Related references
Note: Only part of the references are listed.The 1,8-naphthyridines sulfonamides are NorA efflux pump inhibitors
Cicera Datiane de Morais Oliveira-Tintino et al.
JOURNAL OF GLOBAL ANTIMICROBIAL RESISTANCE (2021)
Antimicrobial Resistance in Bacteria: Mechanisms, Evolution, and Persistence
Eirini Christaki et al.
JOURNAL OF MOLECULAR EVOLUTION (2020)
C-2 phenyl replacements to obtain potent quinoline-based Staphylococcus aureus NorA inhibitors
Tommaso Felicetti et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2020)
Antimicrobial Resistance in ESKAPE Pathogens
David M. P. De Oliveira et al.
CLINICAL MICROBIOLOGY REVIEWS (2020)
Efflux pump activity potentiates the evolution of antibiotic resistance across S. aureus isolates
Andrei Papkou et al.
NATURE COMMUNICATIONS (2020)
Structural Modifications of the Quinolin-4-yloxy Core to Obtain New Staphylococcus aureus NorA Inhibitors
Rolando Cannalire et al.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (2020)
Methicillin-resistant Staphylococcus aureus: an overview of basic and clinical research
Nicholas A. Turner et al.
NATURE REVIEWS MICROBIOLOGY (2019)
Modifications on C6 and C7 Positions of 3-Phenylquinolone Efflux Pump Inhibitors Led to Potent and Safe Antimycobacterial Treatment Adjuvants
Tommaso Felicetti et al.
ACS INFECTIOUS DISEASES (2019)
Efflux pump inhibitors of clinically relevant multidrug resistant bacteria
Andraz Lamut et al.
MEDICINAL RESEARCH REVIEWS (2019)
The challenge of antimicrobial resistance: What economics can contribute
Laurence S. J. Roope et al.
SCIENCE (2019)
Emerging Strategies to Combat ESKAPE Pathogens in the Era of Antimicrobial Resistance: A Review
Mansura S. Mulani et al.
FRONTIERS IN MICROBIOLOGY (2019)
Attributable deaths and disability-adjusted life-years caused by infections with antibiotic-resistant bacteria in the EU and the European Economic Area in 2015: a population-level modelling analysis
Alessandro Cassini et al.
LANCET INFECTIOUS DISEASES (2019)
The Continuing Threat of Methicillin-Resistant Staphylococcus aureus
Mario Gajdacs
ANTIBIOTICS-BASEL (2019)
Bioactive Immunomodulatory Compounds: A Novel Combinatorial Strategy for Integrated Medicine in Oncology? BAIC Exposure in Cancer Cells
Bruna Corradetti et al.
INTEGRATIVE CANCER THERAPIES (2019)
Studies on 2-phenylquinoline Staphylococcus aureus NorA efflux pump inhibitors: New insights on the C-6 position
Tommaso Felicetti et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2018)
2-Phenylquinoline S. aureus NorA Efflux Pump Inhibitors: Evaluation of the Importance of Methoxy Group Introduction
Tommaso Felicetti et al.
JOURNAL OF MEDICINAL CHEMISTRY (2018)
An overview of the antimicrobial resistance mechanisms of bacteria
Wanda C. Reygaert
AIMS MICROBIOLOGY (2018)
Improved Potency of Indole-Based NorA Efflux Pump Inhibitors: From Serendipity toward Rational Design and Development
Federica Buonerba et al.
JOURNAL OF MEDICINAL CHEMISTRY (2017)
Pharmacophore-Based Repositioning of Approved Drugs as Novel Staphylococcus aureus NorA Efflux Pump Inhibitors
Andrea Astolfi et al.
JOURNAL OF MEDICINAL CHEMISTRY (2017)
Investigation on the effect of known potent S. aureus NorA efflux pump inhibitors on the staphylococcal biofilm formation
Stefano Sabatini et al.
RSC ADVANCES (2017)
The Transporter Classification Database (TCDB): recent advances
Milton H. Saier et al.
NUCLEIC ACIDS RESEARCH (2016)
Indole Based Weapons to Fight Antibiotic Resistance: A Structure-Activity Relationship Study
Susan Lepri et al.
JOURNAL OF MEDICINAL CHEMISTRY (2016)
Biofilms: an emergent form of bacterial life
Hans-Curt Flemming et al.
NATURE REVIEWS MICROBIOLOGY (2016)
Mechanisms of Antimicrobial Resistance in ESKAPE Pathogens
Sirijan Santajit et al.
BIOMED RESEARCH INTERNATIONAL (2016)
Boronic species as promising inhibitors of the Staphylococcus aureus NorA efflux pump: Study of 6-substituted pyridine-3-boronic acid derivatives
Fanny Fontaine et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2015)
Molecular mechanisms of antibiotic resistance
Jessica M. A. Blair et al.
NATURE REVIEWS MICROBIOLOGY (2015)
1-(1H-Indol-3-yl)ethanamine Derivatives as Potent Staphylococcus aureus NorA Efflux Pump Inhibitors
Arnaud Hequet et al.
CHEMMEDCHEM (2014)
First Identification of Boronic Species as Novel Potential Inhibitors of the Staphylococcus aureus NorA Efflux Pump
Fanny Fontaine et al.
JOURNAL OF MEDICINAL CHEMISTRY (2014)
Development of N-Methyl-(2-arylquinolin-4-yl)oxypropanamides as Leads to PET Radioligands for Translocator Protein (18 kDa)
Chad Brouwer et al.
JOURNAL OF MEDICINAL CHEMISTRY (2014)
Synthesis of Functionalized Isoquinolin-1(2H)-ones by Copper-Catalyzed -Arylation of Ketones with 2-Halobenzamides
Yan Shi et al.
CHEMISTRY-A EUROPEAN JOURNAL (2013)
Computer-Aided Design, Synthesis and Validation of 2-Phenylquinazolinone Fragments as CDK9 Inhibitors with Anti-HIV-1 Tat-Mediated Transcription Activity
Luca Sancineto et al.
CHEMMEDCHEM (2013)
Structural basis for the inhibition of bacterial multidrug exporters
Ryosuke Nakashima et al.
NATURE (2013)
Chalcone inhibitors of the NorA efflux pump in Staphylococcus aureus whole cells and enriched everted membrane vesicles
Jes Gitz Holler et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2012)
Evolution from a Natural Flavones Nucleus to Obtain 2-(4-Propoxyphenyl)quinoline Derivatives As Potent Inhibitors of the S. aureus NorA Efflux Pump
Stefano Sabatini et al.
JOURNAL OF MEDICINAL CHEMISTRY (2011)
Towards the comprehensive, rapid, and accurate prediction of the favorable tautomeric states of drug-like molecules in aqueous solution
Jeremy R. Greenwood et al.
JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN (2010)
Anti-virulence strategies to combat bacteria-mediated disease
David A. Rasko et al.
NATURE REVIEWS DRUG DISCOVERY (2010)
MacB ABC Transporter Is a Dimer Whose ATPase Activity and Macrolide-binding Capacity Are Regulated by the Membrane Fusion Protein MacA
Hong Ting Lin et al.
JOURNAL OF BIOLOGICAL CHEMISTRY (2009)
Inactivation of Efflux Pumps Abolishes Bacterial Biofilm Formation
Malin Kvist et al.
APPLIED AND ENVIRONMENTAL MICROBIOLOGY (2008)
Selective ruthenium-catalyzed hydration of nitriles to amides in pure aqueous medium under neutral conditions
Victorio Cadierno et al.
CHEMISTRY-A EUROPEAN JOURNAL (2008)
Novel structural analogues of piperine as inhibitors of the NorA efflux pump of Staphylococcus aureus
Ashwani Kumar et al.
JOURNAL OF ANTIMICROBIAL CHEMOTHERAPY (2008)
PHASE: A novel approach to pharmacophore modeling and 3D database searching
Steven L. Dixon et al.
CHEMICAL BIOLOGY & DRUG DESIGN (2006)
Evidence for the existence of a multidrug efflux transporter distinct from NorA in Staphylococcus aureus
GW Kaatz et al.
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY (2000)