Journal
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
Volume 2020, Issue 9, Pages 1141-1144Publisher
WILEY-V C H VERLAG GMBH
DOI: 10.1002/ejoc.201901858
Keywords
Carbamoylation; Quinoxalin-2(1H)-ones; C-H bond activation; Copper catalysis
Categories
Funding
- National Science Foundation of China [21572117]
- Shandong Provincial Key Research and Development Program [2019JZZY021015, 2019GHY112053]
Ask authors/readers for more resources
A direct C-H bond carbamoylation of quinoxalin-2(1H)-ones with hydrazinecarboxamides has been developed. This reaction provides a series of 3-carbamoylquinoxalin-2(1H)-one derivatives in moderate to good yields under mild conditions with a broad range of substrates and functional group tolerance. The present methodology affords a convenient and practical access to pharmaceutically active 3-carbamoylquinoxalin-2(1H)-one derivatives.
Authors
I am an author on this paper
Click your name to claim this paper and add it to your profile.
Reviews
Recommended
No Data Available