Journal
TETRAHEDRON LETTERS
Volume 55, Issue 15, Pages 2430-2433Publisher
PERGAMON-ELSEVIER SCIENCE LTD
DOI: 10.1016/j.tetlet.2014.02.115
Keywords
alpha-Enolicdithioesters; Diazotization; Cascade annulation; 1,2,3-Thiadiazoles; One-pot
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Funding
- Science and Engineering Research Board [SB/S1/OC-30/2013]
- Council of Scientific and Industrial Research, New Delhi, India [02(0072)/12/EMR-II]
- CSIR, New Delhi
- DAAD
- George-August-Universitat-Gottingen
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An operationally simple, economical, and straightforward synthesis of diverse 4,5-disubstituted 1,2,3-thiadiazoles from alpha-enolicdithioesters has been achieved via nitrosation/reduction/diazotization/cyclization sequence in one-pot through the formation of cascade 1-2 (N-S) and 3-4 (C-N) bonds. Importantly, this is the first straightforward entry to highly functionalized 1,2,3-thiadiazoles from dithioesters. (C) 2014 Elsevier Ltd. All rights reserved.
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