Related references
Note: Only part of the references are listed.Highly Enantioselective Construction of Strained Spiro[2,3]hexanes through a Michael Addition/Ring Expansion/Cyclization Cascade
Chuan-Gang Zhao et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2020)
Axial shielding of Pd(II) complexes enables perfect stereoretention in Suzuki-Miyaura cross-coupling of Csp3 boronic acids
Jonathan W. Lehmann et al.
NATURE COMMUNICATIONS (2019)
Asymmetric synthesis of 1-substituted 2-azaspiro[3.3]heptanes: important motifs for modern drug discovery
Leleti Rajender Reddy et al.
CHEMICAL COMMUNICATIONS (2019)
Identification and Characterization of Von Hippel-Lindau-Recruiting Proteolysis Targeting Chimeras (PROTACs) of TANK-Binding Kinase 1
Andrew P. Crew et al.
JOURNAL OF MEDICINAL CHEMISTRY (2018)
Enantioselective Intermolecular [2+2] Photocycloaddition Reaction of Cyclic Enones and Its Application in a Synthesis of (-)-Grandisol
Saner Poplata et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2018)
A Protocol for Direct Stereospecific Amination of Primary, Secondary, and Tertiary Alkylboronic Esters
Emma K. Edelstein et al.
SYNLETT (2018)
Copper-Catalyzed Borylative Ring Closing C-C Coupling toward Spiro- and Dispiroheterocycles
Jordi Royes et al.
ACS CATALYSIS (2018)
Transition-metal-free synthesis of vicinal triborated compounds and selective functionalisation of the internal C-B bond
Elliot Davenport et al.
CHEMICAL COMMUNICATIONS (2018)
Design and Synthesis of Spirocycles
Sambasivarao Kotha et al.
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY (2017)
50 Years of Zweifel Olefination: A Transition-Metal-Free Coupling
Roly J. Armstrong et al.
SYNTHESIS-STUTTGART (2017)
Synthesis of Spirocyclic Pyrrolidines: Advanced Building Blocks for Drug Discovery
Bohdan A. Chalyk et al.
CHEMISTRY-A EUROPEAN JOURNAL (2017)
1-Substituted 2-Azaspiro[3.3]heptanes: Overlooked Motifs for Drug Discovery
Alexander A. Kirichok et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2017)
Ligand-Promoted Borylation of C(sp3)-H Bonds with Palladium(II) Catalysts
Jian He et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2016)
Enantioselective Synthesis of Cyclobutylboronates via a Copper-Catalyzed Desymmetrization Approach
Manuel Guisan-Ceinos et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2016)
The utilization of spirocyclic scaffolds in novel drug discovery
Ya-Jun Zheng et al.
EXPERT OPINION ON DRUG DISCOVERY (2016)
Carbohydrate-Catalyzed Enantioselective Alkene Diboration: Enhanced Reactivity of 1,2-Bonded Diboron Complexes
Lichao Fang et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2016)
Iterative protecting group-free cross-coupling leading to chiral multiply arylated structures
Cathleen M. Crudden et al.
NATURE COMMUNICATIONS (2016)
Organocatalytic Enamine-Activation of Cyclopropanes for Highly Stereoselective Formation of Cyclobutanes
Kim Soholm Halskov et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2015)
Hydroxyl-Directed Cross-Coupling: A Scalable Synthesis of Debromohamigeran E and Other Targets of Interest
Thomas P. Blaisdell et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2015)
The use of spirocyclic scaffolds in drug discovery
Yajun Zheng et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2014)
Four-Membered Ring-Containing Spirocycles: Synthetic Strategies and Opportunities
Erick M. Carreira et al.
CHEMICAL REVIEWS (2014)
Enantiomerically Enriched Tris(boronates): Readily Accessible Conjunctive Reagents for Asymmetric Synthesis
John R. Coombs et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2014)
Hydroxyl-Directed Stereoselective Diboration of Alkenes
Thomas P. Blaisdell et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2014)
Stereospecific Pd-Catalyzed Cross-Coupling Reactions of Secondary Alkylboron Nucleophiles and Aryl Chlorides
Ling Li et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2014)
Asymmetric synthesis from terminal alkenes by cascades of diboration and cross-coupling
Scott N. Mlynarski et al.
NATURE (2014)
Asymmetric Synthesis of 3,3′-Spirooxindoles Fused with Cyclobutanes through Organocatalytic Formal [2+2] Cycloadditions under H-Bond-Directing Dienamine Activation
Liang-Wen Qi et al.
ORGANIC LETTERS (2014)
Asymmetric Diboration of Terminal Alkenes with a Rhodium Catalyst and Subsequent Oxidation: Enantioselective Synthesis of Optically Active 1,2-Diols
Kenji Toribatake et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2013)
Scope and Mechanism of the Pt-Catalyzed Enantioselective Diboration of Monosubstituted Alkenes
John R. Coombs et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2013)
Copper(I)-Catalyzed Borylative exo-Cyclization of Alkenyl Halides Containing Unactivated Double Bond
Koji Kubota et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2013)
Catalytic Enantioselective 1,2-Diboration of 1,3-Dienes: Versatile Reagents for Stereoselective Allylation
Laura T. Kliman et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2012)
Asymmetric organocatalytic diboration of alkenes
Amadeu Bonet et al.
ORGANIC & BIOMOLECULAR CHEMISTRY (2012)
Expanding the Azaspiro[3.3]heptane Family: Synthesis of Novel Highly Functionalized Building Blocks
Johannes A. Burkhard et al.
ORGANIC LETTERS (2012)
Transition-Metal-Free Diboration Reaction by Activation of Diboron Compounds with Simple Lewis Bases
Amadeu Bonet et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2011)
Synthesis of Azaspirocycles and their Evaluation in Drug Discovery
Johannes A. Burkhard et al.
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2010)
Synthesis and Structural Analysis of a New Class of Azaspiro[3.3]heptanes as Building Blocks for Medicinal Chemistry
Johannes A. Burkhard et al.
ORGANIC LETTERS (2010)
Escape from Flatland: Increasing Saturation as an Approach to Improving Clinical Success
Frank Lovering et al.
JOURNAL OF MEDICINAL CHEMISTRY (2009)
Pt-Catalyzed Enantioselective Diboration of Terminal Alkenes with B2(pin)2
Laura T. Kliman et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2009)
Multifaceted Palladium Catalysts Towards the Tandem Diboration-Arylation Reactions of Alkenes
Dirk Penno et al.
CHEMISTRY-A EUROPEAN JOURNAL (2008)
Cross-coupling of cyclopropyl- and cyclobutyltrifluoroborates with aryl and heteroaryl chlorides
Gary A. Molander et al.
JOURNAL OF ORGANIC CHEMISTRY (2008)
DFT studies of β-boryl elimination processes:: Potential role in catalyzed borylation reactions of alkenes
King Chung Lam et al.
ORGANOMETALLICS (2007)
A valuable, inexpensive Cu-I/N-heterocyclic carbene catalyst for the selective diboration of styrene
Vanesa Lillo et al.
CHEMISTRY-A EUROPEAN JOURNAL (2007)
Toward an understanding of the factors responsible for the 1,2-migration of alkyl groups in borate complexes
VK Aggarwal et al.
PURE AND APPLIED CHEMISTRY (2006)
Rh-catalyzed enantioselective diboration of simple alkenes: Reaction development and substrate scope
S Trudeau et al.
JOURNAL OF ORGANIC CHEMISTRY (2005)
Catalytic asymmetric carbohydroxylation of alkenes by a tandem diboration/Suzuki cross-coupling/oxidation reaction
SP Miller et al.
ORGANIC LETTERS (2004)
Rhodium-catalyzed enantioselective diboration of simple alkenes
JB Morgan et al.
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY (2003)