Related references
Note: Only part of the references are listed.Looking toward the Rim of the Active Site Cavity of Druggable Human Carbonic Anhydrase Isoforms
Francesca Mancuso et al.
ACS MEDICINAL CHEMISTRY LETTERS (2020)
Discovery, Optimization, and Characterization of ML417: A Novel and Highly Selective D3 Dopamine Receptor Agonist
Amy E. Moritz et al.
JOURNAL OF MEDICINAL CHEMISTRY (2020)
Discovery of 2,4-diaminopyrimidine derivatives targeting p21-activated kinase 4: Biological evaluation and docking studies
Qiaohua Qin et al.
ARCHIV DER PHARMAZIE (2020)
Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment
Andrea Angeli et al.
METABOLITES (2020)
SLC-0111 enaminone analogs, 3/4-(3-aryl-3-oxopropenyl) aminobenzenesulfonamides, as novel selective subnanomolar inhibitors of the tumor-associated carbonic anhydrase isoform IX
Wagdy M. Eldehna et al.
BIOORGANIC CHEMISTRY (2019)
Exploring structural properties of potent human carbonic anhydrase inhibitors bearing a 4-(cycloalkylamino-1-carbonyl) benzenesulfonamide moiety
Maria Rosa Buemi et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2019)
Novel synthesized SLC-0111 thiazole and thiadiazole analogues: Determination of their carbonic anhydrase inhibitory activity and molecular modeling studies
Mahmoud F. Abo-Ashour et al.
BIOORGANIC CHEMISTRY (2019)
Enhancement of the tail hydrophobic interactions within the carbonic anhydrase IX active site via structural extension: Design and synthesis of novel N-substituted isatins-SLC-0111 hybrids as carbonic anhydrase inhibitors and antitumor agents
Wagdy M. Eldehna et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2019)
The carbonic anhydrase IX inhibitor SLC-0111 sensitises cancer cells to conventional chemotherapy
Elena Andreucci et al.
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (2019)
Structural investigations on coumarins leading to chromeno[4,3-c] pyrazol-4-ones and pyrano[4,3-c]pyrazol-4-ones: New scaffolds for the design of the tumor-associated carbonic anhydrase isoforms IX and XII
Alessandro Bonardi et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2018)
The Crystal Structure of a hCA VII Variant Provides Insights into the Molecular Determinants Responsible for Its Catalytic Behavior
Martina Buonanno et al.
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (2018)
Discovery of 4-Hydroxy-3-(3-(phenylureido)benzenesulfonamides as SLC-0111 Analogues for the Treatment of Hypoxic Tumors Overexpressing Carbonic Anhydrase IX
Murat Bozdag et al.
JOURNAL OF MEDICINAL CHEMISTRY (2018)
Advances in structure-based drug discovery of carbonic anhydrase inhibitors
Claudiu T. Supuran
EXPERT OPINION ON DRUG DISCOVERY (2017)
Carbonic anhydrase XII functions in health and disease
Abdul Waheed et al.
GENE (2017)
Structure-Activity Relationships of Potent, Targeted Covalent Inhibitors That Abolish Both the Transamidation and GTP Binding Activities of Human Tissue Transglutaminase
Abdullah Akbar et al.
JOURNAL OF MEDICINAL CHEMISTRY (2017)
Probing Molecular Interactions between Human Carbonic Anhydrases (hCAs) and a Novel Class of Benzenesulfonamides
Elvira Bruno et al.
JOURNAL OF MEDICINAL CHEMISTRY (2017)
Addition of carbonic anhydrase 9 inhibitor SLC-0111 to temozolomide treatment delays glioblastoma growth in vivo
Nathaniel H. Boyd et al.
JCI INSIGHT (2017)
Synthesis and carbonic anhydrase inhibition of a series of SLC-011.1 analogs
Fabrizio Carta et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2017)
Kinetic and X-ray crystallographic investigations on carbonic anhydrase isoforms I, II, IX and XII of a thioureido analog of SLC-0111
Carrie L. Lomelino et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2016)
InVivo Evaluation of Selective Carbonic Anhydrase Inhibitors as Potential Anticonvulsant Agents
Elvira Bruno et al.
CHEMMEDCHEM (2016)
Carbonic anhydrase inhibitors: Design, synthesis and structural characterization of new heteroaryl-N-carbonylbenzenesulfonamides targeting druggable human carbonic anhydrase isoforms
Maria Rosa Buemi et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2015)
Structure-based screening for the discovery of new carbonic anhydrase VII inhibitors
Laura De Luca et al.
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2014)
Anticancer carbonic anhydrase inhibitors: a patent review (2008-2013)
Simona Maria Monti et al.
EXPERT OPINION ON THERAPEUTIC PATENTS (2013)
Substituted phenoxypropyl-(R)-2-methylpyrrolidine aminomethyl ketones as histamine-3 receptor inverse agonists
Allison L. Zulli et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2012)
Multiple Binding Modes of Inhibitors to Carbonic Anhydrases: How to Design Specific Drugs Targeting 15 Different Isoforms?
Vincenzo Alterio et al.
CHEMICAL REVIEWS (2012)
Carbonic anhydrase inhibitors as emerging drugs for the treatment of obesity
Claudiu T. Supuran
EXPERT OPINION ON EMERGING DRUGS (2012)
Crystal structure of the C183S/C217S mutant of human CA VII in complex with acetazolamide
Anna Di Fiore et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2010)
Identification of Potent and Selective Human Carbonic Anhydrase VII (hCA VII) Inhibitors
Rosaria Gitto et al.
CHEMMEDCHEM (2010)
Design, Synthesis, and Structure-Affinity Relationships of Regioisomeric N-Benzyl Alkyl Ether Piperazine Derivatives as σ-1 Receptor Ligands
Iman A. Moussa et al.
JOURNAL OF MEDICINAL CHEMISTRY (2010)
Discovery of potent furan piperazine sodium channel blockers for treatment of neuropathic pain
Irene Drizin et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2008)
Carbonic anhydrase inhibitors as emerging drugs for the treatment of obesity
Claudiu T. Supuran et al.
EXPERT OPINION ON EMERGING DRUGS (2008)
Carbonic anhydrases: novel therapeutic applications for inhibitors and activators
Claudiu T. Supuran
NATURE REVIEWS DRUG DISCOVERY (2008)
Carbonic anhydrase inhibitors. Inhibition of transmembrane isozymes XII (cancer-associated) and XIV with anions
Alessio Innocenti et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2007)
Version 1.2 of the Crystallography and NMR system
Axel T. Brunger
NATURE PROTOCOLS (2007)
Carbonic anhydrase inhibitors. The mitochondrial isozyme VB as a new target for sulfonamide and sulfamate inhibitors
I Nishimori et al.
JOURNAL OF MEDICINAL CHEMISTRY (2005)
Carbonic anhydrase inhibitors: Inhibition of the transmembrane isozyme XIV with sulfonamides
I Nishimori et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2005)
VEGA: a versatile program to convert, handle and visualize molecular structure on Windows-based PCs
A Pedretti et al.
JOURNAL OF MOLECULAR GRAPHICS & MODELLING (2002)
Share Paper
