4.1 Article

Identification and optimisation of 7-azaindole PAK1 inhibitors with improved potency and kinase selectivity

Related references

Note: Only part of the references are listed.
Article Chemistry, Medicinal

Back Pocket Flexibility Provides Group II p21-Activated Kinase (PAK) Selectivity for Type I 1/2 Kinase Inhibitors

Steven T. Staben et al.

JOURNAL OF MEDICINAL CHEMISTRY (2014)

Article Chemistry, Medicinal

Impact of Stereospecific Intramolecular Hydrogen Bonding on Cell Permeability and Physicochemical Properties

Bjorn Over et al.

JOURNAL OF MEDICINAL CHEMISTRY (2014)

Review Oncology

PAK signalling during the development and progression of cancer

Maria Radu et al.

NATURE REVIEWS CANCER (2014)

Article Chemistry, Medicinal

Synthesis and structure-activity relationship of 2-arylamino-4-aryl-pyrimidines as potent PAK1 inhibitors

Yong Xu et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2013)

Article Chemistry, Medicinal

Discovery, Synthesis, and Characterization of an Orally Bioavailable, Brain Penetrant Inhibitor of Mixed Lineage Kinase

Val S. Goodfellow et al.

JOURNAL OF MEDICINAL CHEMISTRY (2013)

Review Chemistry, Medicinal

p21-Activated kinase inhibitors: a patent review

James J. Crawford et al.

EXPERT OPINION ON THERAPEUTIC PATENTS (2012)

Article Chemistry, Medicinal

Protein-Ligand Crystal Structures Can Guide the Design of Selective Inhibitors of the FGFR Tyrosine Kinase

Richard A. Norman et al.

JOURNAL OF MEDICINAL CHEMISTRY (2012)

Article Chemistry, Medicinal

Discovery of Pyrroloaminopyrazoles as Novel PAK Inhibitors

Chuangxing Guo et al.

JOURNAL OF MEDICINAL CHEMISTRY (2012)

Review Biotechnology & Applied Microbiology

Vemurafenib: the first drug approved for BRAF-mutant cancer

Gideon Bollag et al.

NATURE REVIEWS DRUG DISCOVERY (2012)

Article Multidisciplinary Sciences

Targeting p21-activated kinase 1 (PAK1) to induce apoptosis of tumor cells

Christy C. Ong et al.

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2011)

Article Chemistry, Medicinal

Analysis of Kinase Inhibitor Selectivity using a Thermodynamics-Based Partition Index

Alan C. Cheng et al.

JOURNAL OF MEDICINAL CHEMISTRY (2010)

Article Chemistry, Medicinal

Gini coefficient: A new way to express selectivity of kinase inhibitors against a family of kinases

Piotr P. Graczyk

JOURNAL OF MEDICINAL CHEMISTRY (2007)

Review Oncology

p21-activated kinases in cancer

Rakesh Kumar et al.

NATURE REVIEWS CANCER (2006)