Journal
ORGANIC LETTERS
Volume 15, Issue 20, Pages 5294-5297Publisher
AMER CHEMICAL SOC
DOI: 10.1021/ol402523x
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Funding
- Shenzhen municipality [JC201104210112A, GJHZ20120614144733420, KQTD201103]
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A general protocol for the synthesis of N-alkyl indoles has been developed via a redox neutral C-H activation strategy using a traceless nitroso directing group. A broad scope of substituted N-alkyl indoles has been prepared in good to excellent yields using a very simple Rh catalyst system in the absence of an external oxidant or any other additive. Good to excellent regioselectivity has been achieved for asymmetrically disubstituted acetylenes.
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