Journal
SYNLETT
Volume 32, Issue 10, Pages 1034-1038Publisher
GEORG THIEME VERLAG KG
DOI: 10.1055/s-0037-1610771
Keywords
haloetherification; indolines; azaindolines; morpholines; oxazepines; oxazocines
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A practical method for synthesizing heterocycle-2,3-fused indoline or azaindoline derivatives through haloetherification and cyclization was described and applied in syntheses of six- to eight-membered heterocycle-2,3-fused indoline and azaindoline derivatives, which contain sp(3)-hybridized carbons and might serve as new scaffolds in medicinal chemistry.
We describe a practical method for synthesizing heterocycle-2,3-fused indoline or azaindoline derivatives through haloetherification and cyclization. We applied this method in syntheses of six- to eight-membered heterocycle-2,3-fused indoline and azaindoline derivatives. These derivatives, which contain sp(3)-hybridized carbons, might be useful as new scaffolds in medicinal chemistry.
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