Journal
ORGANIC LETTERS
Volume 21, Issue 12, Pages 4397-4401Publisher
AMER CHEMICAL SOC
DOI: 10.1021/acs.orglett.9b00857
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Funding
- Special Account for Research Grants of NKUA [14952, 10504]
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A straightforward, late-stage diversification strategy for the installation of side chains on readily accessible unsaturated phosphinopeptidic scaffolds based on a Giese-type addition of alkyl radicals has been investigated. Among different alternatives, the preferred methodology is operationally simple as it can be carried out in an open flask with no need for protection of acidic moieties. Direct application to the synthesis of SPPS-compatible building blocks or to longer peptides is also reported.
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