Journal
ORGANIC LETTERS
Volume 22, Issue 9, Pages 3655-3660Publisher
AMER CHEMICAL SOC
DOI: 10.1021/acs.orglett.0c01126
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Funding
- MEXT [17H06091]
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The regioselective Rh(III)-catalyzed C-H amidation of aniline derivatives with dioxazolones as an amidating reagent with a pyrimidine as a directing group leading to the production of 1,2-diaminobenzene derivatives or benzimidazole derivatives is described. The product distribution is controlled by the nature of solvent used. The reaction provides a broad substrate scope for aniline derivatives with various important functional groups including dioxazolones.
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