Related references
Note: Only part of the references are listed.Sensitization of small-diameter sensory neurons is controlled by TRPV1 and TRPA1 association
Mayur J. Patil et al.
FASEB JOURNAL (2020)
Novel therapeutic approach with PAC-14028 cream, a TRPV1 antagonist, for patients with mild-to-moderate atopic dermatitis
P. I. Song et al.
BRITISH JOURNAL OF DERMATOLOGY (2019)
Efficacy and safety of PAC-14028 cream - a novel, topical, nonsteroidal, selective TRPV1 antagonist in patients with mild-to-moderate atopic dermatitis: a phase IIb randomized trial
Y. W. Lee et al.
BRITISH JOURNAL OF DERMATOLOGY (2019)
Regulation of Pain and Itch by TRP Channels
Carlene Moore et al.
NEUROSCIENCE BULLETIN (2018)
Targeting Transient Receptor Potential Vanilloid 1 (TRPV1) Channel Softly: The Discovery of Passerini Adducts as a Topical Treatment for Inflammatory Skin Disorders
Marta Serafini et al.
JOURNAL OF MEDICINAL CHEMISTRY (2018)
Mechanisms of pruritogen-induced activation of itch nerves in isolated mouse skin
F. Ru et al.
JOURNAL OF PHYSIOLOGY-LONDON (2017)
Capsaicin: Friend or Foe in Skin Cancer and Other Related Malignancies?
Simona-Roxana Georgescu et al.
NUTRIENTS (2017)
TRPV1 and TRPA1 in cutaneous neurogenic and chronic inflammation: pro-inflammatory response induced by their activation and their sensitization
Olivier Gouin et al.
PROTEIN & CELL (2017)
The anti-inflammatory mediator palmitoylethanolamide enhances the levels of 2-arachidonoyl-glycerol and potentiates its actions at TRPV1 cation channels
Stefania Petrosino et al.
BRITISH JOURNAL OF PHARMACOLOGY (2016)
Systemic desensitization through TRPA1 channels by capsazepine and mustard oil - a novel strategy against inflammation and pain
Katrin Kistner et al.
SCIENTIFIC REPORTS (2016)
Perspectives of TRPV1 Function on the Neurogenesis and Neural Plasticity
R. Ramirez-Barrantes et al.
NEURAL PLASTICITY (2016)
Bradykinin Induces TRPV1 Exocytotic Recruitment in Peptidergic Nociceptors
Sakthikumar Mathivanan et al.
FRONTIERS IN PHARMACOLOGY (2016)
Transient receptor potential vanilloid type 1 antagonists: a patent review (2011-2014)
Yoonji Lee et al.
EXPERT OPINION ON THERAPEUTIC PATENTS (2015)
Cancer-promoting effect of capsaicin on DMBA/TPA-induced skin tumorigenesis by modulating inflammation, Erk and p38 in mice
Zhaoguo Liu et al.
FOOD AND CHEMICAL TOXICOLOGY (2015)
Structural mechanism underlying capsaicin binding and activation of the TRPV1 ion channel
Fan Yang et al.
NATURE CHEMICAL BIOLOGY (2015)
YASARA View-molecular graphics for all devices-from smartphones to workstations
Elmar Krieger et al.
BIOINFORMATICS (2014)
TRP channels in the skin
Balazs I. Toth et al.
BRITISH JOURNAL OF PHARMACOLOGY (2014)
Neurotrophins, endocannabinoids and thermo-transient receptor potential: a threesome in pain signalling
Isabel Devesa et al.
EUROPEAN JOURNAL OF NEUROSCIENCE (2014)
The ion channel TRPV1 regulates the activation and proinflammatory properties of CD4+ T cells
Samuel Bertin et al.
NATURE IMMUNOLOGY (2014)
Direct evidence for functional TRPV1/TRPA1 heteromers
Michael J. M. Fischer et al.
PFLUGERS ARCHIV-EUROPEAN JOURNAL OF PHYSIOLOGY (2014)
αCGRP is essential for algesic exocytotic mobilization of TRPV1 channels in peptidergic nociceptors
Isabel Devesa et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2014)
The Capsaicin Receptor TRPV1 as a Novel Modulator of Neural Precursor Cell Proliferation
Kristin Stock et al.
STEM CELLS (2014)
Development of PAC-14028, a Novel Transient Receptor Potential Vanilloid Type 1 (TRPV1) Channel Antagonist as a New Drug for Refractory Skin Diseases
Kyung-Min Lim et al.
ARCHIVES OF PHARMACAL RESEARCH (2012)
Activation of transient receptor potential A1 by a non-pungent capsaicin-like compound, capsiate
Kenji Shintaku et al.
BRITISH JOURNAL OF PHARMACOLOGY (2012)
TRPV1-antagonist AMG9810 promotes mouse skin tumorigenesis through EGFR/Akt signaling
Shengqing Li et al.
CARCINOGENESIS (2011)
Antipruritic Effects of TRPV1 Antagonist in Murine Atopic Dermatitis and Itching Models
Jun-Won Yun et al.
JOURNAL OF INVESTIGATIVE DERMATOLOGY (2011)
Topical capsaicin. The fire of a 'hot' medicine is reignited
Alexandru D. P. Papoiu et al.
EXPERT OPINION ON PHARMACOTHERAPY (2010)
Differential contribution of SNARE-dependent exocytosis to inflammatory potentiation of TRPV1 in nociceptors
M. Camprubi-Robles et al.
FASEB JOURNAL (2009)
Contribution of TRPV1 to the bradykinin-evoked nociceptive behavior and excitation of cutaneous sensory neurons
Kimiaki Katanosaka et al.
NEUROSCIENCE RESEARCH (2008)
Pharmacological blockade of the vanilloid receptor TRPV1 elicits marked hyperthermia in humans
Narender R. Gavva et al.
PAIN (2008)
Meta-analysis of cannabinoid ligand binding affinity and receptor distribution: interspecies differences
J. M. McPartland et al.
BRITISH JOURNAL OF PHARMACOLOGY (2007)
The vanilloid receptor TRPV1 is tonically activated in vivo and involved in body temperature regulation
Narender R. Gavva et al.
JOURNAL OF NEUROSCIENCE (2007)
Effects of skin surface temperature on epidermal permeability barrier homeostasis
Mitsuhiro Denda et al.
JOURNAL OF INVESTIGATIVE DERMATOLOGY (2007)
TRPV1 mediates histamine-induced itching via the activation of phospholipase A2 and 12-lipoxygenase
Won-Sik Shim et al.
JOURNAL OF NEUROSCIENCE (2007)
Characterization and comparison of recombinant human and rat TRPV1 receptors: effects of exo- and endocannabinoids
PMW Lam et al.
BRITISH JOURNAL OF ANAESTHESIA (2005)
Expression and distribution of vanilloid receptor 1 (TRPV1) in the adult rat brain
A Tóth et al.
MOLECULAR BRAIN RESEARCH (2005)
Characterization of the mouse cold-menthol receptor TRPM8 and vanilloid receptor type-1 VR1 using a fluorometric imaging plate reader (FLIPR) assay
HJ Behrendt et al.
BRITISH JOURNAL OF PHARMACOLOGY (2004)
The principle of temperature-dependent gating in cold- and heat-sensitive TRP channels
T Voets et al.
NATURE (2004)
A point-charge force field for molecular mechanics simulations of proteins based on condensed-phase quantum mechanical calculations
Y Duan et al.
JOURNAL OF COMPUTATIONAL CHEMISTRY (2003)
Bradykinin lowers the threshold temperature for heat activation of vanilloid receptor 1
T Sugiura et al.
JOURNAL OF NEUROPHYSIOLOGY (2002)
Functional vanilloid receptors in cultured normal human epidermal keratinocytes
K Inoue et al.
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS (2002)