Journal
TETRAHEDRON
Volume 69, Issue 24, Pages 4944-4952Publisher
PERGAMON-ELSEVIER SCIENCE LTD
DOI: 10.1016/j.tet.2013.04.032
Keywords
Amino amide; Alcoholysis; Four-component condensation; Peptide; Phosphinodepsipeptide
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Funding
- National Basic Research Program of China [2013CB328900]
- National Natural Science Foundation of China [20972013]
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Phosphinodepsipeptides are recognized as an important class of enzyme inhibitors as tetrahedrally structural transition-state analogues to natural peptides. A series of phosphinodepsipeptides was synthesized in satisfactory yields via pseudo-four-component condensation reaction of 2-(N-benzoxycarbonylamino)alkanamides/peptide amides, aldehydes, and aryldichlorophosphines, followed by alcoholysis with hydroxyl esters. (C) 2013 Elsevier Ltd. All rights reserved.
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