Journal
CHEMICAL SCIENCE
Volume 6, Issue 2, Pages 987-992Publisher
ROYAL SOC CHEMISTRY
DOI: 10.1039/c4sc02365j
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Funding
- Deutsche Forschungsgemeinschaft [GRK 1626]
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Benzoyl azides were used for the direct and atom economic C-H amidation of electron rich heteroarenes in the presence of phosphoric acid, a photocatalyst and visible light. Hetero-aromatic amides are obtained in good yields at very mild reaction conditions with dinitrogen as the only by-product. The reaction allows the use of aryl-, heteroaryl- or alkenyl acyl azides and has a wide scope for heteroarenes, including pyrroles, indole, furan, benzofuran and thiophene giving good regio-selectivities and yields.
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