4.4 Article

Pd-catalyzed addition of boronic acids to vinylogous imines: a convenient approach to 3-sec-alkyl substituted indoles

Journal

TETRAHEDRON LETTERS
Volume 53, Issue 30, Pages 3873-3875

Publisher

PERGAMON-ELSEVIER SCIENCE LTD
DOI: 10.1016/j.tetlet.2012.05.056

Keywords

Palladium; Conjugate addition; Sulfonylindoles; Vinylogous imines; Boronic acids

Funding

  1. National Natural Science Foundation of China [20502005, J0830415]
  2. Department of Science and Technology Foundation of Hunan Province [2010GK3157]
  3. Hunan Nature Science Foundation [09JJ6024]

Ask authors/readers for more resources

A convenient approach to 3-sec-alkyl substituted indoles was developed via palladium-catalyzed addition of arylboronic acids to vinylogous imines generated in situ from sulfonylindoles under mild conditions. (C) 2012 Elsevier Ltd. All rights reserved.

Authors

I am an author on this paper
Click your name to claim this paper and add it to your profile.

Reviews

Primary Rating

4.4
Not enough ratings

Secondary Ratings

Novelty
-
Significance
-
Scientific rigor
-
Rate this paper

Recommended

No Data Available
No Data Available