Related references
Note: Only part of the references are listed.Novel adamantane-pyrazole and hydrazone hybridized: Design, synthesis, cytotoxic evaluation, SAR study and molecular docking simulation as carbonic anhydrase inhibitors
Mohammed M. S. Wassel et al.
JOURNAL OF MOLECULAR STRUCTURE (2021)
Novel structural hybrids of quinoline and thiazole moieties: Synthesis and evaluation of antibacterial and antifungal activities with molecular modeling studies
Sally Eissa et al.
BIOORGANIC CHEMISTRY (2021)
Development of adamantane scaffold containing 1,3,4-thiadiazole derivatives: Design, synthesis, anti-proliferative activity and molecular docking study targeting EGFR
Mohammed M. S. Wassel et al.
BIOORGANIC CHEMISTRY (2021)
Sulfaguanidine Hybrid with Some New Pyridine-2-One Derivatives: Design, Synthesis, and Antimicrobial Activity against Multidrug-Resistant Bacteria as Dual DNA Gyrase and DHFR Inhibitors
Ahmed Ragab et al.
ANTIBIOTICS-BASEL (2021)
Design, synthesis, in vitro antimicrobial evaluation and molecular docking studies of indol-2-one tagged with morpholinosulfonyl moiety as DNA gyrase inhibitors
Mohamed A. Salem et al.
BIOORGANIC CHEMISTRY (2020)
One-pot synthesis and molecular docking of some new spiropyranindol-2-one derivatives as immunomodulatory agents and in vitro antimicrobial potential with DNA gyrase inhibitor
Mohamed A. Salem et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2020)
Design, synthesis, biological evaluation and molecular docking study based on novel fused pyrazolothiazole scaffold
Hala F. Rizk et al.
JOURNAL OF THE IRANIAN CHEMICAL SOCIETY (2020)
Antimicrobial evaluation of thiadiazino and thiazolo quinoxaline hybrids as potential DNA gyrase inhibitors; design, synthesis, characterization and morphological studies
Yousry A. Ammar et al.
BIOORGANIC CHEMISTRY (2020)
In vitro cytotoxic activity of thiazole-indenoquinoxaline hybrids as apoptotic agents, design, synthesis, physicochemical and pharmacokinetic studies
Eman A. Fayed et al.
BIOORGANIC CHEMISTRY (2020)
Discovery of New Schiff Bases Tethered Pyrazole Moiety: Design, Synthesis, Biological Evaluation, and Molecular Docking Study as Dual Targeting DHFR/DNA Gyrase Inhibitors with Immunomodulatory Activity
Ashraf S. Hassan et al.
MOLECULES (2020)
Design, synthesis, antimicrobial activity and molecular docking studies of some novel di-substituted sulfonylquinoxaline derivatives
Yousry A. Ammar et al.
BIOORGANIC CHEMISTRY (2020)
Design, synthesis, cytotoxicity and molecular modeling studies of some novel fluorinated pyrazole-based heterocycles as anticancer and apoptosis-inducing agents
Eman A. Fayed et al.
MOLECULAR DIVERSITY (2019)
Design, synthesis, molecular docking and biological activity evaluation of some novel indole derivatives as potent anticancer active agents and apoptosis inducers
Ahmed M. Sh El-Sharief et al.
BIOORGANIC CHEMISTRY (2019)
Design, synthesis, biological evaluation and molecular modeling of new coumarin derivatives as potent anticancer agents
Eman A. Fayed et al.
MEDICINAL CHEMISTRY RESEARCH (2019)
Design, synthesis, biological evaluations, molecular docking, and in vivo studies of novel phthalimide analogs
Magdy A. H. Zahran et al.
ARCHIV DER PHARMAZIE (2018)
Design, synthesis, molecular docking of new lipophilic acetamide derivatives affording potential anticancer and antimicrobial agents
Hany E. A. Ahmed et al.
BIOORGANIC CHEMISTRY (2018)
Synthesis, anti-inflammatory, p38α MAP kinase inhibitory activities and molecular docking studies of quinoxaline derivatives containing triazole moiety
Sana Tariq et al.
BIOORGANIC CHEMISTRY (2018)
Design, synthesis, antiproliferative activity, molecular docking and cell cycle analysis of some novel (morpholinosulfonyl) isatins with potential EGFR inhibitory activity
Yousry A. Ammar et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2018)
Design, Synthesis, and Biological Evaluation of Pyrimido[4,5-d]pyrimidine-2,4(1H,3H)-diones as Potent and Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors against L858R/T790M Resistance Mutation
Yongjia Hao et al.
JOURNAL OF MEDICINAL CHEMISTRY (2018)
Antiproliferative activity of the combination of doxorubicin/quercetin on MCF7 breast cancer cell line: A combined study using colorimetric assay and synchrotron infrared microspectroscopy
Nirmeen Elmadany et al.
INFRARED PHYSICS & TECHNOLOGY (2018)
Small Molecule Antagonists of the Interaction between the Histone Deacetylase 6 Zinc-Finger Domain and Ubiquitin
Rachel J. Harding et al.
JOURNAL OF MEDICINAL CHEMISTRY (2017)
Synthesis and Evaluation of New Quinoxaline Derivatives of Dehydroabietic Acid as Potential Antitumor Agents
Wen Gu et al.
MOLECULES (2017)
Cancer Statistics, 2016
Rebecca L. Siegel et al.
CA-A CANCER JOURNAL FOR CLINICIANS (2016)
Synthesis and evaluation of antitumour activities of novel fused tri- and tetracyclic uracil derivatives
Samar ElKalyoubi et al.
JOURNAL OF CHEMICAL RESEARCH (2016)
Design, synthesis, biological evaluation and docking studies of sulfonyl isatin derivatives as monoamine oxidase and caspase-3 inhibitors
Mohsen Tavari et al.
MEDCHEMCOMM (2016)
Synthesis, Characterization and Biological Evaluation of Some Quinoxaline Derivatives: A Promising and Potent New Class of Antitumor and Antimicrobial Agents
Aisha R. Al-Marhabi et al.
MOLECULES (2015)
5-(2-Carboxyethenyl) isatin derivative induces G2/M cell cycle arrest and apoptosis in human leukemia K562 cells
Yao Zhou et al.
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS (2014)
Design, synthesis and biological evaluation of (E)-2-(2-arylhydrazinyl) quinoxalines, a promising and potent new class of anticancer agents
Felipe A. R. Rodrigues et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2014)
Paris saponin I induces apoptosis via increasing the Bax/Bcl-2 ratio and caspase-3 expression in gefitinib-resistant non-small cell lung cancer in vitro and in vivo
Hao Jiang et al.
MOLECULAR MEDICINE REPORTS (2014)
Synthesis of new fluorinated, 2-substituted 5-pyrrolidinylsulfonyl isatin derivatives as caspase-3 and caspase-7 inhibitors: Nonradioactive counterparts of putative PET-compatible apoptosis imaging agents
Panupun Limpachayaporn et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2013)
Design, synthesis and structure-activity relationship of novel quinoxaline derivatives as cancer chemopreventive agent by inhibition of tyrosine kinase receptor
Shadia A. Galar et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2013)
Microwave assisted synthesis and antimicrobial activity of 2-quinoxalinone-3-hydrazone derivatives
Olayinka O. Ajani et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2010)
Synthesis and antitumor activity of novel 6-aryl and 6-alkylpyrazolo[3,4-d] pyrimidin-4-one derivatives
Mervat M. El-Enany et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2010)
New quinoxaline 1, 4-di-N-oxides: Anticancer and hypoxia-selective therapeutic agents
Magda M. F. Ismail et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2010)
Benzylidene/2-chlorobenzylidene hydrazides: Synthesis, antimicrobial activity, QSAR studies and antiviral evaluation
Davinder Kumar et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2010)
Synthesis, trypanocidal activity and docking studies of novel quinoxaline-N-acylhydrazones, designed as cruzain inhibitors candidates
Nelilma C. Romeiro et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2009)
Synthesis of novel quinoxaline derivatives and its cytotoxic activities
Shinji Tanimori et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2009)
New transition metal ion complexes with benzimidazole-5-carboxylic acid hydrazides with antitumor activity
Shadia A. Galal et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2009)
In vitro cytotoxic and antioxidative activity of Cornus mas and Cotinus coggygria
Katarina Savikin et al.
NATURAL PRODUCT RESEARCH (2009)
Artificial Neural Networks from MATLAB® in Medicinal Chemistry. Bayesian-Regularized Genetic Neural Networks (BRGNN): Application to the Prediction of the Antagonistic Activity Against Human Platelet Thrombin Receptor (PAR-1)
Julio Caballero et al.
CURRENT TOPICS IN MEDICINAL CHEMISTRY (2008)
Luminescent biological probes derived from ruthenium(II) estradiol polypyridine complexes
Kenneth Kam-Wing Lo et al.
INORGANIC CHEMISTRY (2008)
The BCL-2 protein family: opposing activities that mediate cell death
Richard J. Youle et al.
NATURE REVIEWS MOLECULAR CELL BIOLOGY (2008)
Privileged structures: A useful concept for the rational design of new lead drug candidates
Carolina D. Duarte et al.
MINI-REVIEWS IN MEDICINAL CHEMISTRY (2007)
Synthesis and antiproliferative properties of N3/8-disubstituted 3,8-diazabicyclo[3.2.1]octane analogues of 3,8-bis[2-(3,4,5-trimethoxyphenyl)pyridin-4-yl]methyl-piperazine
Rosanna Filosa et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2007)
New quinoxaline 1,4-di-N-oxides.: Part 1:: Hypoxia-selective cytotoxins and anticancer agents derived from quinoxaline 1,4-di-N-oxides
Kamelia M. Amin et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2006)
Homogeneous time-resolved fluorescence and its applications for kinase assays in drug discovery
Yong Jia et al.
ANALYTICAL BIOCHEMISTRY (2006)
A combination of docking/dynamics simulations and pharmacophoric modeling to discover new dual c-Src/Abl kinase inhibitors
Fabrizio Manetti et al.
JOURNAL OF MEDICINAL CHEMISTRY (2006)
Sulforhodamine B colorimetric assay for cytotoxicity screening
Vanicha Vichai et al.
NATURE PROTOCOLS (2006)
Part 3: Synthesis and biological evaluation of some analogs of the antitumor agents, 2-{4-[(7-chloro-2-quinoxalinyl)-oxy]phenoxy}propionic acid, and 2-{4-[(7-bromo-2-quinolinyl)-oxy]phenoxy}propionic acid
ST Hazeldine et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2005)
Synthesis of cyclopeptidic analogues of triostin A with quinoxalines or nucleobases as chromophores
B Dietrich et al.
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2005)
Discovery of a potent, non-peptide bradykinin B1 receptor antagonist
DS Su et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2003)
Synthesis, characterization and in vitro anti-invasive activity screening of polyphenolic and heterocyclic compounds
VS Parmar et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2003)
Crystal structures of reversible ketone-based inhibitors of the cysteine protease cruzain
L Huang et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2003)
II. Synthesis and biological evaluation of some bioisosteres and congeners of the antitumor agent, 2-{4-[(7-chloro-2-quinoxalinyl)oxy]phenoxy}propionic acid (XK469)
ST Hazeldine et al.
JOURNAL OF MEDICINAL CHEMISTRY (2002)
Design, synthesis, and biological evaluation of analogues of the antitumor agent, 2-{4-[(7-chloro-2-quinoxalinyl)oxy]phenoxy}propionic acid (XK469)
ST Hazeldine et al.
JOURNAL OF MEDICINAL CHEMISTRY (2001)
Share Paper
