Journal
CHEMICAL COMMUNICATIONS
Volume 52, Issue 9, Pages 1907-1910Publisher
ROYAL SOC CHEMISTRY
DOI: 10.1039/c5cc08895j
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Funding
- NSFC [21232004, 21332005, 21272095, 21472071]
- PAPD of Jiangsu Higher Education Institutions
- Robert A. Welch Foundation (USA) [D-1361]
- NIH (USA) [R33DA031860]
- Outstanding Youth Fund of JSNU [YQ2015003]
- NSF of Jiangsu Province [BK20151163]
- Open Foundation of Jiangsu Key Laboratory [K201505]
- NATIONAL INSTITUTE ON DRUG ABUSE [R33DA031860] Funding Source: NIH RePORTER
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A new cascade three-component halosulfonylation of 1,7-enynes for efficient synthesis of densely functionalized 3,4-dihydroquinolin-2(1H)-ones has been established from readily accessible arylsulfonyl hydrazides and NIS (or NBS). The reaction pathway involves in situ-generated sulfonyl radical-triggered alpha,beta-conjugated addition/6-exo-dig cyclization/radical coupling sequence, resulting in continuous multiple bond-forming events including C-S, C-C and C-I (or C-Br) bonds to rapidly build up molecular complexity.
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