Journal
ORGANIC LETTERS
Volume 16, Issue 4, Pages 1228-1231Publisher
AMER CHEMICAL SOC
DOI: 10.1021/ol5001507
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Funding
- MEXT
- JSPS, Japan
- Uehara Memorial Foundation
- Grants-in-Aid for Scientific Research [25620084] Funding Source: KAKEN
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A Cu-catalyzed aminoboration of 1-methylenecyclopropanes with bis(pinacolato)diboron and O-benzoyl-N,N-dialkylhydroxylamines has been developed. The Cu catalysis provides a rapid and concise access to (borylmethyl)cyclopropylamines in a highly regio- and diastereoselective manner. The products obtained can be useful building blocks for the synthesis of potential antidepressants, trans-2-arylcyclopropylamine derivatives.
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