4.8 Article

Palladium(0)-Catalyzed Dearomative Arylation of Indoles: Convenient Access to Spiroindolenine Derivatives

Journal

ORGANIC LETTERS
Volume 14, Issue 14, Pages 3772-3775

Publisher

AMER CHEMICAL SOC
DOI: 10.1021/ol301663h

Keywords

-

Funding

  1. National Basic Research Program of China (973 Program) [2009CB825300]
  2. National Natural Science Foundation of China [20923005, 20932008, 21025209, 21121062]

Ask authors/readers for more resources

Dearomatization of an indole via palladium(0)-catalyzed cross-coupling reaction has been realized. With readily available triphenylphosphine as ligand, various spiroindolenine derivatives have been obtained in good to excellent yields, and enantioselective control is also feasible with chiral ligands.

Authors

I am an author on this paper
Click your name to claim this paper and add it to your profile.

Reviews

Primary Rating

4.8
Not enough ratings

Secondary Ratings

Novelty
-
Significance
-
Scientific rigor
-
Rate this paper

Recommended

No Data Available
No Data Available