4.0 Article

Effective Inhibitors of Tyrosyl-DNA Phosphodiesterase 1 Based on Monoterpenoids as Potential Agents for Antitumor Therapy

Related references

Note: Only part of the references are listed.
Review Chemistry, Medicinal

Dual DNA topoisomerase 1 and tyrosyl-DNA phosphodiesterase 1 inhibition for improved anticancer activity

Alexandra Zakharenko et al.

MEDICINAL RESEARCH REVIEWS (2019)

Article Oncology

Novel Inhibitors of DNA Repair Enzyme TDP1 Combining Monoterpenoid and Adamantane Fragments

Evgcnii S. Mozhaitsev et al.

ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY (2019)

Article Chemistry, Medicinal

Novel tyrosyl-DNA phosphodiesterase 1 inhibitors enhance the therapeutic impact of topotecan on in vivo tumor models

A. L. Zakharenko et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2019)

Article Biochemistry & Molecular Biology

Aminoadamantanes containing monoterpene-derived fragments as potent tyrosyl-DNA phosphodiesterase 1 inhibitors

Konstantin Yu. Ponomarev et al.

BIOORGANIC CHEMISTRY (2018)

Article Biochemistry & Molecular Biology

Novel Semisynthetic Derivatives of Bile Acids as Effective Tyrosyl-DNA Phosphodiesterase 1 Inhibitors

Oksana V. Salomatina et al.

MOLECULES (2018)

Article Biochemistry & Molecular Biology

Synthesis and evaluation of aryliden- and hetarylidenfuranone derivatives of usnic acid as highly potent Tdp1 inhibitors

Olga Zakharova et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2018)

Article Biochemistry & Molecular Biology

A Novel Class of Tyrosyl-DNA Phosphodiesterase 1 Inhibitors That Contains the Octahydro-2H-chromen-4-ol Scaffold

Nikolai S. Li-Zhulanov et al.

MOLECULES (2018)

Article Chemistry, Medicinal

Achyrodimer F, a tyrosyl-DNA phosphodiesterase I inhibitor from an Australian fungus of the family Cortinariaceae

Li-Wen Tian et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2017)

Article Biochemistry & Molecular Biology

New inhibitors of tyrosyl-DNA phosphodiesterase I (Tdp 1) combining 7-hydroxycoumarin and monoterpenoid moieties

Tatyana Khomenko et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2016)

Article Plant Sciences

Tyrosyl-DNA Phosphodiesterase 1 Inhibitors: Usnic Acid Enamines Enhance the Cytotoxic Effect of Camptothecin

Alexandra Zakharenko et al.

JOURNAL OF NATURAL PRODUCTS (2016)

Article Biochemistry & Molecular Biology

Synthesis and biological evaluation of novel tyrosyl-DNA phosphodiesterase 1 inhibitors with a benzopentathiepine moiety

Alexandra Zakharenko et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2015)

Article Biochemistry & Molecular Biology

A synthesis, in silico, in vitro and in vivo study of thieno[2,3-b]pyridine anticancer analogues

Homayon J. Arabshahi et al.

MEDCHEMCOMM (2015)

Article Chemistry, Medicinal

Diamidine Compounds for Selective Inhibition of Protein Arginine Methyltransferase 1

Leilei Yan et al.

JOURNAL OF MEDICINAL CHEMISTRY (2014)

Editorial Material Chemistry, Medicinal

Tyrosyl-DNA Phosphodiesterase 1 (Tdp1) inhibitors

Shar-yin N. Huang et al.

EXPERT OPINION ON THERAPEUTIC PATENTS (2011)

Article Biochemistry & Molecular Biology

AP-site cleavage activity of tyrosyl-DNA phosphodiesterase 1

Natalia A. Lebedeva et al.

FEBS LETTERS (2011)

Article Biochemistry & Molecular Biology

Tdp1 protects against oxidative DNA damage in non-dividing fission yeast

Samia Ben Hassine et al.

EMBO JOURNAL (2009)

Software Review Chemistry, Multidisciplinary

OLEX2: a complete structure solution, refinement and analysis program

Oleg V. Dolomanov et al.

JOURNAL OF APPLIED CRYSTALLOGRAPHY (2009)

Article Chemistry, Medicinal

Empirical Scoring Functions for Advanced Protein-Ligand Docking with PLANTS

Oliver Korb et al.

JOURNAL OF CHEMICAL INFORMATION AND MODELING (2009)

Article Chemistry, Medicinal

Benchmarking the reliability of QikProp. Correlation between experimental and predicted values

Leukothea Ioakimidis et al.

QSAR & COMBINATORIAL SCIENCE (2008)

Review Oncology

Topoisomerase I inhibitors: camptothecins and beyond

Yves Pommier

NATURE REVIEWS CANCER (2006)

Article Biochemistry & Molecular Biology

General and targeted statistical potentials for protein-ligand interactions

WTM Mooij et al.

PROTEINS-STRUCTURE FUNCTION AND BIOINFORMATICS (2005)

Letter Biochemistry & Molecular Biology

Announcing the worldwide Protein Data Bank

H Berman et al.

NATURE STRUCTURAL BIOLOGY (2003)

Article Biochemistry & Molecular Biology

Improved protein-ligand docking using GOLD

ML Verdonk et al.

PROTEINS-STRUCTURE FUNCTION AND GENETICS (2003)

Article Chemistry, Multidisciplinary

The Cambridge Structural Database: a quarter of a million crystal structures and rising

FH Allen

ACTA CRYSTALLOGRAPHICA SECTION B-STRUCTURAL SCIENCE (2002)

Article Multidisciplinary Sciences

The tyrosyl-DNA phosphodiesterase Tdp1 is a member of the phospholipase D superfamily

H Interthal et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2001)

Article Biochemistry & Molecular Biology

The Protein Data Bank

HM Berman et al.

NUCLEIC ACIDS RESEARCH (2000)