Journal
SYNLETT
Volume 24, Issue 11, Pages 1448-1454Publisher
GEORG THIEME VERLAG KG
DOI: 10.1055/s-0033-1338703
Keywords
amination; phenols; metal-free; arylamines; carbazoles
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Funding
- National Natural Science Foundation of China [31071720]
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Herein, we disclose the metal-free synthesis of arylamines via the direct amination of phenols using aminating reagents. This reaction procedure uses easy accessible aminating reagents and provides a versatile synthetic route to a broad range of arylamines with various functionalities in good to excellent yield. By using a two-step route of amination and oxidative coupling reaction, we synthesized three naturally occurring carbazole alkaloids: murrayafoline A, mukonine, and clausenine from two commercially available phenols.
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