Journal
TETRAHEDRON
Volume 67, Issue 24, Pages 4327-4332Publisher
PERGAMON-ELSEVIER SCIENCE LTD
DOI: 10.1016/j.tet.2011.02.067
Keywords
Annulation; Alkylation; Indole; Communesin; Alcohol
Categories
Funding
- Dartmouth College
- Walter and Constance Burke Foundation
Ask authors/readers for more resources
An efficient method for the annulation of indoles with 2-aminobenzyl alcohols, catalyzed by TFA, to furnish 5,6-fused indoline aminals is reported. This method can be extended to the alkylation of indoles at C3. 2-Aminobenzyl alcohols are used directly without recourse to protection of the aniline nitrogen or activation of the alcohol. (C) 2011 Elsevier Ltd. All rights reserved.
Authors
I am an author on this paper
Click your name to claim this paper and add it to your profile.
Reviews
Recommended
No Data Available
Share Paper
