Journal
ORGANIC LETTERS
Volume 15, Issue 4, Pages 788-791Publisher
AMER CHEMICAL SOC
DOI: 10.1021/ol303440y
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Funding
- NSFC [91021004]
- National Basic Research Program of China [2011CB921402]
- Key Project of Science and Technology of the Department of Education, Anhui Province, China [KJ2010ZD05]
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An efficient palladium-catalyzed synthesis of 3-acylindoles using free (N-H) indoles and nitrites has been developed. The acylation reaction proceeded well under the Pd(OAc)(2)/2,2'-bipyridine system and with D-(+)-camphorsulfonic acid as the additive. A possible mechanism involving carbopalladation of nitrites and subsequent hydrolysis of ketimines Is proposed.
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