Journal
SYNLETT
Volume -, Issue 14, Pages 2089-2092Publisher
GEORG THIEME VERLAG KG
DOI: 10.1055/s-2008-1078019
Keywords
click chemistry; aromatic azides; Huisgen cycloaddition; chemoselectivity; 1,4-triazoles
Categories
Funding
- EPSRC
- The University of Nottingham
Ask authors/readers for more resources
The practical and efficient one-pot azidation of anilines with the reagent combination t-BuONO and TMSN3 has become a useful addition to the click-chemistry toolbox. Herein we report a modification of this methodology, using microwave radiation to significantly enhance the rate of fori-nation of 1,4-triazoles from in situ generated azides.
Authors
I am an author on this paper
Click your name to claim this paper and add it to your profile.
Reviews
Recommended
No Data Available
Share Paper
