flutemetamol in Healthy Volunteers and Patients with Probable Alzheimer Disease
Natalie Nelissen et al.
JOURNAL OF NUCLEAR MEDICINE (2009)
ROMIDEPSIN FOR THE TREATMENT OF CUTANEOUS T-CELL LYMPHOMA
Clara Campas-Moya
DRUGS OF TODAY (2009)
Synthesis of 1,2,3-triazole-linked pyrrolobenzodiazepine conjugates employing 'click' chemistry: DNA-binding affinity and anticancer activity
Ahmed Kamal et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2008)
1,5-Benzothiazepine, a versatile pharmacophore: A review
Jitender B. Bariwal et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2008)
Icatibant
Konrad Bork et al.
NATURE REVIEWS DRUG DISCOVERY (2008)
Synthesis and antimicrobial activity of some new thiazolyl thiazolidine-2,4-dione derivatives
Oya Bozdag-Duendar et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2007)
Benzothiophene selective estrogen receptor modulators with modulated oxidative activity and receptor affinity
Zhihui Qin et al.
JOURNAL OF MEDICINAL CHEMISTRY (2007)
Synthesis and antitumor properties of 2,5-bis(3′-indolyl)thiophenes:: Analogues of marine alkaloid nortopsentin
Patrizia Diana et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2007)
Focal adhesion kinase: A potential target in cancer therapy
Maroesja J. van Nimwegen et al.
BIOCHEMICAL PHARMACOLOGY (2007)
Synthesis and biological evaluation of 2-(3′,4′,5′-trimethoxybenzoyl)-3-amino 5-aryl thiophenes as a new class of tubulin inhibitors
Romeo Romagnoli et al.
JOURNAL OF MEDICINAL CHEMISTRY (2006)
Enantioselective organocatalytic tandem Michael-aldol reactions: One-pot synthesis of chiral thiochromenes
Wei Wang et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2006)
Anticancer activities of some newly synthesized pyridine, pyrane, and pyrimidine derivatives
Abdel-Galil E. Amr et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2006)
Dasatinib in imatinib-resistant Philadelphia chromosome-positive leukemias
Moshe Talpaz et al.
NEW ENGLAND JOURNAL OF MEDICINE (2006)
Angiogenesis as a therapeutic target
N Ferrara et al.
NATURE (2005)
Parallel synthesis and biological evaluation of 5,6,7,8-tetrahydrobenzothieno[2,3-d]pyrimidin-4(3H)-one cytotoxic agents selective for p21-deficient cells
LD Jennings et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2005)
Inhibition of tumor cell proliferation by thieno[2,3-d]pyrimidin-4(1H)-one-based analogs
YD Wang et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2005)
Synthesis, biological activity and modelling studies of two novel anti HIV PR inhibitors with a thiophene containing hydroxyethylamino core
C Bonini et al.
TETRAHEDRON (2005)
Nitazoxanide: A new thiazolide antiparasitic agent
LM Fox et al.
CLINICAL INFECTIOUS DISEASES (2005)
Timeline - The discovery of receptor tyrosine kinases: targets for cancer therapy
A Gschwind et al.
NATURE REVIEWS CANCER (2004)
Efficacy and safety of ivermectin and thiabendazole in the treatment of strongyloidiasis
R Igual-Adell et al.
EXPERT OPINION ON PHARMACOTHERAPY (2004)
Investigation of anticancer mechanism of thiadiazole-based compound in human non-small cell lung cancer A549 cells
JY Chou et al.
BIOCHEMICAL PHARMACOLOGY (2003)
The antimicrobial natural product chuangxinmycin and some synthetic analogues are potent and selective inhibitors of bacterial tryptophanyl tRNA synthetase
MJ Brown et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2002)
Structure-activity relationships in 1,4-benzodioxan-related compounds.: 7.: Selectivity of 4-phenylchroman analogues for α1-adrenoreceptor subtypes
W Quaglia et al.
JOURNAL OF MEDICINAL CHEMISTRY (2002)
Novel 5-substituted 2,4-thiazolidinedione and 2,4-oxazolidinedione derivatives as insulin sensitizers with antidiabetic activities
Y Momose et al.
JOURNAL OF MEDICINAL CHEMISTRY (2002)
Rosiglitazone - A review of its use in the management of type 2 diabetes mellitus
AJ Wagstaff et al.
DRUGS (2002)
Receptor tyrosine kinase signalling as a target for cancer intervention strategies
E Zwick et al.
ENDOCRINE-RELATED CANCER (2001)
Raloxifene - A review of its use in postmenopausal osteoporosis
D Clemett et al.
DRUGS (2000)
Clopidogrel - A review of its use in the prevention of atherothrombosis
B Jarvis et al.
DRUGS (2000)
Synthesis and pharmacological evaluation of thiopyran analogues of the dopamine D3 receptor-selective agonist (4aR,10bR)-(+)-trans-3,4,4a,10b-tetrahydro-4-n-propyl-2H,5H-[1]benzopyrano[4,3-b]-1,4-oxazin-9-ol (PD 128907)
LA van Vliet et al.
JOURNAL OF MEDICINAL CHEMISTRY (2000)
Share Paper
